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INHIBIT

CLASIFICATION

Penicillins

Cel
l
Wal
l
S
y
n
t
h
e
s
i
s

Beta
Lacta
ms
Cephalosporins

Carbapenems

No
lacta
m

Monobactams
Beta-lactamase
inhib.
Glycopeptides

DNA
topoisomer

Vancomycin
Teicoplanin

Bacitracin
Polymyxin B

AminoGentamycin
Neomycin
Streptomycin
Amikacin
Tobramycin
glycosides
Tetracyclin
Doxycycline
Demeclocylin *
Minocycline
Tetracyclin
Tigecyclin
s
Oxazolidon
Linezolid
ones
50 Streptogra
Quinupristin/Dalfopristin
S
mins
Cloramphenicol
Macrolides
Erythromycin
Azithromycin
Clarithromycin
Lincosamid
Clindamycin
Lincomycin
es
Fluorquinolones Ciprofloxacin
Norfloxacin
Levofloxacin
Ofloxacin
Sparfloxacin
Moxifloxacin
Gemifloxacin Enofloxaci
n
30
S

Protein
Synthesis

ANTIBIOTICS
Penicinillase Sensible
Natural
Penicillin G: Na, K, Procainic, Benzathine
Penicillins
(IV, IM)
(narrow spectrum)
Penicillin V: VO
Aminopenicillins Ampicillin
(broad spectrum)
Amoxicillin
Penicinillase Resistant (very narrow spectrum)
Nafcillin
Oxacillin
Dicloxacillin
Antipseudomonal (extended spectrum)
Ticarcillin
Carboxipenicillin Carbenicillin
s
Piperacillin
Ureidopenicillins Azlocillin
Mezlocillin
1 Generation
Cefazolin
Cephalexine
Cephapirin
Cefadroxil
Cephadrine
Cephalotin
Cefuroxime Cefamandole Cefprozil
Cefoxitin
Cefonicid
Cefmetazo
2 Generation
le
Cefotetan
Cefaclor
Cefoperazo Ceftriaxone
Ceftazidim
3 Generation
ne
e
Cefpodoxim Ceftizoxime
Cefotaxim
e
e
Cefdinir
Ceftibuten
Cefixime
Cefditoren
4 Generation
Cefepime
Cefpirome *
5 Generation
Ceftaroline
Meropenem
Ertapene
Doripene
Imipenem +
m
m
Cylastatine
Aztreonam
Sulbactam
Tazobactam
Clavulanic Acid

ases
Folic Acid
Synthesis
DNA
(damage)
mRNA
synth.

Quinolones
Sulfonamides
DHFR inhibitors
Metronidazole
Rifampim

Nalidixic Acid
Sulfamethoxazole
Ag
(SMX)
Sulfadiazine
Trimethroprim (TMP)

Sulfasalazi Sulfisoxaz
ne
ole
Pirymethamine

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