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1.

Pemicu sekresi insulin/insulin secretagogue: Sulfonylurea

2.

Glinid Penambah sensitifitas insulin: Metformin, Tiazolidindion

3.

Penghambat glukoneogenesis: Metformin

4.

Penghambat absorpsi glukosa: penghambat Glukosidase alfa, acarbose

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