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File2 916 1352573
File2 916 1352573
File2 916 1352573
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First Generation Antipsychotic Medications
Second Generation Antipsychotic Medications
dopamine2 (D2)
High Potency : haloperidol
Haldol D2
Low Potency :
chlorpromazine Morefine
H1
M1
D2
Positive symptoms
Mesocortical pathway
Negative symtoms
Nigrostriatal pathway
EPS
Tuberoinfundibular pathways
Prolactin
Extrapyramidal Symptoms
Anticholinergic Effects
Antiadrenergic Effects
Antihistamine Effects
Neuroleptic
Malignant Syndrome
Acute dystonia
Akathisia
Parkinsonism
Tardive dyskinesia
Dry mouth
Blurred vision
Constipation
Urinary retention
Postural
hypotension
Neuroleptic Malignant Syndrome
39-41 WBC
12000
CK,CPK,K,GOT,GPT
Haldol ( Binin-U ):
5mg, 50mg
5HT2A
SDA
D2
MARTA
Serotonin-Dopamine Antagonism
Risperidone (Risperdal)
Consta 25 37.5
Ziprasidone (Geodon)
Abilify
Solian
Clozapine (Clozaril)
Olanzapine (Zyprexa)
,10mg
Quetiapine (Seroquel)
Zotepine (Lodopin)
EPS Risperdial
:Olanzapine, Seroquel
Solian
QTc prolongation
Cloazpine
Cloazpine, Olanzapine
Cloazpine
Cloazpine,Lodpine
Geoden, Cloazpine,
Olanzapine, Seroquel,
Clozapine olanzapine risperidone
First Generation Antipsychotic Medications
Second Generation Antipsychotic Medications
Carbamazepine Tegretal
Valproate Depakine, Convulex
Benzodiazepine BZD, Rivtoril
Inderal
3050
0.6-1.2meq/dl
1.5-2.0meq/dl
2.0-4.0meq/dl
EKG
4.0meq/dl
Carbamazepine
Tegretal
Steven-
Johsons syndrom
Lamictal
Stevens - Johnson
Steven-Johsons syndrom
macrolide or
doxycycline .
Valproate
Depakine, Convulex
Carbamazepine
First Generation Antipsychotic Medications
Second Generation Antipsychotic Medications
Benzodiapine BZD
Xanax Gendergine , Rivotril, Ative, Lexoten,
Librium, Erispam, Valium, serenal ,
Alpraline
Buspirone Buspar
BZD
hypnotics
BZD:
Dalmadorm * cap 15 mg
Stilnox:
Eszo:
Imovan, Genclone:
First Generation Antipsychotic Medications
Second Generation Antipsychotic Medications
-CPY450
TCA
MAOI
SSRI
2A SARI)
SNRI
NRI
(NDRI)
SDRI
NaSSA
TCA
Tofranil
MAOI
tryamine
SARI
Trazodone, Cirzodone Mesyrel ,
150-400 150-600
SSRI
Prozac Zactin Fluoxetine , Cipram
SNRI
Effexor
75-225
20-30mmHg
2-3
Ixel
MAOI digoxin clonidin
NRI
Reboxetine( Edronax, Vestra):
Atomoxetine ( Strattera):
NDRI
Bupropion
100mg,bid.
2-4
Wellbutrin SR
Bupropion
NaSSA
Remeron ( Mirtazapine )
30mg
SSRI Effexor
SGPT
First Generation Antipsychotic Medications
Second Generation Antipsychotic Medications
Artane
Bipiden
Akenton
Inderal
PK-merz FC