Enzyme Inducers & Inhibitors

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P450 isoform

CYP1A2

CYP2C9

CYP2C19

CYP2D6

CYP2E1
CYP3A4

Inducer
Omeprazole
Lansoprazole
Phenytoin
Tobacco smoke
Barbiturates
Rifampicin
Carbamazepine
Rifampicin
Omeprazole
Dexamethasone
Rifampicin

Alcohol (chronic)
Isoniazid
Carbamazepine
Phenytoin
Barbiturates
Dexamethasone
Primidone
Rifampicin
St. Johns Wort
Bosentan
Efavirenz
Nevirapine

Inhibitor
Amiodarone
Cimetidine
Fluoroquinolones
Fluvoxamine
Amiodarone
Azole antifungals
Isoniazid
Cimetidine
Fluoxetine
Tranylcypromine
Amiodarone
Bupropion
Cordarone
Duloxetine
Fluoxetine
Paroxetine
Ritonavir
Sertraline
Disulfram
Cimetidine
Clarithromycin
Erythromycin
Itraconazole
Ketoconazole
Grapefruit Juice
Aprepitant
Diltiazem
Protease Inhibitor
Imatinib
Verapamil

I can do all things through Christ who strengthens


me. Phil. 4:13

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