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Antibacterials Lecture Notes For Blues
Antibacterials Lecture Notes For Blues
1. Penicillins
2. Cephalosporins
3. Vancomycin
1. Lincosamides
2. Tetracyclines
3. Aminoglycosides
1. Ketolides
Bactericidal Bacteriostatic
1. Vancomycin 1. Tetracyclines
2. Cephalosporins 2. Glycylcyclines
3. Aminoglycosides 3. Sulfonamides
4. Fluoroquinolones
1. Penicillins
2. Macrolides
3. Lincosamides
4. Ketolides
5. Metronidazole
1. Penicillins – Ex. Amoxicillin, Ampicillin, Co – Amoxiclav and
Cloxacillin ( Penicillinase resistant antibiotics )
- With meals
- Hepatotoxic
- No IM route
4. Lincosamides – Ex. Clindamycin and Lincomycin
5. Vancomycin
- Ototoxic
- Photosensitivity
- 1 hour before and 2 hours after meals with a full glass of water
- MIO, nephrotoxic
- Before meals
A. Rifampicin
- Hepatotoxic
- Empty stomach
B. Isoniazid INH
- Hepatotoxic
- Agranulocytosis
- No alcohol ingestion
C. Pyrazinamide PZA
- Hepatotoxic
D. Ethambutol
Fungus
- Cellular organism with a hard cell wall that contains chitin and
polysaccharides and a cell membrane that contains ergosterol
Mycosis
Azoles - Fluconazole
2. Azoles – Ketoconazole
3. Antimetabolites – Flucytosine
4. Echinocandins – Caspofungin
Side effects
1. Local ( cream, lotion, spray )
2. Suppository or troche
3. Vaginal suppository
Helminths
Anthelmintics
1. Mebendazole
2. Pyrantel pamoate
3. Albendazole