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SEDATIVE-HYPNOTIC DRUGS

Benzodlazep1nes Non-benzodlazeplnes Other CNS


Zopiclonc depressants
Eszopiclone Chloral hydrate
Zolpidem Triclophus
Hypnotic Antlanxlety Antlconvulsant
Zaleplon Paraldehyde
Diazepam Diazepam Diazepam Glutclhin,ide
Flurazcpam 01lun.Jia1.cpoxidc Lorazepan1 Mclhaqualonc
Nitrazepam Oxazepam Clonazepam tvteprobamntc
AJprazolam Lorazepam Clobazam Pmmethazine
Tcmazepam Alprazolam Chlorproma7ine
. Amitrlptyline
Triazolam
Barbiturates Morphine

Long acting Short acting Ultra-short acting


Phenoba rbi tone Butobarbitone Thiopentone
Pentobarbilone Mclhohcxilone
ANTIEPILEPTIC DRUGS

Barbiturate Hydantoin Succlnlmlde Benzodlazeplnes Newer drugs


Phcnobarbitonc Phcnytoin Ethosuximidc Clonazcpan1 Topiramatc
Fosphenytoin Diazepam Zonisa1nide
.
Lorazepam Levetiracetam
lctobazam Vigabatrin
Tiagabine
Lacosamide
Oeoxybarblturate lmlnostllbene Aliphatic
Primidone Carbamazepine carboxyllc acid
Phenyltrlazlne Cyclic GABA
Oxcarbazepine Valproate sod analogues
(Valproic acid) Lamotrigine
Gaba pentin
Divalprocx Pregabalin
1
AN l lPARKINSONIAN DRUGS

Drugs affecting brain Drugs effecting brain


dopam1nerg1c system cholinerglc system

Dopamine Dopamlnergic COMT Central Antlhistaminlcs


precursor agonists Inhibitors antlchollnerglcs
Levodopa Bromocriptinc Entncaponc Trihexyphenidyl Orphcnadrinc
Ropinirolc Tolcaponc Procyclidine Promethazine
Pramipcxolc Biperiden

Peripheral MAO-B Glutamate (NMDA receptor)


decarboxylase Inhibitors agonist (Dopamine facilitator)
Inhibitors Selegiline Amantadine
Carbidopa Rasagiline
Benserazlde
ANTIPSYCHOTIC DRUGS
(Neuroleptic drugs)

Phenothlazines Thloxanthlne Atypical


Rupenthixol an tipsyeholies
Clozapine
Aliphatic Piperldine Plperazlne Risperidone
Other he1erocyctic
side chain side chain Olanz.apine
side chain compounds
Quetiapine
Chlorpromazint' Thioridazine Trifluoperazine Pimozide Aripiprazole
Tri'1upro1nazine Fluphena1.ine Loxnpine Ziprasidonc
Amisulpiride
Butyrophenones Zotepine
Haloperidol
TriAupcridol
Penfluridol
DRUGS FOR MANIA AND BIPOLAR DISORDER

Lithium An1fconvulsants Atypical


carbonate anti psychotics
Sodium valproah?
Carbamazepine Olanzapine
l..amotrig ine Risperidnne
Queliap ine
Aripiprazo.le
HALLUCINOGENS
(Psychotomimetics, Psychedelics, Psychody sleptics)

lndole alkylamlnes Phenylalkylamlnes Arylcyclohexyl- Cannabinolds


Lysergic acid Nlesca line amine Tetra hydro-
diethylr1mide (LSD) Ecstasy Phcncyclidine cannabino l ('.1 THC)
Lyscrgic acid amide (t.ilcthylinc dioxy-
Psilocybin n1cth.:unphetan1inc)
Ha rmine YABA
Dimethy l tryptan1inc (Mcthan1pheta111.ine
+ methylhexanantlne)

www.carnbodiarned.com
OPIOID ANALGESICS AND ANTAGONISTS

Opioid Ll receptor ogon1sts Complex action op101ds Pure opioid


antagonists

Natural opl111m Semlsynthetlc Synthetic Agonlst-antagonlsts NaJo xone


alkaloids 0DI0lds 0Dlolds (K anal eslcs) Naltrexone
Morphine Oiacctyln1orphinc Pethidine Nnlorplllinc Nairn ~fene
Codeine (Heroin} (Mcperidine) Pentazocine
Pholcodinc Methadone Butorphanol
Ethylmorphine Fentanyl
Dextro- Partial µ agonlst +
propo~yphene K antaaonlst
Tramadol
Buprenorphine
Atypical
~

Aeversible inhlbltoJS ~ Sele ctive sero t,o nln


ol MAO -A (RIMAs) r aupt ake lnhl bltor,s cssRia)
1 1

C
antidepressants
fwloclobemide Fluox cline Traiz odon,e
Clo,r gylin e f luvox amin e Mian serin
~

Par,o,xeline Mirl azap ine


I
~rtri llinc Bupm pion
C itnlop ram Tian e'p line
EscHalopram Amin eptin e
~ Dapu );elin ~ AtO'fflOXCtinl?1
I

Trlcy cllc antid epre ssan ts (TCA st


Sera loni1n and noradrenaline
j
rauptaka Inhibitors fSNRls)
'I I
NA + >HT reuptake Predornlnantly NA Pn k1 f,,x inc
\ 1
, Inhibitors reuptake Inhibitors II Dulo~etine
convu1san1s [Ana1ept_
1c_ __. \ P s y c fi o s tl m u la n ts
,
1

S tr y c h n in e D o x a p ra m A m p h e ta m in e s A r m o d a fi n il
P ic ru to x in l\f\ c \l "l y \ p \, ~11\._\a tc
B ic u cu ll in e
P 't !m o \i n e
A l(1m o x .e ti 1 ,e C o c a in e
Pen l)·len et e lr a z o le
1

M o d a li n il C a f f e in e

COGNITION E N H A N
CERS
(C e re b ra a c ll v e d ru
'
gs)
- -

Cholinergic
activators G lu ta m a te (NMDA) I
. M ls c e ll a n e o u s d rl u
Riva s ti g m in e " a n ta g o n is t gs l
~ile n ,a n li n e· - - - - , P ir..,c ~ t.,m
Do,ncpczil J i. Citict...,\inc
Galan ta mine Pyriti'nol Piribedil
T a c ri n e r ·yrilhioxi,~e)
- D1\1ydroer@,('\,1xine
G in k g o b i\ob a
(C o d e rg o c ri n e )
ANTIHYPERTENSIVE DRUGS (1)

Diuretics Renln-anglotensin Sympathetic


system lnhlbttors Inhibitors

!Zldes High celling Pot sparing


p-adrenerglc a +P
lrochJorothiazide I furoscmide Spironolactone blockers adrenerglc
:>rthalidone (olhers) 1Eplerenone / PropranoJol blockers
1pamide I I AntiJoride Meloprolol Labrtalol
'
IAt<.'nolol Carvedilol
(olhcrs)

ACE Inhibitors Anglotensln (AT,) Direct renln


receptor blockers Inhibitor a-adrenerglc Central
Caplopril
EnalapriJ Losartan Aliskiren blockers sympalhol
Lisinopril Candesartan Prazot-in Clonidinc
PerinJopril Vals.irtan Terazosi.n Methyldop,
R.imipril Tclmisorl:iln Doxazosin
Frn,inopril lrbcsart,1n l'hentolaminc
Quinapril Olm<.--sartan Phl•noxybcnz.1mine Contd..
Trando:l.ipril www.cambodlamed.com
ANTIHVPERTENSIVE DRUGS (2)

Calcium channel blockers Vasodilators

Phenyl- Benzothiazepine Dlhydropyrldlnes Arteriolar dilator Arteriolar +


alkylamine Diltiazcm Nifcdipine Hydralnzine venodllator

Verapamil Felodipine Minoxidil Nitr~russide
Amlodipine D.iazoxide sod.
Nitrendipine
Lacidipine
Lercanidipine
Benidipine
ANTIANGINAL DRUGS

Nitrates I
!\-blockers Calcium channel Pot channel Other
blockers opener enUanginal
drugs

1
Short acting Long acting Propranolol Vcrapamil Nicorandil Trimetazidine
Clyccryl trinitratc lsosorbide ~lcloprolol I Diltiazcm Ranolazinc
lsosorbide dinitrate Atenolnl Amlodipine lvabradine
dinitrate (oral) (others) I Nitrendipine Oxyphedrinc
(sublingual) lsosorbide ----- (others) Dipyridamole
mononitrate
Erythritol
tetranitratC!
Pentaerythritol
tetra nitrate
DRUGS FOR PERIPHERAL VASCULAR DISEASES

Rheological Phosphodlesterase-3 Antlplatelet Antioxidants


agent Inhibitor druas Vitamin E
Pentoxiphylline 1Cilostazol Aspirin
(Oxpen tifyllinc) Clopidogrcl
Ticlopidine

Vasodilators
I
Direct acting ~-adrenergic u-adrenerglc Calcium channel
Cyclandclate aaonlsts blockers blockers
Xanthinol Prazosin
.
[rr~iacycl 1n
J Isoxsuprine NiJedipine
nicotinate Phcnoxybcnzamine Nitrcndipine (PG~
'
DRUGS FOR CONGESTIVE HEART FAILURE

lnotroplc drugs Diuretics Aldosterone


antagonists

Cardiac Sympathc,. PDE3 High celling Thlazlde like


Spirono lactone
glycosldes mlmellcs Inhibitors
Digoxin Dob u tan,ine lnilmrino1ne
IFu rose mide Hvdrochloro-
,
Eplerenone
J
Bumclilnidc lhi.tzidc
Ouabain Dopamine Milrinonc Mc tolazonc t 1-edrenerg1c
Xipamidc block-e n;
Ren1n-ang1otens1n Inhibitors
Vasodllators I 1\lletuprolul
Bboprolnl
I I Nebivolol
ACE inhibitors Anglotensln AT 1 Venodllators Arteriolar + ' C11rvcdilol
r tor blockers venodilator
Enalapril Gi yceryl-
Ramipril Los.,rt.in trlnitrate Sod.
(others) Candesartilll lsosorbide- n1troprussidc
I(others) J initrate

Arteriolar dilator
PDE: Phosphodiestcrusc: ACE: Angiotcnsin con,·crting cnzymc Hydra lazine
HAEMATINICS

Iron Maturation factors Adjuvant


Vitnmin 8 12: haematinlcs
Cyan ocobalamin Copper
Oral iron Parenteral iron Hydroxocobalamin Pyridoxine
Ferrous sulfate lron-dextran Methylcobalamin Riboflavin
Ferrous fumara te Folic acid:
lron-sorbitol-
Ferrous gluconate Folinic acid
citric acid
Ferrous succinate Ferrous s ucrose (leucovorin,
Ferrous a minoatc Ferric carboxy- citrovorum factor)
Ferric a n,n,oniun, maltose
citrate
Ferric hydrox-y
polymaltose
Carbonyl iron
Iron-cal. complex
DIURETICS

High celling Medium efficacy Weak/adjunctive


diuretics

Furose,nide
(fnasen,ide) Benzothladlazlnes Thlazlde-llke Carbonic Osmotic
Bumetanide Hyd rochloroth iaz ide Chlorthalidonc anhydrase diuretic
Tora!>Cmidc H yd roflumethiclZ ide tvle tolazone Inhibitor
Mannitol
Benzthiazidc Xlpamide Acelazol,,n,ide lsosorbidc
I

lndapamidc I Glycerol
ANTI0IURETICS Oopamide '

Potassium sparing
diuretics
I 1
Antldluretlc hormone Natrluretlcs Mlscellaneous
and Its analogues
Thia:r.idl'S Carbamazepinc
Vasoprl>s..,;in Aldosterone Renal eplthellal Na+
Amiloride Chlorpropam idc antagonists
Dc:-moprc~~in channel Inhibitors
lndomcth,,cin
LyprL$.,;i n Spironolaclone Anliloridc
I Tcrliprcssin
www.cambodiamed.com
Eplerenone Triamterene
ANTIARRHYTHMIC DRUGS

Class I Class IV
Membrane stabiltz1ng agents Calcium channel
blockers

(A) (B) (C) Verapamil


Moderately decrease Diltiazcn,
Little decrease In Marked decrease In
dv/dt of Ophase dv/dt of Ophase dv/dt of Ophase
Class Ill
Quini<lin~ Lidocaine Propafenone Agents widening
Procainamide f\1exlletine Flecainide action potential
Disopyramide
Class II
Amiodarone
Antladrenerglc Drnnedaronc
agents
Drugs for Dofetilide
PSVT lbutilidc
Propranolol
Adenosine Sota lol (class 111
Dlgoxin property as well)
Esrnolol
PSVT: Poroxysmal suprnvcntricular tachycardia
ANTICOAGU LANTS

Parenteral anticoagulants Oral anticoagulants

Indirect thrombln Direct Coumarln Direct factor Oral direct


Inhibitors thrombln derivatives xa Inhibitor thrombln Inhibitor
Inhibitors Bishydroxycoun,arin
Ht'parin (unfractionated) Rivaroxaban Dabigatran-
Lo\v molecular \veight Lcpirudin (dicumarol) clcxilale
heparins Bivalirudin Warfarin sod.
(Enoxaparin, Reviparin, Argatroban Acenocoumarol In vitro anticoagulants
Nadroparin, Dalleparin, (Nicoumalonc)
Heparin
Pilmaparin, Ardcpilrin) Ethyl-biscoum•
Sou. edetat~
fondaparinux acelate
Sod. citrate
I Danaparoid Sod. oxalate

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