Classification of Drugs

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ANS

Cholinomimetics
Drug Type Sub Type
1. Acetylcholine Direct Acting Muscarinic Choline esters
2. Bethanechol
3. Carbachol
4. Methacholine

5. Muscarine Direct Acting Muscarinic Agonist


6. Pilocarpine
7. Nicotine Direct Acting Nicotine Agonist

8. Edrophonium Indirect Acting Alcohol


Short Acting
9. Neostigmine Indirect Acting Carbamates
10. Physostigmine Intermediate Acting
11. Pyrisdotigmine
12. Echothiophate Indirect Acting Organophosphates
13. Parathion/Malathion Long Acting
14. Sarin
Sympathomimetics
15. Dobutamine Direct Acting Catecholamines
16. Dopamine
17. Epinephrine
18. Isoproterenol
19. Norepinepheine

20. Phenylephrine Non-catecholamine D1 D2 Agonist


21. Albuterol Non-catecholamine β2 Agonist
22. Formetrol
23. Indacaterol
24. Metaproterenol
25. Salmetrol
26. Terbutaline

27. Amphetamine Indirect Acting Phenylisopropylamine


28. Ephedrine
29. Methamphetamine
30. Cocaine Catecholamine releasing agent.
31. Tyramine
Adrenoceptor Blockers
Drug Type Sub type
32. Phentolamin Non-selective α blocker α blocker
33. Phenoxybenzamine
34. Daxasosin Selective α blocker α1 blocker
35. Prazosin
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36. Tamsulosin
37. Terazosin

38. Yohimbine Selective α Blocker α2 blocker


39. Betaxolol Non- Selective β Blocker β Blocker
40. Nadolol Pindolol
41. Propranolol
42. Timolol

43. Atenolol Selective β Blocker β1 Blocker


44. Esmolol
45. Metoprolol
46. Nebivolol
47. Butoxamine Selective β Blocker β2 Blocker
48. Carvedilol Both α & β Blocker α+ β Blocker
49. Labetalol
Cholinoceptor Blockers and Cholinesterase regenerators
Drug Type Sub Type
50. Aclidinium Non-Selective Antimuscarinic Antimuscarinic
51. Atropine
52. Benztropine
53. Cycophentolate
54. Dicyclomine
55. Glycopyrolate
56. Homatropine
57. Ipratopium
58. Oxybutynin
59. Scopolamine
60. Tiotropium
61. Tropicamide

62. Darifenacin Selective Antimuscarinic Antimuscarinic


63. Fesoterodine
64. Pirenzepine
65. Solifenacin
66. Telenzepine
67. Tolterodine
68. Hexamethonium Ganglion Blocker Antinicotinic Ganglion
69. Mecamylamine Blocker
70. Pralidoxine
71. Trimethaphan

CNS
Sedative hypnotics
Drug Type
1. Alprazolam Benzodiazepines
2. Chlordiazepoxide

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3. Clonazapam
4. Clorazepate
5. Diazepam
6. Flurazepam
7. Lorazepam
8. Midazolam
9. Flumezenil Benzodiazepines Antagonist
10. Butabarbital Barbiturates
11. Pentobarbital
12. Phenobarbital
13. Secobarbital
14. Thiopental
15. Zaleplon Newer Drugs
16. Zolpidem
17. Busprione 5-HT Agonist
Alcohols
18. Ethanol Alcohol
19. Ethylene Glycol
20. Methanol
Antiseizure Drugs
21. Ethosuximide Cyclic Ureides
22. Phenytion
23. Phenobarbital
24. Carbamazepine Tricycle
25. Clonazepam Benzodiazepines
26. Diazepam
27. Gabapentin GABA Derivatives
28. Pregabalin
29. Vigabatrin
30. Lamotrigine Miscellaneous
31. Levetiracetam
32. Tiagabine
33. Topiramate
34. Valproate
35. Zonisamide
General Anesthetics
Drug Type Sub Type
36. Desflurane Inhaled Anesthetics Inhaled Anesthetics
37. Enflurane
38. Halothane
39. Isoflurane
40. Nitrous Oxide
41. Methohexital IV Anesthetic Barbiturates
42. Thiopental
43. Midazolam IV Anesthetic Benzodiazepines
44. Ketamine IV Anesthetic Dissociative
45. Etomidate IV Anesthetic Imidazole
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46. Fentanyl IV Anesthetic Opioids
47. Morphine
48. Propofol IV Anesthetic Phenols
Local Anesthesia
49. Bupivacaine Amides
50. Lidocaine
51. Mepivacaine
52. Prilocaine
53. Cocaine Esters
54. Procaine
55. Tetracaine
Skeletal Muscle Relaxant
56. Succinylcholine Depolarizing
57. Atracurium Non-Deploarizing
58. D-Tubocurarine
59. Mivacurium
60. Baclofen Centrally Acting
61. Cyclobenzaprine
62. Diazepam
63. Tizanidine
64. Dantrolene Direct Acting
Drugs Movement Disorders
65. Levodopa Dopamine Precursor
66. Apomorphine Dopamine agonists
67. Bromocriptine
68. Pramipexole
69. Ropinirole

70. Rasagiline MAO inhibitors


71. Selegiline
72. Entacapone COMT Inhibitors
73. Tolcapone
74. Benztropine Antimuscrinic
75. Haloperidol For Huntington’s disease
76. Reserpine
77. Tetrabenazine

78. Clonidine For tourette’s syndrome


79. Haloperidol
Antipsychotics
80. Chlorpromazine Phenothiazines
81. Fluphenazine
82. Thioridazine
83. Thiothixene Thioxanthene
84. Haloperidol Butyrophenones
85. Clozapine Atypicals
86. Olanzapine

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87. Quetiapine
88. Risperidone
89. Lithium Mood Stablizer
90. Carbamazepine Alternative Drugs for Bipolar Effective disorder
91. Lamotrigine
92. Valproic Acid
Antidepressants
93. Amitriptyline Tricyclic Antidepressants
94. Clomipramine
95. Impipramine
96. Citalopram Selective Serotonin reuptake inhibitors
97. Fluoxetine
98. Paroexetine
99. Sertraline
100. Desvenlafaxine Serotonin norepinephrine reuptake inhibitors
101. Duloxetine
102. Venlafaxine
103. Nafazodone 5-HT2 antagonist
104. Trazodone
105. Amoxapine Heterocyclics
106. Bupropion
107. Maprotiline
108. Mirtazepine
109. Isocarboxazid Mono amine oxidase inhibitors
110. Selegiline
Opioids
111. Fentanyl Strong Agonists
112. Hydromorphone
113. Methadone
114. Morphine
115. Oxymorphone
116. Codeine Partial Agonists
117. Hydrocodone
118. Buperonorphine Mixed opioid agonist-anatagonist
119. Nalbuphine
120. Naloxone Opioid antagonist
121. Naltrexone
122. Codeine Antitussive
123. Dextromethorphan
124. Tramadol Opioids substitutes
Drugs used to treat dependence & addiction
125. Naloxone Opioid Antagonist
126. Naltrexone
127. Methadone Synthetic opioid
128. Buprenorphine Partial µ-receptor
129. Varenicline N-receptor Partial agonist

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130. Oxazepam Benzodiazepines
131. Lorazepam
132. Acamprosate NMDA receptor antagonist
133. Rimonabant Rimonabant

Chemotherapeutic Agents
Anti Bacterial Drugs
Beta-Lactam & Other Cell Wall Synthesis Inhibitors
Drug Type Sub Type
1. Nafcillin Penicillin, Narrow Spectrum
2. Oxacillin
3. Penicillin G
4. Penicillin V
5. Ampicillin Penicillin, Wider Spectrum
6. Amoxcillin
7. Pipelacillim
8. Ticarcillin
Cephalosporins
Drug Type Sub Type
9. Cephalexin Cephalosporins, 1st Generation
10. Cefotetan Cephalosporins, 2nd Generation
11. Cefoxitin
12. Cefuroxime
13. Ceftriaxone Cephalosporins, 3rd Generation
14. Cefotaxime
15. Ceftazidime
16. Cefepime Cephalosporins, 4th Generation
Carbapenems
17. Doripenem Carbapenems
18. Ertapenem
19. Imipenem
20. Meropenem
Monobactams
21. Aztreonam Monobactams
Glycopeptides
22. Vancomycin Glycopeptides
23. Teicoplanin
Lipopeptide
24. Daptomycin Lipopeptide
Tetracyclines,
25. Doxycyline Tetracyclines
26. Minocycline
27. Tetracycline
28. Tigecycline
Macrolides,
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29. Azithyromycin Macrolides
30. Clarithromycin
31. Erythromycin
32. Fidaxomicin
33. Telithromycin
Lincosamide
34. Clindamycin Lincosamide
Streptogramins
35. Quinupristin – Dalfopristin Streptogramins
Chloramphenicol
36. Chloramphenicol Chloramphenicol
Oxazolidinone
37. Linezolid Oxazolidinone
Aminoglycosides & Spectinomycin
38. Amikacin Aminoglycosides
39. Gentamicin
40. Neomycin
41. Streptomycin
42. Tobramycin
Sulfonamides & Trimethoprim.
43. Pyrimethamine Folate Antagonists
44. Sulfadiazine
45. Sulfisoxazole
46. Sulfonamides
47. Trimethoprim
Fluoroquinolones
48. Ciprofloxacin Fluoroquinolones
49. Gemifloxacin
50. Levoflaxcin
51. Moxifloxacin
52. Norfloxacin
53. Ofloxacin
Antimycobacterial drugs
54. Isoniazid Antimycobacterial drugs
55. Rifabutin
56. Rifampin
57. Rifapentone
58. Ethambutol
59. Pyrazinamide
60. Streptomycin
Anti Fungal Agents
Drug Type

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61. Amphotericin B Azoles
62. Fluconazole
63. Itraconazole
64. Ketoconazole
65. Posaconazole
66. Vorizonazole
67. Anidulafungin Echinocandins
68. Caspofungin
69. Micafungin
70. Flucytosine
71. Griseofulvin
72. Terbinafine
Antivirals & Antiretroviral
Drug Type Sub Type
73. Acyclovir Anti Herpes Anti Herpes
74. Penciclovir
75. Valacyclovir
76. Cidofovir Drug for Cytomegalovirus Drug for Cytomegalovirus
77. Ganciclovir
78. Valganciclovir
79. Interferon  α
80. Adefovir-dipivoxil Anti Hepatitis Anti Hepatitis
81. Entecavir
82. Lamivudine
83. Ribavirin
84. Sofosubvir
85. Amantadine Anti Influenza Anti Influenza
86. Oseltamivir
87. Rimantacline
88. Zanamivir
89. Abacavir Anti retroviral drug , NRTIs
90. Didanosine
91. Emtricitabine
92. Lamivudine
93. Stavudine
94. Tenofovir
95. Zalcitabine
96. Zidovudine
97. Delaviridine Anti retroviral , NNRTIs
98. Efavirenz
99. Etravirine
100. Nevirapine
101. Atazanavir Anti retroviral , Protease Inhibitors
102. Darunavir
103. Fosamprenavir
104. Indinavir
105. Nelfinavir

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106. Ritonavir
107. Enfuvirtide Anti retroviral, Entry Inhibitors
108. Maraviroc
Miscellaneous anti Microbial agents & urinary antiseptics
Drug Type
109. Metronidazole Nitroimidazoles
110. Tinidazole
111. Nitrofurantion Urinary Antiseptics
112. Methenamine Salts
113. Alcohol Other antiseptic
114. Chlorhexidine
115. Aldehydes Disinfectant
116. Compound
117. Peroxyden
Anti Protozoal Drugs
Drug Type
118. Artemisins Anti Malarials
119. Atoraquone
120. Chloroquine
121. Mefloquine
122. Promaquine
123. Diloxamide Anti Amebic agents
124. Iodoquinol
125. Metronidazole
126. Paromomycin
127. Pentamidine Miscellaneous
128. Suramin
Anti helminthic drugs
Drug Type
129. Albendazole Drugs against nematodes
130. Diethylcarbamazine
131. Ivermectin
132. Mebendazole
133. Pyrantel Pomoate
134. Bithionol Drugs against Trematodes
135. Praziquantel
136. Niclosamide Drugs against Cestodes
Cancer Chemotherapy
Drug Type
137. Cyclophosphamide Alkylating agent
138. Methotrexate Anti metabolite
139. 6- Mercaptopurine
140. 5- Fluorouracil
141. Vincristine Vinca alkaloids
142. Etoposide Podophyllotoxins
143. Topotecan Campthothecins

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144. Paclitaxel Taxanes
145. Doxorubicin Antracyclines
146. Imatinib Tyrosine Kinase inhibitors
147. Trastuzumab Growth factor receptor Inhibitors
148. Bevacizumab Vascular endothelial growth factor inhibitors
149. Bortezomib Proteasome inhibitors

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