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PHARMA PATENTS GRANTED DURING 2010-11 TO 2013-14 ( UP TO 31-7-2013)

Application No Date of Filing Patent No Patent Grant Date Title Applicant


1074/MUM/2006 07-07-2006 239822 01-04-2010 A MODIFIED RELEASE PHARMACEUTICAL COMPOSITION PANACEA BIOTEC LIMITED
OF BICALUTAMIDE
1115/MUMNP/2007 25-07-2007 238424 02-04-2010 A TRIAZOLO [4,5-d]PYRIMIDINE COMPOUND OF ASTRA ZENECA AB
FORMULA (II)
3902/DELNP/2005 01-09-2005 239827 05-04-2010 A GEL FORMULATIONS ANTARES PHARMA IPL AG
359/CAL/1995 31-03-1995 239838 06-04-2010 A 1 H-SUBSTITUTED-INDOLE-3-GLYOXYLAMIDE ELI LILLY AND COMPANY
COMPOUND AND PROCESS OF PREPARATION THEREOF

13/CAL/2000 10-01-2000 239851 06-04-2010 NOVEL BENZOTHIOPHENE COMPOUNDS, ELI LILLY AND COMPANY
INTERMEDIATES, COMPOSITIONS AND METHODS
THEREOF
3803/DELNP/2005 26-08-2005 239895 07-04-2010 A PHARMACEUTICAL COMPOSITION FOR TREATING OR JARROW FORMULAS, INC.
PREVENTING HUMAN IMMUNODEFICIENCY VIRUS (HIV)
INFECTION, MALARIA OR BOTH
3702/DELNP/2006 28-06-2006 239909 09-04-2010 FURANCARBONYLGUANIDINE DERIVATIVES, THEIR KOREA RESEARCH INSTITUTE OF
PREPARATION AND PHARMACEUTICAL COMPOSITIONS CHEMICAL TECHNOLOGY.
CONTAINING THEM
1165/DELNP/2005 23-03-2005 239936 12-04-2010 A PHARMACEUTICAL FORMULATION FOR TREATMENT SHIRE LLC
OF PATIENTS HAVING ATTENTION DEFICIT
HYPERACTIVITY DISORDER(ADHD)
2221/DELNP/2006 24-04-2006 239954 15-04-2010 NUTRITIONAL COMPOSITION AGAINST SIDE EFECTS OF NESTEC S.A.
CHEMOTHERAPY OR RADIOTHERAPY
1053/DELNP/2004 20-04-2004 239997 21-04-2010 A LYOPHILIZED PHARMACEUTICAL COMPOSITION PFIZER PRODUCTS INC.
5037/DELNP/2005 03-11-2005 240018 23-04-2010 SUBSTITUTED-1-PHTHALAZINAMES AS VR-1 MERCK SHARP & DOHME LIMITED
ANTAGONISTS
2695/DEL/2005 07-10-2005 240034 23-04-2010 A PROCESS TO OBTAIN A PHARMACEUTICAL PRODUCT MADAN, DR. ANIL KUMAR
WITH AN ENHANCED DISSOLUTION RATE AND THE
PHARMACEUTICAL PRODUCT RESULTING THEREOF

IN/PCT/2002/01295/DEL 27-12-2002 240070 27-04-2010 A PHARMACEUTICAL COMPOSITION FOR INTRANASAL ASUBIO PHARMA CO., LTD
ADMINSTRATION COMPRISING A HUMAN
PARATHYROID HORMONE PEPTIDE OR ITS DERIVATIVE"

877/MUMNP/2007 11-06-2007 240123 28-04-2010 AN OILY ISOTROPE PHARMACEUTICAL COMPOSITION SA VETOQUINOL

402/DELNP/2006 23-01-2006 240207 29-04-2010 A FLUORO SUBSTITUTED OMEGA-CARBOXYARYL BAYER HEALTHCARE LLC
DIPHENYL UREA COMPOUND OR A SALT, AN ISOLATED
STEREOISOMER THEREOF

365/DELNP/2005 01-02-2005 240219 29-04-2010 A COMPOUND 2-(3-AMINOARYL) AMINO-4-ARYL- AB SCIENCE


THIAZOLES OF FORMULA I.
50/CAL/2001 30-01-2001 240197 29-04-2010 A VACCINE PREPARED FOR THE TREATMENT OR RICAN LIMITED
PROPHYLAXIS OF HELICOBACTER PYLORI INFECTION

3435/DELNP/2004 04-11-2004 240229 30-04-2010 A 3, 17-DISUBSTITUTED MORPHINAN COMPOUND AND JENKEN BIOSCIENCES, INC
PHARMACEUTICAL COMPOSITION THEREOF
1599/DELNP/2005 20-04-2005 240249 30-04-2010 AN IMIDAZOLE COMPOUND USES AS CARDIOVASCULAR PORTELA & C.A., SA.
AGENTS
1516/DELNP/2005 15-04-2005 240264 30-04-2010 AN ANALOGUE OF KAHALALIDE F PHARMA MAR, S.A.U
4540/DELNP/2006 07-08-2006 240268 30-04-2010 NEW AZABICYCLIC COMPOUNDS, A PROCESS FOR THEIR LES LABORATORIES SERVIER
PREPARATION AND PHARMACEUTICAL. COMPOSITIONS
CONTAINING THEM
927/KOLNP/2006 13-04-2006 240314 04-05-2010 DERIVATIVES OF N-[PHENYL (PYRROLIDINE-2-YL) SANOFI-AVENTIS
METHYL ] BENZAMIDE AND N-[ ( AZEPAN-2-YL )
PHENYLMETHYL ] BENZAMIDE, PREPARATION METHOD
THEREOF AND APPLICATION OF SAME IN
THERAPEUTICS
IN/PCT/2002/01272/DEL 20-12-2002 240340 05-05-2010 A COMPOSITION USEFUL AGAINST NEURONAL DAMAGE HUNTER FLEMING LIMITED

30/DELNP/2003 10-01-2003 240341 05-05-2010 A PYRIDOPYRROLOPYRIMIDINE COMPOUND USED AS PHARMA MAR, S.A.
ANTITUMOURAL AGENT
1286/DELNP/2005 31-03-2005 240358 05-05-2010 DEVELOPMENT OF NOVEL HEREBAL FORMULATION COUNCIL OF SCIENTIFIC & INDUSTRIAL
USED AS AN ANTI-DIABETIC ON TRADITIONAL RESEARCH
INDIGENOUS KNOWLEDGE
IN/PCT/2001/01142/MUM 19-09-2001 240371 06-05-2010 ANTHELMINTIC COMPOSITIONS ASHMONT HOLDINGS LIMITED
6170/DELNP/2005 30-12-2005 240378 06-05-2010 HYDROXYPYRIDINE CGRP RECEPTOR ANTAGONISTS MERCK AND CO.INC.
4733/DELNP/2005 18-10-2005 240379 06-05-2010 PHARMACEUTICAL FORMULATION OF THE SODIUM BOEHRINGER INGELHEIM
SALT OF TELMISARTAN INTERNATIONAL GMBH
IN/PCT/2001/00708/DEL 08-08-2001 240383 06-05-2010 A BRANCHED CHAIN AMINO ACID-DEPENDENT WARNER-LAMBERT COMPANY
AMINOTRANSFERASE INHIBITORS COMPOUND
779/MUMNP/2006 05-07-2006 240396 07-05-2010 A PHARMACEUTICAL COMPOSITION CONTAINING MERZ PHARMA GMBH & CO. KGAA
MEMANTINE FOR THE TREATMENT OF MILD AND MILD-
TO-MODERATE ALZHEIMER S DISEASE
1330/DEL/2004 19-07-2004 240422 10-05-2010 A HERBAL COMPOSITION FOR THE TREATMENT OF HIV PANDEY , SANTOSH KUMAR
AND A PROCESS OF PREPARING THE SAME
446/KOLNP/2004 02-04-2004 240474 12-05-2010 PHARMACEUTICAL COMPOSITION COMPRISING GAMA- KALVINSH IVARS
BUTYROBETAINE
5950/DELNP/2005 20-12-2005 240515 14-05-2010 HETEROARYLOXY NITROGENOUS SATURATED BANYU PHARMACEUTICAL CO.,LTD.
HETEROCYCLIC DERIVATIVE
767/DELNP/2006 15-02-2006 240599 19-05-2010 , SPRAY-DRIED AMORPHOUS POWDER BOEHRINGER INGELHEIM PHARMA
GMBH & CO. KG.
1903/DELNP/2004 02-07-2004 240690 26-05-2010 COMPOSITION, SYNTHESIS, DIAGNOSTIC AND MICHAEL A. MURPHY 
THERAPEUTIC APPLICATIONS OF POLYAMINES
1564/DELNP/2005 19-04-2005 240734 26-05-2010 AN IMMUNOGEN FOR PREPARATION OF THERAPEUTIC INSTITUTE OF IMMUNOLOGY, PLA
VACCINES FOR TREATMENT OF HEPATITIS B AND
PRODUCING METHOD THEREOF
2657/DELNP/2004 09-09-2004 240755 28-05-2010 PHARMACEUTICAL PREPARATION CONTAINING EURO-CELTIQUE S.A.,
OXYCODONE AND NALOXONE"
450/DELNP/2005 07-02-2005 240762 28-05-2010 A METALLOPROTEINASE INHIBITOR COMPOUND AND ASTRAZENEECA AB
PHARMACEUTICAL COMPOSITIONS CONTAINING THE
SAME
762/DEL/2000 25-08-2000 240763 28-05-2010 AN IMPROVED MALE CONTRACEPTIVE FORMULATION SUJOY KUMAR GUHA

714/MUMNP/2006 19-06-2006 240768 31-05-2010 COMPOSITION AND METHOD FOR REDUCING THE HINDUSTAN UNILEVER LIMITED
EFFECTS OF STRESS ON SKIN CONDITION
946/KOLNP/2006 17-04-2006 240787 01-06-2010 DERIVATIVES OF N-[PHENYL(ALKYLPIPERIDINE-2- SANOFI-AVENTIS
YL)METHYL]BENZAMIDE
1693/DELNP/2004 15-06-2004 240817 02-06-2010 ISOTRETINOIN NANOPARTICULATE COMPOSITIONS RANBAXY LABORATORIES LIMITED
5582/DELNP/2005 01-12-2005 240818 02-06-2010 A SUBSTITUTED BENZAMIDE COMPOUND AND ASTELLAS PHARMA INC.
PHARMACEUTICAL COMPOSITION THEREOF
921/DEL/1998 13-04-1998 240834 03-06-2010 A CELL STRUCTURE MEDIUM COMPOSITION FOR THE BAYER CORPORATION
PRODUCTION OF RECOMBINANT FACTOR VIII
4611/DELNP/2005 10-10-2005 240846 04-06-2010 SELECTIVE SPIROCYCLIC GLUCOCORTICOID RECEPTOR MERCK SHARP & DOHME CORP.,
MODULATORS
640/DELNP/2005 18-02-2005 240871 07-06-2010 COMPOSITION FOR SOLUBILIZATION OF PACLITAXEL DAEHWA PHARM. CO., LTD.
AND PREPARATION METHOD THEREOF
IN/PCT/2002/1483/KOL 02-12-2002 240925 10-06-2010 A TOPICAL ORAL COMPOSITION THE PROCTER & GAMBLE COMPANY
2210/CAL/1998 23-12-1998 240930 10-06-2010 PRODRUGS OF ASPARTYL PROTEASE INHIBITORS VERTEX PHARMACEUTICALS
INCORPORATED
1185/DEL/1999 07-09-1999 240939 10-06-2010 A SPATTER CURE COMPOUND AND A PROCESS FOR THE MADAN MOHAN BANDYOPADHYAY
PREPARATION THEREOF FOR USE DURING THE
WELDING PROCESS
925/KOLNP/2006 13-04-2006 240989 14-06-2010 N - HETEROCYCLYL - METHYLBENZAMIDE DERIVATIVE SANOFI-AVENTIS
COMPOUNDS
3115/DELNP/2005 13-07-2005 240990 14-06-2010 A PHARMACEUTICAL COMPOSITION COMPRISING AN ASTRAZENECA AB
AROMATASE INHIBITOR,A PROGESTIN AND AN
OESTROGEN
461/DELNP/2005 07-02-2005 241002 14-06-2010 COMPOSITION COMPRISING THE EXTRACT OF Helixir Co., Ltd.
ACTINIDIA ARGUTA AND RELATED SPECIES FOR THE
PREVENTION AND TREATMENT OF ALLERGIC DISEASE
AND NON-ALLERGIC INFLAMMATORY DISEASE

5320/DELNP/2005 21-11-2005 241017 15-06-2010 MACROCYCLIC QUINAZOLINE DERIVATIVES AS JANSSEN PHARMACEUTICA N.V.
ANTIPROLIFERATIVES AGENTS
228/DELNP/2004 03-02-2004 241018 15-06-2010 NOVEL COMPOUNDS AS ANTI-INFLAMMATORY, 4SC AG Germany
IMMUNOMODULATORY AND ANTI-PROLIFERATORY
AGENTS
250/MUM/2004 01-03-2004 241016 15-06-2010 GASTRIC RETENTION CONTROLLED DRUG DELIVERY SUN PHARMA ADVANCED RESEARCH
SYSTEM COMPANY LIMITED
1910/KOLNP/2004 13-12-2004 241066 17-06-2010 TRICYCLIC COMPOUNDS AS MODULATORS OF STEROID ELI LILLY AND COMPANY
HORMONE NUCLEAR RECEPTORS
1077/MUMNP/2005 03-10-2005 241110 17-06-2010 POLYMERIC OLIGONUCLEOTIDE PRODRUGS ENZON PHARMACEUTICALS, INC.
207/CAL/1998 09-02-1998 241050 17-06-2010 PEPTIDES FOR DIAGNOSING AND TREATMENT OF GERHILD WILDNER
AUTOIMMUNE DISEASES
IN/PCT/2003/00001/DEL 01-01-2003 241117 18-06-2010 TOPICAL LIPOSOMAL FORMULATION COMPRISING CENTRO DE INVESTIGACIÓN Y
CLOBETASOL PROPIONATE ENCAPSULATED IN DESARROLLO DE MEDICAMENTOS
LIPOSOMES (CIDEM)
1210/DEL/2004 30-06-2004 241119 18-06-2010 A NOVEL COBALT COMPLEX USEFUL FOR REVERSAL OF INDIAN COUNCIL OF MEDICAL
DRUG RESISTANCE AND THE PREPARATION THEREOF RESEARCH

1437/MUMNP/2006 27-11-2006 241166 22-06-2010 AN IMMEDIATE RELEASE DOSAGE FORMULATION MERZ PHARMA GMBH & CO. KGAA
COMPRISING MEMANTINE OR NERAMEXANE
3593/DELNP/2004 17-11-2004 241169 22-06-2010 IMMUNE STIMULATING AND CONTROLLING EYEGENE INC.,
COMPOSITION COMPRISING BACTERIAL
CHROMOSOMAL DNA FRAGMENTS AND NON-TOXIC
LIPOPOLYSACCHARIDES
797/DELNP/2006 16-02-2006 241200 23-06-2010 A COMPOSITION FOR TREATMENT OF DIABETES AYURVEDIC-LIFE INTERNATIONAL, LLC.
3456/DELNP/2005 03-08-2005 241228 24-06-2010 A COMPOSITION MATERIAL FOR TRANSMUCOSAL MAGLE HOLDING AB
DELIVERY
IN/PCT/2002/00673/DEL 05-07-2002 241240 24-06-2010 BENZAMIDAZOLE DERIVATIVE TEIJIN LIMITED
2008/DEL/1998 14-07-1998 241229 24-06-2010 A TRIAOLO[4, 5-D] PYRIMIDINE COMPOUND OF ASTRAZENECA UK LIMITED,
FORMULA (I)
3338/CHENP/2006 14-09-2006 241259 25-06-2010 A PHARMACEUTICAL FORMULATION FOR TREATMENT THE REGENTS OF THE UNIVERSITY OF
OF AIRWAY MUCUS HYPERSECRETION CALIFORNIA
510/DELNP/2005 10-02-2005 241260 25-06-2010 PHARMACEUTICAL COMPOSITIONS FOR INHALATION BOEHRINGER INGELHEIM PHARMA
CONTAINING A NEW ANTICHOLINERGIC IN GMBH & CO. KG.
CONJUNCTION WITH CORTICOSTEROIDS AND
BETAMIMETICS
2187/DELNP/2006 21-04-2006 241296 28-06-2010 A COMPOSITION USEFUL FOR TREATMENT OF A ALLERGAN  INC.
POSTERIOR SEGMENT OF AN EYE
1095/CHENP/2006 30-03-2006 241325 29-06-2010 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE IRM LLC
INHIBITORS
3331/DEL/1997 20-11-1997 241306 29-06-2010 ACTIVE FLUOXASTROBIN COMPOUND COMBINATION BAYER AKTIENGESELLSCHAFT

1184/DEL/2004 25-06-2004 241416 02-07-2010 A CHEMOTHERAPEUTIC COMPOSITION USED IN THE The Secretary, Department of
TREATMENT OF CANCER. Biotechnology
2245/DELNP/2006 24-04-2006 241460 06-07-2010 MACROCYCLIC CARBOXYLIC ACIDS AND INTERMUNE INC.
ACYLSULFONAMIDES AS INHIBITORS OF HCV
REPLICATION
609/CHENP/2007 12-02-2007 241476 07-07-2010 STABLE PEGYLATED INTERFERON ALPHA FORMULATION SCHERING CORPORATION

3781/DELNP/2004 30-11-2004 241529 10-07-2010 A HYDROGEL SUSTAINED-RELEASE PREPARATION TYPE ASTELLAS PHARMA INC
TABLET
7602/DELNP/2006 15-12-2006 241533 12-07-2010 SUBSTITUTED PYRROLOTRIAZINE COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY
IN/PCT/2001/00757/DEL 24-08-2001 241535 12-07-2010 A PHARMACEUTICAL COMPOSITION" TRIANGLE PHARMACEUTICALS, INC.
845/KOLNP/2006 06-04-2006 241537 12-07-2010 SELECTIVE KINASE INHIBITORS CYTOPIA RESEARCH PTY LTD.
1374/MUMNP/2007 10-09-2007 241588 14-07-2010 A CONSUMABLE FILM ADAPTED TO RAPIDLY DISSOLVE WARNER - LAMBERT COMPANY LLC.
IN THE MOUTH OF A CONSUMER
5778/DELNP/2006 05-10-2006 241591 14-07-2010 (3,3-Difluoropyrrolidin-1-y1)-((2S,4S)-4-(4-(pyrimidin-2- PFIZER PRODUCTS INC
y1) piperazin-1-yl)pyrrolidin-2-yl)methanone

529/MUMNP/2006 09-05-2006 241597 14-07-2010 METHOXY PHOSPHONATE NUCLEOTIDE PRODRUG GILEAD SCIENCES, INC.
1243/MUM/2005 03-10-2005 241583 14-07-2010 A HERBAL PAIN- RELIEF COMPOSITION PHARMACON REMEDIES [BOMBAY]
PVT. LTD.,
1610/DELNP/2005 20-04-2005 241646 17-07-2010 A BIOADHESIVE PHARMACEUTICAL COMPOSITION COLUMBIA LABORATORIES (BERMUDA)
COMPRISING AN IONIC TREATING AGENT AND AN IONIC LIMITED
POLYMER POLYCARBOPHIL
IN/PCT/1999/00001/DEL 07-12-1999 241656 19-07-2010 PYRIMIDINONE COMPOUNDS AND PROCESS FOR BORYUNG PHARMACEUTICAL CO. LTD.,
PREPARING THE SAME
215/DELNP/2006 12-01-2006 241658 19-07-2010 INFANT OR FOLLOW-ON FORMULA NESTEC S.A.
1649/DELNP/2006 27-03-2006 241659 19-07-2010 A COMBINATION COMPRISING CANDESARTAN OR A ASTRAZENECA UK LIMITED.
PHARMACEUTICALLY ACCEPTABLE SALT THEREOF
3409/DELNP/2005 01-08-2005 241660 19-07-2010 PHARMACEUTICAL LIQUID FORMULATION ARAKIS LTD
1960/DELNP/2004 08-07-2004 241677 20-07-2010 A PHARMACEUTICAL COMPOSITION COMPRISING A NERVIANO MEDICAL SCIENCES S.R.L.
PHARMACEUTICALLY ACCEPTABLE CARRIER OR
EXCIPIENT AND, AS ACTIVE INGREDIENT, AN ACRYLOYL
DISTAMYCIN DERIVATIVE
2258/DELNP/2006 24-04-2006 241685 20-07-2010 A COMPOSITION LI, GUOQIAO
769/DELNP/2006 15-02-2006 241721 22-07-2010 ANTIMICROBIAL COMPOSITIONS CONTAINING THE TRUSTEES OF COLUMBIA
SYNERGISTIC COMBINATIONS OF QUATERNARY UNIVERSITY IN THE CITY OF NEW YORK
AMMONIUM COMPOUNDS AND ESSENTIAL OILS
AND/OR CONSTITUENTS THEREOF
1415/MUMNP/2005 20-12-2005 241735 22-07-2010 AN ISOLATED ANTIBODY BAYER SCHERING PHARMA
AKTIENGESELLSCHAFT
IN/PCT/2002/00588/DEL 10-06-2002 241773 24-07-2010 PYRROLO[2,3-d] PYRIMIDINE COMPOUNDS PFIZER PRODUCTS INC.
2090/DEL/1998 20-07-1998 241782 24-07-2010 A PHARMACEUTICAL COMPOSITION COMPRISING 5-[4- SMITHKLINE BEECHAM P.L.C
[2(N-METHYL-N-(2-PYRIDYL)AMINO]
ETHOXY]BENZYL]THIAZOLIDINE-2,4-DIONE
128/DELNP/2004 19-01-2004 241823 27-07-2010 A PROLONGED RELEASE MUCOADHESIVE TABLET BIOALLIANCE PHARMA
2226/DEL/2004 08-11-2004 241827 27-07-2010 A COMPOSITION FOR ENHANCING BIOAVAILABILITY OF COUNCIL OF SCIENTIFIC AND
DRUGS/NUTRACEUTICALS. INDUSTRIAL RESEARCH
708/CHENP/2004 05-04-2004 241838 28-07-2010 AN ANGIOTENSIN PEPTIDE MOIETY-CARRIER CYTOS BIOTECHNOLOGY AG
CONJUGATE.
462/KOLNP/2005 18-03-2005 241844 28-07-2010 9, 10-DEHYDRO-DESOXY-EPOTHILONE COMPOUNDS SLOAN-KETTERING INSTITUTE FOR
CANCER RESEARCH
5943/DELNP/2005 20-12-2005 241905 30-07-2010 BENZODIAZEPINE CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP.,
2868/CHENP/2004 16-12-2004 241952 02-08-2010 A COMPOSITION FOR ENHANCING IMMUNE RESPONSE CYTOS BIOTECHNOLOGY AG

1683/MUMNP/2007 15-10-2007 241989 04-08-2010 TABLET- TYPE CONTROLLED-RELEASE PREPARATION HENNIG ARZNEIMITTEL GMBH & CO.
CONTAINING CINNARIZINE AND DIMENHYDRINATE FOR KG
COMBATING VERTIGO
1278/DELNP/2005 31-03-2005 241999 05-08-2010 SUBSTITUTED CARBAMIC ACID QUINOLIN-6-YL ESTERS COUNCIL OF SCIENTIFIC & INDUSTRIAL
AS ACETYLCHOLINESTERASE INHIBITORS RESEARCH
3331/DELNP/2006 09-06-2006 242015 06-08-2010 A 2-QUINOLINONE OR 2-QUINOXALINONE COMPOUND JANSSEN PHARMACEUTICA N.V.

5565/DELNP/2006 25-09-2006 242021 06-08-2010 THE COMPOUNDS 2-[(2-FLUORO-6- PFIZER INC


METHOXZYPHENOXY)(3-FLUOROPHENYL)
METHYL]MORPHOLINE AND PHARMACEUTICALLY
ACCEPTABLE SALTS THEREOF
1182/DELNP/2005 24-03-2005 242025 06-08-2010 AN OCULAR TREATMENT SOLUTION FOR THE JIN JUN ZHANG
TREATMENT OR PREVENTION OF POSTERIOR CAPSULAR
OPACIFICATION
2630/DELNP/2004 08-09-2004 242026 06-08-2010 A QUINAZOLINE DERIVATIVE ASTRAZENECA AB
471/CHENP/2006 06-02-2006 242036 06-08-2010 METHODS AND COMPOSITIONS FOR CANCER THERAPY HENRY FORD HEALTH SYSTEM
USING NOVEL ADENOVIRUS
53/DEL/2004 12-01-2004 242024 06-08-2010 A PHARMACEUTICAL PREPARATION FOR THE EURO-CELTIQUE S.A.,
PREVENTION OR THE TREATMENT OF INFECTIONS IN
THE INTERIOR OF THE HUMAN OR ANIMAL BODY

4759/DELNP/2005 19-10-2005 242056 09-08-2010 PHARMACEUTICAL COMPOSITION FOR A MERCK SHARP & DOHME CORP.,
ATHEROSCLEROSIS,DYSLIPIDEMIAS AND RELATED
CONDITIONS
1265/DELNP/2006 08-03-2006 242095 11-08-2010 AN ORAL COMPOSITION OF ITRACONAZOLE HAVING HANMI PHARM.CO. LTD.
IMPROVED ITRACONAZOLE BIOAVAILABILITY

413/MUM/2003 25-04-2003 242111 11-08-2010 CRYSTALLINE CLOPIDOGREL BESYLATE AND PROCESS CADILA HEALTHCARE LIMITED
FOR PREPARATION THEREOF
489/DEL/2001 16-04-2001 242113 11-08-2010 A RUMEN BYPASS COMPOSITION CONTAINING A JUBILANT ORGANOSYS LIMITED
BIOACTIVE SUBSTANCE
2472/DELNP/2005 08-06-2005 242134 16-08-2010 THE COMPOUND (-) TENATOPRAZOLE, OR (-)-5- SIDEM PHARMA SA
METHOXY -2[[(4-METHOXY-3,5-DIMETHYL-2-
PYRIDYL)METHYL]SULFINYL]IMIDAZO-[4,5-B]PYRIDINE

1058/MUMNP/2007 13-07-2007 242149 17-08-2010 NOVEL HETEROCYCLIC COMPOUNDS USEFUL FOR THE GLENMARK PHARMACEUTICALS S. A.
TREATMENT OF INFLAMMATORY AND ALLERGIC
DISORDERS
IN/PCT/2002/00772/DEL 07-08-2002 242177 18-08-2010 PARTNERS OF PTB1 DOMAIN OF FE65, PREPARATION AVENTIS PHARMA S.A.,
AND USES
1350/DELNP/2003 25-08-2003 242195 18-08-2010 A COMPLEX FOR ORAL DELIVERY OF DRUGS, COUNCIL OF SCIENTIFIC & INDUSTRIAL
THERAPEUTIC PROTEINS AND PEPTIDES AND VACCINES RESEARCH

991/DEL/2003 12-08-2003 242180 18-08-2010 A COMPOSITION USEFUL FOR THE TREATMENT OF COUNCIL OF SCIENTIFIC AND
LEISHMANIASIS INDUSTRIAL RESEARCH
3296/DELNP/2006 08-06-2006 242247 19-08-2010 AMINOBENZIMIDAZOLES AND BENZIMIDAZOLES AS TIBOTEC PHARMACEUTICALS LTD.
INHIBITORS OF RESPIRATORY SYNCYTIAL VIRUS
REPLICATION
1855/KOLNP/2006 04-07-2006 242344 24-08-2010 INHIBITOR OF PROTEIN MODIFICATION PRODUCTS TOKAI UNIVERSITY EDUCATIONAL
FORMATION SYSTEM
1702/KOLNP/2006 20-06-2006 242347 24-08-2010 NOVEL COMBINATION OF ANTICHOLINERGIC AND beta MEDA PHARMA GMBH & CO. KG
MIMETICS FOR THE TREATMENT OF RESPIRATORY
DISEASES
4232/KOLNP/2007 05-11-2007 242351 24-08-2010 COMPOUND USEFUL AS AMPA RECEPTOR ELI LILLY AND COMPANY
POTENTIATORS
3811/KOLNP/2007 08-10-2007 242352 24-08-2010 PHARMACEUTICAL COMPOSITION AND METHOD USING TOYAMA CHEMICAL CO., LTD.
ANTIFUNGAL AGENT IN COMBINATION
2071/KOLNP/2006 24-07-2006 242354 24-08-2010 PHARMACEUTICAL COMPOSITION FOR PROMOTING OTSUKA PHARMACEUTICAL
ANGIOGENESIS. CO. LTD
4484/KOLNP/2007 21-11-2007 242367 24-08-2010 A PHARMACEUTICAL COMPOSITION ADVANCED SCIENTIFIC DEVELOPMENTS

135/DEL/2003 18-02-2003 242387 25-08-2010 HERBAL HEALTH PROTECTIVE AND PROMOTIVE COUNCIL OF SCIENTIFIC AND
NUTRACEUTICAL FORMULATION FOR DIABETICS AND INDUSTRIAL RESEARCH
PROCESS FOR PREPARING THE SAME
327/DEL/2000 28-03-2000 242390 25-08-2010 NOVEL α-HYDROXY-9, 12-TRICOSDIENOIC ACID COUNCIL OF SCIENTIFIC AND
USEFUL AS THERAPEUTIC AGENT INDUSTRIAL RESEARCH
3140/DELNP/2006 01-06-2006 242466 27-08-2010 MORPHOLINYL CONTAINING BENZIMIDAZOLES AS TIBOTEC PHARMACEUTICALS LTD.
INHIBITORS OF RESPIRATORY SYNCYTIAL VIRUS
REPLICATION
6010/DELNP/2005 22-12-2005 242467 27-08-2010 A COMPOSITION FOR THE BETTER TREATMENT OF INDENA S.P.A.
RHEUMATOID ARTHRITIS
403/CHENP/2004 27-02-2004 242497 30-08-2010 PHARMACEUTICAL COMPOSITION COMPRISING NOVARTIS AG
LUMIRACOXIB
2991/DELNP/2005 05-07-2005 242504 30-08-2010 A COMPOSITIONS FOR INTRANASAL DELIVERY OF ARCHIMEDES DEVELOPMENT LIMITED
FENTANYL
2785/KOLNP/2006 25-09-2006 242537 31-08-2010 BENZIMIDAZOLE DERIVATIVE AND A PROCESS FOR THE TAKEDA PHARMACEUTICAL COMPANY
PREPARATION THEREOF LIMITED
849/KOLNP/2007 09-03-2007 242552 01-09-2010 SULPHONAMIDE DERIVATIVES, THE PREPARATION LABORATORIOS DEL DR. ESTEVE, S.A.
THEREOF AND THE APPLICATION OF SAME AS
MEDICAMENTS
2628/DELNP/2006 10-05-2006 242729 07-09-2010 AN OIL-BASED FORMULATION FOR NASAL APPLICATION MATTERN UDO

2159/MUM/2006 29-12-2006 242722 07-09-2010 A COMPOSITION FOR BODY WEIGHT LOSS Dr. Kishori Ganpat Apte
3415/DELNP/2004 03-11-2004 242804 14-09-2010 MODIFIED RELEASE PHARMACEUTICAL FORMULATION ASTRAZENECA AB

258/DELNP/2005 24-01-2005 242831 15-09-2010 AN ANTI-MICROBIAL COMPOSITION THE QUIGLEY CORPORATION


1449/MUM/2005 21-11-2005 242838 15-09-2010 COMPOSITION FOR ENHANCING ANTIBACTERIAL ADVANCED ENZYME TECHNOLOGIES
ACTIVITY OF ANTIBACTERIAL AGENTS LIMITED
24/DELNP/2005 04-01-2005 242889 17-09-2010 COMPOUNDS HAVING ANTI-PARASITIC,IN PARTICULAR CENTRE NATIONAL DE LA RECHERCHE
ANTIMALARIAL ATIVITY AND COMPOSITIONS THEREOF SCIENTIFIQUE (CNRS)

39/DELNP/2005 05-01-2005 242893 17-09-2010 A SUSTAINED-RELEASE PHARMACEUTICAL PHARMACIA CORPORATION,


COMPOSITION
2266/DELNP/2004 04-08-2004 242898 17-09-2010 A PHARMACEUTICAL COMPOSITION COMPRISING 4-(3'- ASTRAZENECA AB,
CHLORO-4'-FLUOROANILINO)-7- METHOXY-6-(3-
MORPHOLINOPROPOXY) QUINAZOLINE OR A
PHARMACEUTICALLY-ACCEPTABLE SALT THEREOF
3455/DELNP/2004 05-11-2004 242901 17-09-2010 A COMPOUND FOR COMBATING URINARY TRACT MOUNT COOK BIOSCIENCES 
DYSFUNCTION AND A FORMULATION THEREOF INC. 
43/DELNP/2005 05-01-2005 242902 17-09-2010 A SUSTAINED-RELEASE PHARMACEUTICAL PHARMACIA CORPORATION
COMPOSITION
5590/DELNP/2005 01-12-2005 242904 17-09-2010 3-DEMETHYL-AND 3-DEMETHYLTHIO-COLLCHICHINE INDENA S.P.A.
DERIVATIVES
1613/DELNP/2003 07-10-2003 242910 18-09-2010 A PHARMACEUTICAL COMPOSITION FOR THE HF ARZNEIMITTELFORSCHUNG GMBH
TREATMENT OF COGNITIVE DISTURBANCES
OCCURRING AS SEQUELAE
4138/DELNP/2004 27-12-2004 242912 18-09-2010 AN ORALLY DELIVERABLE PHARMACEUTICAL PHARMACIA CORPORATION
COMPOSITION
1114/DELNP/2005 21-03-2005 242928 20-09-2010 A PHARMACEUTICAL COMPOSITION FOR PREPARING A BIOGEN IDEC MA INC.,
MEDICAMENT FOR THE TREATMENT OF CHRONIC
DEMYELINATING MOTOR NEUROPATHY

2015/DELNP/2006 12-04-2006 242935 20-09-2010 IMPLANTS WITH ATTACHED SILYLATED THERAPEUTIC SMART TECH LP.,
AGENTS
382/DELNP/2005 02-02-2005 242939 21-09-2010 A COMPOUND 1-(4-BENZOYLPIPERAZIN-1-YL)-2-(4- BRISTOL-MYERS SQUIBB COMPANY
FLUORO-7-(1 H-1,2,3-TRIAZOL-1-YL)-1H-PYRROLO[2,3-
YL)ETHANE-1,2-DIONE OF FORMULA (A)

416/DELNP/2005 03-02-2005 242987 23-09-2010 ANTIBODIES AND IMMUNOCONJUGATES BINDING TO BOARD OF REGENTS, THE UNIVERSITY
AMINOPHOSPHOLIPIDS AND THEIR USE IN TREATING OF TEXAS SYSTEM
VIRAL INFECTIONS
865/DELNP/2005 04-03-2005 243032 24-09-2010 NOVEL COMPOUND, A COMPSITION COMPRISING SUCH GALDERMA RESEARCH &
NOVEL COMPOUND AND A PROCESS THEREOF" DEVELOPMENT, S.N.C.,

2728/CHENP/2006 24-07-2006 243035 24-09-2010 ANALOGS OF BENZOQUINONE-CONTAINING INFINITY DISCOVERY INC


ANSAMYCINS FOR THE TREATMENT OF CANCER
1669/DELNP/2005 25-04-2005 243061 27-09-2010 A DIRECTLY TABLETABLE GASTRORESISTANT SPHEROID ETHYPHARM
AND METHOD FOR PREPARING THE SAME

1310/DELNP/2005 01-04-2005 243091 27-09-2010 CYCLIC NUCLEOTIDE PHOSPHODIESTERASE INHIBITOR NEURO3D


COMPOUNDS
555/DELNP/2005 14-02-2005 243249 30-09-2010 CANNABINOID LIQUID FORMULATIONS FOR MUCOSAL GW PAHRMA LIMITED
ADMINISTRATION
3243/DELNP/2006 06-06-2006 243281 01-10-2010 N-ARYL PIPERIDINE SUBSTITUTED JANSSEN PHARMACEUTICA N.V.
BIPHENYLCARBOXAMIDES AS INHIBITORS OF
APOLIPOPROTE IN B
1045/KOLNP/2005 01-06-2005 243339 06-10-2010 NEW BIOREVERSIBLE ESTER PRODRUG AND ORION CORPORATION
PHARMACEUTICAL COMPOSITON CONTAINING THE
SAME
2241/DELNP/2003 22-12-2003 243378 08-10-2010 A DISPIRO 1,2,4,-TRIOXOLANE MEDICINES FOR MALARIA VENTURE
2219/DELNP/2005 25-05-2005 243438 18-10-2010 A COMPOSITION FOR TREATING PULMONARY TRANSAVE, INC.
INFECTION IN A PATIENT
1482/DELNP/2005 13-04-2005 243445 19-10-2010 LACTOFERRIN COMPOSITIONS AGENNIX INCORPORATED
IN/PCT/2002/00248/DEL 28-02-2002 243451 19-10-2010 A PHARMACEUTICAL COMPOSITION (MEDICAMENT) SCHERING AKTIENGESELLSCHAFT

1572/DELNP/2005 19-04-2005 243463 19-10-2010 A MILNACIPRAN FORMULATION THAT PROVIDES COLLEGIUM PHARMACEUTICAL, INC
PULSATILE RELEASE OF MILNACIPRAN
IN/PCT/2001/01164/DEL 18-12-2001 243473 20-10-2010 ANESTHETIC COMPOSITION FOR INTRAVENOUS KUHNIL PHARM CO., LTD.
INJECTION COMPRISING PROPOFOL
1709/DELNP/2003 20-10-2003 243499 21-10-2010 A PIPERIDINYL BENZOXAZOLONE COMPOUND OF EURO-CELTIQUE, S.A
FORMULA I
267/DELNP/2005 24-01-2005 243502 21-10-2010 4-(SUBSTITUTED ARYL)-5-HYDROXYISOQUINOLINONE KYORIN PHARMACEUTICAL CO.,LTD
DERIVATIVE
1680/DELNP/2003 16-10-2003 243508 21-10-2010 SPIROPYRAZOLE COMPOUNDS EXHIBITING AFFINITY EURO-CELTIQUE, S.A
FOR THE OPIOID RECEPTOR-LIKE (ORLI) RECEPTOR
3854/DELNP/2004 06-12-2004 243509 21-10-2010 A BIFUNCTIONAL COMPOUND COMPRISING A PROTEIN DUOTOL AB
CONJUGATED WITH AN IMMUNOMODULATING
NUCLEIE ACID
2958/DELNP/2004 29-09-2004 243516 21-10-2010 A PHARMACEUTICAL COMPOSITION COMPRISING AN PFIZER INC
EP4 RECEPTOR ANTAGONIST
890/DELNP/2007 02-02-2007 243571 26-10-2010 AMINOPYRIDINE COMPOUNDS AS PROTEIN KINASE PFIZER INC.
INHIBITORS FOR THE TREATMENT OF CANCER

153/DEL/2004 30-01-2004 243559 26-10-2010 A NOVEL COMBINATORIAL LIBRARY OF 3 AND 30- COUNCIL OF SCIENTIFIC AND
SUBSTITUTED LUP-20(29)- ENE DERIVATIVES USEFUL AS INDUSTRIAL RESEARCH
ANTI-MALARIAL AGENTS
IN/PCT/2002/00150/DEL 04-02-2002 243610 27-10-2010 AN AQUEOUS COMPOSITION COLGATE-PALMOLIVE COMPANY
47/DEL/2000 21-01-2000 243577 27-10-2010 A THERAPEUTIC COMPOSITION FOR PANACEA BIOTEC LIMITED
TOPICAL/TRANSDERMAL USE AND A PROCESS FOR
PREPARATION THEREOF
1299/DEL/1999 28-09-1999 243594 27-10-2010 CONTROLLED RELEASE COMPOSITION COMPRISING PANACEA BIOTEC LIMITED
NIMESULIDE
567/CHE/2004 17-06-2004 243595 27-10-2010 NOVEL INTERMEDIATE FOR THE PRERPARATION OF ORCHID CHEMICALS &
CEFOTIAM PHARMACEUTICALS LTD
IN/PCT/2000/207/KOL 10-08-2000 243613 28-10-2010 A CYCLOALKENE COMPOUND TAKEDA PHARMACEUTICAL COMPANY
LIMITED
648/DELNP/2003 29-04-2003 243648 28-10-2010 A SOLID ORAL CONTROLLED-RELEASE COMPOSITION EURO-CELTIQUE S.A.

1113/DELNP/2006 02-03-2006 243668 29-10-2010 AMIDOMETHYL- SUBSTITUTED 1-(CARBOXYALKYL)- SOLVAY PHARMACEUTICALS GMBH
CYCLOPENTYLCARBONYLAMINO-BENZAZEPINE-N-
ACETIC ACID COMPOUNDS OF THE GENERAL FORMULA
1, ITS COMPOSITION AND PROCESS FOR PREPARING
THE SAME
02196/DELNP/2003 16-12-2003 243687 29-10-2010 VITAMIN D ANALOGUES AND COMPOSITION GALDERMA RESEARCH &
CONTAINING THE SAME DEVELOPMENT S.N.C
5192/DELNP/2006 11-09-2006 243714 02-11-2010 CONTROLLED-RELEASE PHARMACEUTICAL EISAI R & D MANAGEMENT CO. 
COMPOSITION AND METHOD FOR PRODUCING THE LTD.
SAME
1778/DELNP/2004 22-06-2004 243759 03-11-2010 QUICK RELEASE FLUDARA TABLET COMPOSITION ALCAFLEU MANAGEMENT GMBH & CO.
KG,
2054/DELNP/2003 02-12-2003 243790 08-11-2010 TOPICAL APPLICATION OF THIAZOLYLAMIDES AICURIS GMBH & CO.KG
118/DELNP/2005 13-01-2005 243791 08-11-2010 MULTI-COMPONENT PHARMACEUTICAL CAPSULE FOR GLAXO GROUP LIMITED
RETAINING DRUG SUBSTANCE
IN/PCT/2002/01271/DEL 20-12-2002 243802 08-11-2010 A COMPOSITION USEFUL FOR PROTECTING AGAINST HUNTER-FLEMING LIMITED
ACUTE OR CHRONIC NEURONAL DAMAGE
1133/DELNP/2005 22-03-2005 243822 09-11-2010 A THERAPEUTIC COMPOSITION FOR THE TREATMENT STEROGENE BIOSEPARATIONS, INC.,
OF CANCER
3875/DELNP/2006 05-07-2006 243848 09-11-2010 FORMULATION FOR TREATING OBESITY AND SCANDINAVIAN CLINICAL NUTRITION I
ASSOCIATED METABOLIC SYNDROME SVERIGE AB 
922/MUM/2006 13-06-2006 243835 09-11-2010 HERBAL COMPOSITION FOR RELIEVING PAIN FROM BABULAL BHAWARLAL JAIN
JOINTS AND BONES AND METHOD THEREOF
1326/DELNP/2005 01-04-2005 243859 10-11-2010 PHARAMACEUTICAL COMPOSITION COMPRISING HANMI PHARM CO., LTD
CRYSTALLINE SIBUTRAMINE METHANESUFONATE
HEMIHYDRATE
253/DELNP/2005 24-01-2005 243870 10-11-2010 PYRIMIDYL SULPHONE AMIDE DERIVATIVES AS ASTRAZENECA AB
CHEMOKINE RECEPTOR MODULATORS
2174/DELNP/2005 24-05-2005 243874 10-11-2010 PULVERULENT FORMULATION FOR INHALATION BOEHRINGER INGELHEIM PHARMA
CONTAINING TIOTROPIUM GMBH & CO. KG
1485/DELNP/2005 13-04-2005 243878 10-11-2010 A METHOD FOR MANUFACTURING MEDICAMENT AND INSTITUT PASTEUR AND INSTITUT
A MEDICAMENT THEREOF NATIONAL DE LA SANTE ET DE LA
RECHERCHE MEDICALE
IN/PCT/2002/00758/DEL 02-08-2002 243881 10-11-2010 CONDENSATION DERIVATIVES OF THICOLCHICINE AND INDENA S.P.A.
BACCATIN AS ANTITUMOR AGENTS
746/DELNP/2004 23-03-2004 243912 10-11-2010 A PHARMACEUTICAL COMPOSITION FOR ORAL APOGEPHA ARZNEIMITTEL GMBH
ADMINISTRATION
308/DELNP/2005 27-01-2005 243913 10-11-2010 NOVEL BENZOIMIDAZOLE DERIVATIVES USEFUL AS PFIZER PRODUCTS INC.
ANTIPROLIFERATIVE AGENTS"
90/MUM/2005 28-01-2005 243858 10-11-2010 SYNERGISTIC INJECTABLE COMBINATION OF SANJEEV KHANDELWAL
ANTISPASMODIC AND ANTIPYRETIC - ANALGESIC
IN/PCT/2002/00438/DEL 29-04-2002 243922 11-11-2010 A SOLID ORAL CONTROLLED RELEASED COMPOSITION EURO-CELTIQUE S.A.

301/DELNP/2005 27-01-2005 243930 11-11-2010 ECHINACEA ANGUSTIFOLIA ROOT EXTRACT INDENA S.P.A
COMPOSITION AND PROCESS FOR PREPARATION
THEREOF
182/DELNP/2005 18-01-2005 243957 11-11-2010 A 1H-IMIDAZO[4,5-C] QUINOLINE 4-PHTHALIMIDE TEVA PHARMACEUTICAL WORKS
COMPOUND OF FORMULA (II) AND PROCESS FOR PRIVATE LIMITED COMPANY
PREPARING THE SAME
1268/DEL/2002 17-12-2002 243921 11-11-2010 A MEDICINAL COMPOSITION FOR TREATMENT OF SANDEEP SINGH
HYPOXIA
51/DEL/2001 22-01-2001 243924 11-11-2010 THERAPEUTIC COMPOSITION CONTAINING NIMESULIDE PANACEA BIOTEC LIMITED
AND PROCESS FOR THEIR PREPARATION

542/DEL/2004 22-03-2004 243944 11-11-2010 A MEDICINAL COMPOSTION USEFUL IN TREATMENT OF BANARSI LAL DUA
HIV/AIDS
696/DEL/2004 12-04-2004 243949 11-11-2010 DIMMER OF PHENAZINE-1-CARBOXYLIC ACID AND TO DEPARTMENT OF BIOTECHNOLOGY,
THE PROCESS OF PREPARATION THEREOF
577/DELNP/2003 16-04-2003 243972 12-11-2010 PHARMACEUTICAL COMPOSITION COMPRISING AKL TECHNOLOGIES LIMITED
GINKGOLIDE AND APOCYNIN
29/DELNP/2003 08-01-2003 243999 15-11-2010 BRANCHED-CHAIN LIPOPHILIC COMPOUND, D-PHARM LTD.
PHARMACEUTICAL COMPOSITION AND USES THEREOF

994/DELNP/2005 15-03-2005 244000 15-11-2010 INHALATION COMPOSITIONS WITH HIGH DRUG RATIOS NORTON HEALTHCARE LTD.

996/DELNP/2005 15-03-2005 244005 15-11-2010 INHALATION COMPOSITION NORTON HEALTHCARE LTD


816/DEL/2004 30-04-2004 244027 15-11-2010 A SYNERGISTIC HERBAL COMPOSITION FOR THE PRASAD VAIDYA BANKE
TREATMENT OF ANIMAL BITE ESPECIALLY SNAKE BITE
AND EARLY STAGES OF HYDROPHOBIA.
582/DEL/2003 08-04-2003 244034 15-11-2010 A HERBAL COMPOSITION AGAINST BRONCHIAL THE DIRECTOR, CENTRAL COUNCIL FOR
ASTHMA AND PROCESS FOR PREPARATION THEREOF RESEARCH IN UNANI MEDICINE

1611/DELNP/2003 07-10-2003 244074 16-11-2010 A PHARMACEUTICAL COMPOSITION FOR THE HF ARZNEIMITTELFORSCHUNG GMBH
TREATMENT OF DEFUNCTIONALIZATION
MANIFESTATIONS OR CHRONIC PSYCHIARTIC
SYMPTOMS
313/DELNP/2005 27-01-2005 244095 18-11-2010 BENZIMIDAZOL COMPOUNS BOEHRINGER INGELHEIM PHARMA
GMBH & CO. KG.,
998/DELNP/2006 24-02-2006 244106 18-11-2010 PIPERIDINE COMPOUNDS EURO-CELTIQUE S. A.
601/MUMNP/2005 13-06-2005 244113 18-11-2010 BENZOYLGUANIDINE DERIVATIVES BOEHRINGER INGELHEIM PHARMA
GMBH & CO. KG
796/DEL/2003 11-06-2003 244158 22-11-2010 A FORMULATION FOR DELIVERY OF BIOACTIVE AGENT NATIONAL INSTITUTE OF
PHARMACEUTICAL EDUCATION AND
RESEARCH (NIPER)
1832/DELNP/2003 06-11-2003 244188 23-11-2010 QUICK-DISINTEGRATING TABLET IN THE BUCCAL CAVITY ASTELLAS PHARMA INC.
AND MANUFACTURING METHOD THEREOF
460/DELNP/2005 07-02-2005 244195 23-11-2010 1,2,4-TRIAZOLE DERIVATIVE, METHOD FOR PREPARING CJ CORPORATION
THE SAME, AND PHARMACEUTICAL COMPOSITION
CONTAINING THE SAME
2297/DELNP/2003 31-12-2003 244197 23-11-2010 A COMPOSITION FOR PHARMACOLOGICAL THERAPY OF HF ARZNEIMITTELFORSCHUNG GMBH
NICOTINE DEPENDENCE
475/DEL/1997 25-02-1997 244182 23-11-2010 A PHARMACEUTICAL COMPOSITION COMPRISING AN PFIZER INC.
ESTROGEN AGONIST/ANTAGONIST
5114/DELNP/2006 05-09-2006 244217 24-11-2010 A POWDERY COMPOSITION COMPRISING A STEROIDAL BAYER SCHERING PHARMA
MOLECULE AND A PHARMACEUTICALLY ACCEPTABLE AKTIENGESELLSCHAFT
CARRIER
2530/KOLNP/2006 04-09-2006 244233 25-11-2010 DIPEPTIDYL PEPTIDASE INHBITORS TAKEDA PHARMACEUTICAL COMPANY
LIMITED
855/MUM/2007 03-05-2007 244264 26-11-2010 POTENTIZED FORMULATION OF CAPSAICIN ANALOG RAJESH SHAH

37/DEL/2004 08-01-2004 244306 30-11-2010 4-ARYL-2,6-DIMETHYL-3, 5-DICARBOETHOXY-1, 4- COUNCIL OF SCIENTIFIC AND


DIHYDROPYRIDINES AND CORRESPONDING HYDROXY INDUSTRIAL RESEARCH
DERIVATIVES
2439/KOLNP/2006 28-08-2006 244339 01-12-2010 A THIAZOLE DERIVATIVE TAISHO PHARMACEUTICAL
CO. LTD
IN/PCT/2001/01189/DEL 20-12-2001 244342 01-12-2010 OPTICALLY ACTIVE QUINOLINE CARBOXYLIC ACID EU Biotech Development Ltd.
DERIVATIVES
823/CAL/1999 05-10-1999 244355 02-12-2010 A POLYPHARMACEUTICAL COMPOSITION FOR THE MR. ABDUL MUEED
TREATMENT OF HYPERTENSION
1623/DELNP/2005 21-04-2005 244379 06-12-2010 SUSTAINED RELEASE COMPOSITION FOR ORAL HANMI PHARM. CO., LTD.
ADMINISTRATION OF DRUGS
1434/DELNP/2005 08-04-2005 244381 06-12-2010 MICROSPHERE FOR CONTROLLED RELEASE OF TIANJIN TASLY GROUP CO., LTD.
TEMOZOLOMIDE AND MEHTOD FOR PREPARATION
THEREOF
225/MUMNP/2006 24-02-2006 244464 07-12-2010 STERILE PREPARATIONS OF PHOSPHOLIPIDS AND ANTI- The Board of Regents of the University
INFLAMMATORY PHARMACEUTICALS AND METHODS of Texas System
FOR MAKING AND USING SAME
693/MUMNP/2006 13-06-2006 244465 07-12-2010 OXAZOLIDINONE-QUINOLONE HYBRID ANTIBIOTICS MORPHOCHEM AKTIENGESELLSCHAFT
FUR KOMBINATORISCHE CHEMIE.

557/MUM/2004 14-05-2004 244433 07-12-2010 A CONTROLLED RELEASE DELIVERY COMPOSITION OF CADILA HEALTHCARE LIMITED
METFORMIN
7293/DELNP/2006 04-12-2006 244472 08-12-2010 PHARMACEUTICAL COMPOSITION OF CORTICOSTEROID ALMIRALL  S.A.
AND ANTAAGONIST OF M3 MUSCARINIC RECEPTORS
FOR USE IN THE RESPIRATORY DISORDERS
3668/DELNP/2005 18-08-2005 244474 08-12-2010 A NOVEL (E)-4-CARBOXYSTYRYL-4-CHLOROBENZYL TEMPLE UNIVERSITY - OF THE
SULFONE COMPOUND COMMONWEALTH SYSTEM OF HIGHER
EDUCATION
1682/MUMNP/2007 15-10-2007 244488 08-12-2010 PELLET- TYPE CONTROLLED- RELEASE PREPARATION HENNIG ARZNEIMITTEL GMBH & CO.
CONTAINING CINNARIZINE AND DIMENHYDRINATE FOR KG.
COMBATING VERTIGO
579/MUM/2003 06-06-2003 244479 08-12-2010 AN IMMEDIATE RELEASE FORMULATION OF CADILA HEALTHCARE LIMITED
FLUVASTATIN
22/MUM/2004 09-01-2004 244489 08-12-2010 NOVEL SUBSTITUTED HYDROXAMIC ACID DERIVATIVES CADILA HEALTHCARE LIMITED

5050/DELNP/2006 01-09-2006 244519 09-12-2010 A SYNERGISTIC COMPOSITION FOR REGULATING THE GIULIANI S.P.A.
TROPHISM OF FOLLICLES AND OPTIONALLY THE SKIN
PRODUCTION OF SEBUM
3467/DELNP/2006 16-06-2006 244529 09-12-2010 3-CYANO-QUINOLINE COMPOUNDS AS KINASE JANSSEN PHARMACEUTICA N.V.
INHIBITORS, PHARMACEUTICAL COMPOSITION
THEREOF AND PROCESS FOR PREPARATION
1449/CAL/1997 05-08-1997 244524 09-12-2010 PHARMACEUTICAL COMPOSITION CONTAINING 4- MERCK PATENT GESELLSCHAFT MIT
OXOBUTANOIC ACIDS RESCHRANKTER HAFTUNG
1476/DELNP/2005 13-04-2005 244563 10-12-2010 A NON-EFFERVESCENT TABLET FORMULATION FOR BAYER CONSUMER CARE AG
ORAL ADMINISTRATION OF SODIUM IBUPROFEN
894/MUM/2007 10-05-2007 244558 10-12-2010 HOMEOPATHY BASED FORMULATION FOR TREATMENT RAJESH SHAH
OF LICHEN PLANUS
3719/DELNP/2004 24-11-2004 244635 13-12-2010 A DUAL COMPONENT ANTIPLAQUE ORAL COLGATE-PALMOLIVE COMPANY
COMPOSITION
25/CAL/1998 06-01-1998 244606 13-12-2010 PHARMACEUTICAL COMPOSITION IN THE FORM OF SONUS PHARMACEUTICALS INC
EMULSION MICRO EMULSION OR MICELLAR SOLUTION
FOR DELIVERY OF POORLY SOLUBLE DRUGS

198/MUM/2004 20-02-2004 244585 13-12-2010 NOVEL DRUG DELIVERY SYSTEM TORRENT PHARMACEUTICALS LTD.
838/CAL/1999 12-10-1999 244608 13-12-2010 A POLYPHARMACEUTICAL COMPOSITION FOR THE MR. ABDAL MUEED
TREATMENT OF CORYZA CATARRH POLYPUS TONSILS,
HEADACHE MIGRAINE APTHAE THRUSH SPRUE
GLOSSITIS ITCHING AND PUSTULES
2056/MUM/2006 15-12-2006 244626 13-12-2010 STABLE DUAL RELEASE PHARMACEUTICAL TABLET IPCA LABORATORIES LIMITED
COMPRISING METOPROLOL AND CHLORTHALIDONE

3536/KOLNP/2006 27-11-2006 244638 14-12-2010 HISTAMINE H3 RECEPTIOR AGENTS, PREPARATION AND ELI LILLY AND COMPANY
THERAPEUTIC USES
4710/KOLNP/2007 05-12-2007 244647 14-12-2010 A SUBSTITUTED TETRAHYDROCARBAZOLE COMPOUND ELI LILLY AND COMPANY
USEFUL AS ANDROGEN RECEPTOR MODULATORS
(SARM) AND PHARMACEUTICAL COMPOSITION
THEREOF
5917/DELNP/2005 19-12-2005 244662 15-12-2010 A TOPICAL COMPOSITION FOR THE TREATMENT OF POLICHEM S.A
ONYCHOSCHIZIA
1010/KOLNP/2006 20-04-2006 244695 15-12-2010 AQUEOUS SOLUTION PREPARATION CONTAINING SENJU PHARMACEUTICAL CO., LTD.
AMINOGLYCOSIDE ANTIBIOTIC AND BROMFENAC
472/DELNP/2005 08-02-2005 244698 15-12-2010 A PHARMACEUTICAL FORMULATION IN THE FORM OF BRISTOL-MYERS SQUIBB COMPANY
AN INCLUSION COMPLEX
IN/PCT/2001/00453/DEL 31-05-2001 244699 15-12-2010 AN IMPROVED COMPOSITION OF A DRUG MALIREDDY S. REDDY
1012/MUM/2005 26-08-2005 244675 15-12-2010 NOVEL DRUG DELIVERY SYSTEM TORRENT PHARMACEUTICALS LIMITED

1397/DELNP/2003 01-09-2003 244724 17-12-2010 A DELAYED RELEASE ORAL SOLID COMPOSITION PENWEST PHARMACEUTICALS CO
569/DELNP/2003 16-04-2003 244734 17-12-2010 A PHARMACEUTICAL COMPOSITION COMPRISING FOURNIER LABORATORIES IRELAND
PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR LIMITED
(PPAR) AND COENZYME Q10.
IN/PCT/2002/00622/DEL 19-06-2002 244741 17-12-2010 COMPOUNDS SPECIFIC TO ADENOSINE A1 A2 AND A3, OSI PHARMACEUTICAL INC.
RECEPTORS AND USES THEREOF
3306/KOLNP/2006 10-11-2006 244780 20-12-2010 A CYCLIC AMIDE COMPOUND AND A COMPOSITION TAKEDA PHARMACEUTICAL COMPANY
COMPRISING THE SAME LIMITED
301/DELNP/2003 05-03-2003 244794 20-12-2010 SULFONAMIDE DERIVATIVES BEARING BOTH LIPOPHILIC APPLIED RESEARCH SYSTEMS ARS
AND IONISABLE MOIETIES AS INHIBITOR OF PROTEIN HOLDING N.V
JUNKINASES
196/DELNP/2005 19-01-2005 244809 21-12-2010 SUSTAINED RELEASE FORMULATIONS COMPRISING GLAXO GROUP LIMITED
LAMOTRIGINE
680/DELNP/2005 21-02-2005 244827 21-12-2010 NUCLEOSIDE ANALOG COMPOUND ALBERT EINSTEIN COLLEGE OF
MEDICINE OF YESHIVA UNIVERSITY
6238/DELNP/2006 25-10-2006 244837 21-12-2010 4-PHENYLAMINO-QUINAZOLIN-6-YL-AMIDES AND A WARNER -LAMBERT COMPANY
PHARMACEUTICAL COMPOSITION COMPRISING THE LLC 
SAME
1739/DELNP/2003 23-10-2003 244886 23-12-2010 4-ANILINOQUINOLINE-3-CARBOXAMIDE OF THE ASTRA ZENECA AB
FORMULA I (A)
911/MUM/2005 05-08-2005 244866 23-12-2010 TOPICAL PHARMACEUTICAL COMPOSITIONS GLENMARK PHARMACEUTICALS
CONTAINING ADAPALENE AND CLINDAMYCIN LIMITED
IN/PCT/2002/00340/DEL 28-03-2002 244925 27-12-2010 FORMULATION FOR MENOPAUSAL WOMEN DRUGTECH CORPORATION
812/KOLNP/2006 04-04-2006 244997 28-12-2010 MODAFINIL MODIFIED RELEASE PHARMACEUTICAL CEPHALON, INC
COMPOSITIONS
2982/CHENP/2006 14-08-2006 245016 29-12-2010 GLP-1 ANALOGUES SOCIETE DE CONSEILS DE RECHERCHES
ET D"APPLICATIONS SCIENTIFIQUES SAS

1341/CHE/2005 21-09-2005 245033 29-12-2010 DERIVATIVES OF 4,6-DISUBSTITUTED 1,2,4- TRIAZOLO- JAWAHARLAL NEHRU CENTRE FOR
1,3,4-THIADIAZOLE, A PROCESS AND USES THEREOF ADVANCED SCIENTIFIC RESEARCH

756/KOLNP/2006 29-03-2006 245052 30-12-2010 CONDENSED RING COMPOUND AND USE THEREOF ONO PHARMACEUTICAL CO., LTD.
984/CHENP/2005 20-05-2005 245117 03-01-2011 COMPOSTION COMPRISING A CHEMOTHERAPEUTIC M/S. THE BOARD OF TRUSTEES OF THE
AGENT AND AN ENDOTHELIN B AGONIST. UNIVERSITY OF ILLINOIS

688/DELNP/2006 10-02-2006 245128 04-01-2011 A SUBSTITUTED QUINAZOLINE COMPOUND INCLUDING ARRY BIOPHARMA, INC.
RESOLVED ENANTIOMERS,DIASTEREOMERS,AND
PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF

4781/DELNP/2005 19-10-2005 245131 04-01-2011 N-[1-(3-CHLORO-1-NAPHTHALENYL)ETHYL]-2-[4-(4- GLAXO GROUP LIMITED


FLUOROPHENYL)-1-METHYL-4-PIPERIDINYL]-N-
METHYLACETAMIDE OR A PHARMACEUTICALLY
ACCEPTABLE SALT THEREOF, ITS COMPOSITION AND
PROCESS FOR PREPARING THE SAME
1578/DELNP/2004 07-06-2004 245132 04-01-2011 NITROGEN-CONTAINING HETEROARYL DERIVATIVES BTG INTERNATIONAL LTD.,
3710/DELNP/2004 24-11-2004 245171 06-01-2011 A COMPOSITIONS FOR LOWERING INTRAOCULAR ALCON, INC
PRESSURE AND PROVIDING NEUROPROTECTIOIN IN A
PATIENT IN NEED THEREOF
6740/DELNP/2006 14-11-2006 245187 06-01-2011 CINNAMIDE COMPOUND EISAI R&D MANAGEMENT CO., LTD
2605/DELNP/2006 09-05-2006 245196 06-01-2011 RADIOLABELED 3,7-BIS [2-(4-NITRO [3,5-3H] PHENYL) ASTRAZENECA AB
ETHYL] -3,7-DIAZABICYCLO [3,3,1] NONANE

1295/DELNP/2003 14-08-2003 245212 07-01-2011 PHARMACEUTICAL COMPOSITIION CONTAINING ONE BOEHRINGER INGELHEIM PHARMA
OR MORE TIOTROPIUM SALTS GMBH & CO. KG.
IN/PCT/2002/00728/DEL 29-07-2002 245257 11-01-2011 SULFONAMIDE COMPOUNDS THAT MODULATE THE TEXAS BIOTECHNOLOGY CORPORATION
ACTIVITY OF ENDOTHELIN
281/DELNP/2005 25-01-2005 245306 13-01-2011 A PHARMACEUTICAL COMPOSITION FOR INHIBITING HELIX BIOPHARMA CORP.
GROWTH OF CANCER CELLS
709/DELNP/2005 22-02-2005 245310 13-01-2011 N-PYRID-2YL,N'-4,7-DI-HALO- MEDIVIR AB
TETRAHYDROCYCLOPROPA (-C-) CHROMEN-1-YL(THIO)
UREA COMPOUNDS OF THE FORMULA U
291/DELNP/2005 25-01-2005 245335 13-01-2011 A COMPOSITION COMPRISING A SYNERGISTIC RATIO OF PFIZER INC.
AN ALPHA-2-DELTA LIGAND AND A PDEV INHIBITOR

344/DELNP/2005 28-01-2005 245337 13-01-2011 A 2'-C-METHYL-RIBOFURANOSYL CYTIDINE-3'-O-L- IDENIX (CAYMAN) LIMITED


VALINE ESTER COMPOUND
654/DELNP/2005 18-02-2005 245339 13-01-2011 A NOVEL CYTOTOXIC LINKABLE TAXANE COMPOUND IMMUNOGEN, INC

560/DELNP/2005 14-02-2005 245340 13-01-2011 AQUEOUS PHARMACEUTICAL COMPOSITION FOR BOEHRINGER INGELHEIM PHARMA
INHALATION GMBH & CO. KG
108/DELNP/2005 12-01-2005 245350 14-01-2011 1 2-CYANO-4-FLUOROPYRROLIDINE DERIVATIVE" ASTELLAS PHARMA INC.
678/MUMNP/2005 27-06-2005 245363 17-01-2011 ORALLY ADMINISTRABLE PREPARATION BAYER SCHERING PHARMA
AKTIENGESELLSCHAFT
207/DELNP/2005 19-01-2005 245368 17-01-2011 PHARMACEUTICAL COMPOSITION FOR TRANSDERMAL ACRUX DDS PTY.LTD.
DELIVERY
1136/DELNP/2005 22-03-2005 245372 17-01-2011 A PHARMACEUTICAL COMPOUND AND COMPOSITION BAUSCH & LOMB INCORPORATED
THEREOF
419/DELNP/2005 03-02-2005 245396 18-01-2011 A SUSTAINED RELEASE BICIFADINE COMPOSITION NASCIME LIMITED
123/DELNP/2005 13-01-2005 245400 18-01-2011 COMPOSITION FOR TOPICALLY TREATING SEBORRHEIC PARKS, L., DEAN
DERMATITIS
214/DELNP/2005 19-01-2005 245401 18-01-2011 AN ORALLY CONSUMABLE FILM COMPOSITION FOR COLGATE-PALMOLIVE COMPANY
DELIVERING BREATH FRESHENING AGENTS TO THE
ORAL CAVITY
1029/DELNP/2005 16-03-2005 245410 18-01-2011 A PHARMACEUTICAL COMPOSITION COMPRISING A WYETH
HUMAN INTERLEUKIN-11(IL-11')POLYPEPTIDE"
IN/PCT/2002/01202/DEL 05-12-2002 245422 19-01-2011 PHARMACEUTICAL COMPOSITIONS CONTAINING D-PHARM LTD.
PHOSPHOLIPID DERIVATIVES OF VALPROIC ACIDS"
IN/PCT/2002/00852/DEL 28-08-2002 245424 19-01-2011 PYRROLOPYRIMIDONE DERIVATIVES AND PROCESS OF S.K. CHEMICALS CO., LTD.
PREPARATION THEREOF
3677/DELNP/2005 19-08-2005 245428 19-01-2011 A FACTOR VIII COMPOSITION BAXTER INTERNATIONAL INC.
2052/DELNP/2005 13-05-2005 245431 19-01-2011 TIZANIDINE COMPOSITION TEVA PHARMACEUTICAL INDUSTRIES
LTD.
1752/DELNP/2005 29-04-2005 245446 19-01-2011 A PHARMACEUTICAL COMPOSITION COMPRISING NEUROPHARMACOLOGY SERVICES,LLC.
OXYTOCIN
1708/DELNP/2005 27-04-2005 245448 19-01-2011 PYRIDOPYRROLIZINE AND PYRIDOINDOLIZINE MERCK FROSST CANADA & CO.
DERIVATIVES
1633/DELNP/2005 21-04-2005 245450 19-01-2011 PHENYLNAPHTHALENE COMPOUNDS AND LES LABORATOIRES SERVIER
PHARMACEUTICAL COMPOSITION THEREOF
5949/DELNP/2005 20-12-2005 245452 20-01-2011 COMPOUNDS FOR TREATING OCULAR HYPERTENSION MERCK & CO.INC.
AND COMPOSITIONS THEREOF
1090/DELNP/2005 21-03-2005 245455 20-01-2011 6-METHYL-2[4-(4--MORPHOLINO) ANILINO] NICOTINIC B & C BIOPHARM
ACID AND METHOD FOR PREPARING THEREOF

1139/DELNP/2005 23-03-2005 245458 20-01-2011 AN INJECTABLE EMULSION FORMULATION OF A BAXTER INTERNATIONAL INC.
VOLATILE ANESTHETIC
1361/DELNP/2005 05-04-2005 245460 20-01-2011 AN ASIALO-INTERFERON PHARMACEUTICAL THE GENERAL HOSPITAL CORPORATION
COMPOSITION
1420/DELNP/2005 07-04-2005 245492 21-01-2011 NOVEL QUINOLYLPROPYLPIPERIDINE COMPOUNDS AND NOVEXEL
PROCESS FOR PREPARATION THEREOF
2224/DELNP/2004 30-07-2004 245502 21-01-2011 CARBAMOYL SUBSTITUTED COMPOUNDS USEFUL TANABE SEIYAKU CO. LTD
FORαLß2 INHIBITION OF INTEGRIN MEDIATED
CELL ADHESION
99/KOLNP/2007 09-01-2007 245570 25-01-2011 OXAZOLE DERIVATIVES AS HISTAMINE H3 RECEPTOR ELI LILLY AND COMPANY
AGENTS, PREPARATION AND THERAPEUTIC USES

2093/DELNP/2005 17-05-2005 245573 25-01-2011 A 3,5 SUBSTITUTED OXAZOLIDINONE COMPOUND OF ASTRAZENECA AB


THE FORMULA (I)
751/DELNP/2005 24-02-2005 245578 25-01-2011 A 3-(SULFONAMIDOETHYL)-INDOLE COMPOUND AND A BOEHRINGER INGELHEIM
METHOD OF MAKING FORMULA (I) PHARMACEUTICALS INC.
2090/DELNP/2005 17-05-2005 245583 25-01-2011 A CONTROLLED RELEASE TABLET CONTAINING CILAG AG
TOPIRAMATE, TRAMADOL HYDROCHLORIDE AND
XANTHAN GUM
2007/DELNP/2004 13-07-2004 245611 27-01-2011 AN OSMOTIC PHARMACEUTICAL TABLET PFIZER PRODUCTS INC
2918/DELNP/2004 28-03-2004 245616 27-01-2011 AN INDAZOL COMPOUND JNK INHIBITOR EISAI R&D MANAGEMENT CO., LTD
1871/KOLNP/2007 25-05-2007 245644 28-01-2011 A COMPOUND OF FORMULA (I) AND A COMPOSITION ELI LILLY AND COMPANY
USED AS ALLOSTERIC POTENTIATORS OF THE M4
MUSCARINIC RECEPTOR

1073/DELNP/2003 08-07-2003 245684 28-01-2011 A GELDANAMYCIN DERIVATIVE THE UNITED STATES OF AMERICA,
REPRESENTED BY THE SECRETARY,
DEPARTMENT OF HEALTH AND HUMAN
SERVICES
IN/PCT/2002/01240/DEL 13-12-2002 245685 28-01-2011 A COMPOUND OF THE 3`-O-VALINYL ESTER OF 2`- IDENIX (CAYMAN) LIMITED
DEOXY-[BETA]-L-CYTIDINE
3501/DELNP/2004 09-11-2004 245725 31-01-2011 A HERBAL COMPOSITION USEFUL FOR GASTRO- COUNCIL OF SCIENTIFIC & INDUSTRIAL
INTESTINAL DISORDERS & PROCESS THEREOF RESEARCH.
910/CHE/2005 08-07-2005 245780 01-02-2011 NOVEL BIO-ACTIVE DERIVATIVES ORCHID CHEMICALS &
PHARMACEUTICALS LTD
318/KOLNP/2007 29-01-2007 245805 02-02-2011 VAGINAL RING CONTAINING PROGESTERONE THE POPULATION COUNCIL, INC.
RECEPTOR MODULATORS
1154/DEL/2001 16-11-2001 245820 02-02-2011 NOVEL DIALLYLDISULPHIDE COMPOUNDS HAVING DEPARTMENT OF SCIENCE AND
ANTILIPIDEMIC AND ANTIOXIDANT ACTIVITY TECHNOLOGY
1501/MUMNP/2006 07-12-2006 245843 03-02-2011 A PHARMACEUTICAL COMPOSITION COMPRISING BOEHRINGER INGELHEIM PHARMA
TIOTROPIUM AND FORMOTEROL GMBH & CO. KG.
1124/MUM/2004 20-10-2004 245846 03-02-2011 SEDATIVES LOADED INTRANASAL NASOADHESIVE AMBIKANANDAN MISRA
MICROEMULSIONS FOR BRAIN TARGETED DELIVERY IN
INSOMNIA
843/CHE/2006 12-05-2006 245854 03-02-2011 NOVEL THROMBOLYTIC MOLECULES AND A PROCESS BHARAT BIOTECH INTERNATIONAL
THEREFOR LIMITED
2543/DELNP/2005 13-06-2005 245887 04-02-2011 A COMPOSITION FOR TREATING PERSONS SUFFERING ALCON, INC.
FROM ACUTE OR CHRONIC DEGENERATIVE
CONDITIONS OR DISEASES OF THE EYE

3220/DELNP/2005 20-07-2005 245920 07-02-2011 PHARMACEUTICAL COMPOSITION USEFUL AGAINST CENTRO DE INGENIERIA GENETICA Y
NEOPLASIA BIOTECNOLOGIA
3029/DELNP/2005 06-07-2005 245936 07-02-2011 A LACTOFERRIN COMPOSITION FOR TREATING AGENNIX INCORPORATED
BACTEREMIA OR SEPSIS
3254/DELNP/2005 22-07-2005 245943 07-02-2011 COMPOSITION FOR PREVENTIVE TREATMENT OF COLD PRONOVA MEDICAL B.V.
SORES
3481/DELNP/2004 09-11-2004 245978 08-02-2011 COMPOSITION, FORMULATIONS & KIT FOR TREATMENT EPIGENESIS PHARMACEUTICALS, LLC.
OF RESPIRATORY & LUNG DISEASE WITH
DEHYDROEPIANDROSTERONE(S) STEROID & AN ANTI-
MUSCARINIC AGENT(S)
6091/DELNP/2005 27-12-2005 245986 09-02-2011 MODIFIED-RELEASE COMPOSITION BIOVAIL LABORATORIES
INTERNATIONAL SRL.
2139/KOLNP/2006 28-07-2006 246005 09-02-2011 NOVEL INHIBITORS OF GLUTAMINYL CYCLASE PROBIODRUG AG
935/KOLNP/2006 13-04-2006 246008 09-02-2011 COMPOSITIONS USEFUL AS INHIBITORS OF PROTEIN VERTEX PHARMACEUTICALS
KINASES INCORPORATED
232/DELNP/2004 03-02-2004 246010 09-02-2011 ANTITUMORAL ANALOGUES OF ECTEINASCIDIN PHARMA MAR, SA.
IN/PCT/2002/00703/DEL 16-07-2002 246021 09-02-2011 A COMPOSITION USEFUL AGAINST ASEPTIC HU, SHIQING
INFLAMMMATIONS AND STUBBORN PAINS
372/DELNP/2003 12-03-2003 246112 15-02-2011 17-METHYLENE STEROIDS, PROCESS FOR THEIR SCHERING AKTIENGESELLSCHAFT
PRODUCTION AND PHARMACEUTICAL COMPOSITIONS
THAT CONTAIN THESE COMPOUNDS
5042/DELNP/2005 03-11-2005 246115 15-02-2011 HETEROARYL AMIDE DERIVATIVES AND THEIR USE AS ASTRAZENECA AB
P2X<sub>7</sub> , RECEPTOR ANTAGONISTS
1301/KOLNP/2006 17-05-2006 246121 15-02-2011 DUAL MOLECULES CONTAINING PEROXY DERIVATIVE, CENTRE NATIONAL DE LA RECHERCHE
THE SYNTHESIS SCIENTIFIQUE
1125/KOLNP/2007 02-04-2007 246133 15-02-2011 HALOGENATED BENZAMIDE DERIVATIVES ROMARK LABORATORIES, L.C.
2037/DELNP/2006 13-04-2006 246159 17-02-2011 A COMPOUND OF FORMULA (I) FOR USE AS PFIZER INC.
MEDICAMENT
252/MUM/2007 09-02-2007 246147 17-02-2011 A PHARMACEUTICAL COMPOSITION AND A PROCESS INDUS BIOTECH PRIVATE LIMITED
THEREOF
1588/DEL/1998 10-06-1998 246186 18-02-2011 A 4 -SUBSTITUED-9-DEOXO-9A-AZA-9A- PFIZER PRODUCTS INC.
HOMOERYTHROMYCIN A COMPOUND"
3827/DELNP/2004 02-12-2004 246195 21-02-2011 PHARMACEUTICAL COMPOSITION AND PROCESS OF INSIGNION HOLDINGS LIMITED
PREPRATION THEREOF
828/KOLNP/2006 05-04-2006 246198 21-02-2011 2,4-DIOXO-3-QUINAZOLINYL SULFONYLUREAS PORTOLA PHARMACEUTICALS, INC.
1428/DELNP/2005 07-04-2005 246202 21-02-2011 A GLP-2 PEPTIDE AND PHARMACEUTICAL NOVA NORDISK A/S
COMPOSITION THEREOF
4753/DELNP/2005 19-10-2005 246215 21-02-2011 AN ARYL AMINOTHIAZOLE COMPOUND NEUROGENETIC PHARMACEUTICALS ,
INC.
1594/DELNP/2004 08-06-2004 246226 22-02-2011 HYDRAZONOPYRAZOLE DERIVATIVES AND THEIR USE AS KINETEK PHARMACEUTICALS INC
THERAPEUTICS
3736/DELNP/2006 29-06-2006 246229 22-02-2011 A PARENTERAL PHARMACEUTICAL COMPOSITION PFIZER PRODUCTS INC.
1241/DELNP/2005 30-03-2005 246249 22-02-2011 A COMPOUND OF FORMULA (I) OR ASTRAZENECA AB
PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF
5369/DELNP/2005 23-11-2005 246279 23-02-2011 BETA-STRAND MIMETICS AND METHODS RELATING CHOONGWAE PHARMA CORPORATION
THERETO
1872/KOLNP/2007 25-05-2007 246285 23-02-2011 AN AMIDE OF COMPOUND 2-DEOXY-2, 2- ELI LILLY AND COMPANY
DIFLUOROCYTIDINE AND PHARMACEUTICAL
COMPOSITION THEREOF
2713/DEL/2006 19-12-2006 246278 23-02-2011 PHARMACEUTICAL COMPOSITION LES LABORATOIRES SERVIER
172/DELNP/2007 08-01-2007 246305 24-02-2011 BIS(THIO-HYDRAZIDE AMIDE) SALTS FOR TREATMENT SYNTA PHARMACEUTICALS CORP
OF CANCERS, PHARMACEUTICAL COMPOSITION AND
METHOD OF PREPARATION THEREOF

961/CHENP/2004 05-05-2004 246323 24-02-2011 CYCLOOXYGENASE -2 INHIBITOR/HISTONE NOVARTIS AG


DEACETYLASE INHIBITOR COMBINATION
402/CHENP/2004 27-02-2004 246328 24-02-2011 AN AEROSOL SUSPENSION FORMULATION FOR SCHERING CORPORATION
INHALATION
7329/DELNP/2006 05-12-2006 246335 24-02-2011 A PHARMACEUTICAL COMPOSITION SUITABLE FOR USE ALMIRALL&nbsp; S.A.
IN THE RESPIRATORY DISORDERS COMPRISING PDE4
INHIBITORS AND ANTAGONIST OF M3 MUSCARINIC
RECEPTORS
IN/PCT/2002/00749/DEL 01-08-2002 246355 25-02-2011 A SYNERGISTIC PHARMACEUTICAL COMPOSITION AVENTIS PHARMA S.A.
COMPRISING A COMBINATION OF CAMPTOTHECIN
WITH CAPECITABINE
1748/DELNP/2003 27-10-2003 246359 25-02-2011 A NOVEL COMPOUND HAVING CORTICOTROPIN- EISAI R & D MANAGEMENT CO. LTD
RELEASING FACTOR RECEPTOR ANTAGONISTIC
ACTIVITY, SALTS THEREOF AND HYDRATES OF THE
FOREGOING
IN/PCT/2002/00724/DEL 24-07-2002 246366 25-02-2011 A TWO COMPONENT EFFERVESCENT DENTIFRICE COLGATE-PALMOLIVE COMPANY
COMPOSITION AND METHOD THEREOF
263/CHENP/2006 20-01-2006 246396 25-02-2011 HEPARIN-DERIVED OLIGOSACCHARIDE MIXTURES, AVENTIS PHARMA S.A.
PREPARATION THEREOF AND PHARMACEUTICAL
COMPOSITIONS CONTAINING SAID MIXTURES
IN/PCT/2002/00262/MUM 04-03-2002 246466 28-02-2011 A GRANULE FORMULATION AND A PROCESS FOR ASTRAZENECA AB
PREPARING THE SAME
1515/DELNP/2005 15-04-2005 246467 01-03-2011 A BAICALEIN DERIVATIVE JENKEN BIOSCIENCES,INC.
250/DELNP/2005 24-01-2005 246481 01-03-2011 HETERO BIARYL COMPOUNDS WARNER-LAMBERT COMPANY LLC
1376/DELNP/2005 05-04-2005 246487 01-03-2011 A COMPOUND N-ALKYNYL-2-ALKOXY-2-(SUBSTITUTED SYNGENTA LIMITED
PHENOXY ALKYLAMIDES) OF GENERAL FORMULA (I)
AND PHARMACEUTICAL COMPOSITION THEREOF

208/DELNP/2005 19-01-2005 246494 01-03-2011 PHARMACEUTICAL COMPOSITION FOR TRANSDERMAL CRUX DDS PTY. LTD.
DELIVERY OF PHYSIOLOGICALLY ACTIVE AGENT

1025/DEL/2003 19-08-2003 246484 01-03-2011 A NOVEL CONTROLLED RELEASE FORMULATION OF NATIONAL INSTITUTE OF
AZITHROMYCIN PHARMACEUTICAL EDUCATION AND
RESEARCH (NIPER)
1201/CHENP/2006 06-04-2006 246515 02-03-2011 METHYLPHENIDATE SOLUTION AND ASSOCIATED MALLINCKRODT INC.
METHODS OF ADMINISTRATION AND PRODUCTION

917/CHE/2006 29-05-2006 246524 02-03-2011 2-(2-AMINO-1, 6-DIHYDRO-6-OXO-PURIN-9-YL) F. Hoffmann-La Roche AG


METHOXY-1, 3-PROPANEDIOL DERIVATIVE
1399/DELNP/2003 01-09-2003 246558 04-03-2011 A DELAYED RELEASE ORAL SOLID COMPOSITION PENWEST PHARMACEUTICALS CO.
2849/DELNP/2004 23-09-2004 246560 04-03-2011 A B-AMINO ACID OF FORMULA IA AND COMPOSITIONS WARNER-LAMBERT COMPANY LLC
THEREOF
3160/DELNP/2004 13-10-2004 246574 04-03-2011 SUSTAINED RELEASE COMPOSITION FOR TREATING APOTEX INC
IRON INDUCED CARDIAC DISEASE
2720/DELNP/2004 15-09-2004 246581 04-03-2011 COMPOUND OF FORMULA (I) AS TROPANE PFIZER INC.
DERIVATIVES
IN/PCT/2002/00135/DEL 31-01-2002 246584 07-03-2011 PHENOXYPROPIONIC ACID ALKOXYCARBONYL ANILID DONBU HANNONG CHEMICAL CO.,LTD
COMPOUNDS AND PREPARATION THEREOF
3401/KOLNP/2006 17-11-2006 246620 08-03-2011 COMPOUNDS FOR TREATING DYSLIPIDEMIA ELI LILLY AND COMPANY
1327/CHENP/2007 30-03-2007 246642 08-03-2011 2-AMINOPYRIDINE COMPOUNDS USEFUL AS BETA- MERCK & CO INC
SECRET ASE INHIBITORS FOR THE TREATMENT OF
ALZHEMER'S DISEASE
1363/DELNP/2005 05-04-2005 246655 09-03-2011 ALKENYL ESTERS OF AMINO SUBSTITUTED ALKONIC YEDA RESEARCH AND DEVELOPMENT
ACID CO. LTD.
766/CHENP/2007 22-02-2007 246671 10-03-2011 ACIDIC SOLID ORAL COMPOSITIONS WITHOUT EROSIVE TOMS GRUPPEN A/S
POTENTIAL IN SALIVA AND METHOD FOR REDUCTION
OF EROSIVE POTENTIAL IN SALIVA
647/KOLNP/2003 20-05-2003 246761 15-03-2011 AEROGEL POWDER AND A PROCESS FOR ASPEN AEROGELS, INC.
MANUFACTURING IT
423/KOLNP/2003 08-04-2003 246771 15-03-2011 A METHOD OF PREPARING A COMPOSITION OF CEPHALON INC
PARTICLES, AND THE COMPOSITION THEREOF
1256/DEL/2005 16-05-2005 246763 15-03-2011 NEW PYROOLIDINE AND THIAZOLIDINE COMPOUNDS, A LES LABORATOIRES SERVIER
PROCES FOR THEIR PREPARATION AND
PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

1034/KOLNP/2006 21-04-2006 246789 16-03-2011 BENZIMIDAZOLE DERIVATIVES : PREPARATION AND S*BIO PTE LTD.
PHARMACEUTICAL APPLICATIONS
1826/KOLNP/2006 30-06-2006 246799 16-03-2011 A SOFT CAPSULE OF BUTYLPHTHALIDE SHIJIAZHUANG PHARMA. GROUP
ZHONGQI PHARMACEUTICAL
TECHNOLOGY (SHIJIAZHUANG) CO.,
LTD.
1411/CHENP/2005 24-06-2005 246807 16-03-2011 1,2,4-TRIAMINOBENZENE DERIVATIVES USEFUL FOR H. LUNDBECK A/S
TREATING DISORDERS OF THE CENTRAL NERVOUS
SYSTEM
115/KOL/2008 16-01-2008 246818 16-03-2011 PHARMACEUTICAL COMPOSITION FOR THE DEVELOPMENT CENTER FOR
TREATMENT OF RHEUMATOIDARTHRITIS BIOTECHNOLOGY
1885/CHENP/2006 29-05-2006 246853 17-03-2011 ANGIOGENIC PEPTIDES RAMOT AT TEL AVIV UNIVERSITY LTD.
6802/DELNP/2006 15-11-2006 246923 22-03-2011 2-PYRIDYL SUBSTITUTED IMIDAZOLE COMPOUND AS SK CHEMICALS CO.LTD
ALK5 ALK4 INHIBITORS AND A COMPOSITION THEREOF

01281/DELNP/2003 13-08-2003 246948 22-03-2011 CIS-1(5-CYANO-PYRIDIN-2-YL)-3-(4,7-DIFLUORO- MEDIVIR AB


1,1A,2,7B-TETRAHYDRO CYCLOPROPA[C]CHROMEN-1-
YL)-UREA OF FORMULA 1
2098/DELNP/2005 17-05-2005 246952 23-03-2011 A PHARMACEUTICAL COMPOSITION COMPRISING BIOMARIN PHARMACEUTICAL INC.
PRECURSOR HUMAN N-ACETYLGALACTOSAMINE-4-
SULFATASE
1759/DELNP/2004 21-06-2004 246961 23-03-2011 ORAL PHARMACEUTICAL COMPOSITION FOR UCB FARCHIM SA
IMPROVING PALATABILITY AND AVOIDING UNDESIRED
REACTION PRODUCTS CONTAINING AT LEAST TWO
SEPARATE FORMULATIONS
796/KOLNP/2006 03-04-2006 246966 23-03-2011 FUSED PENTACYCLIC POLYETHERS UNIVERSITY OF NORTH CAROLINA AT
WILMINGTON
719/DELNP/2005 22-02-2005 247029 25-03-2011 PHARMACEUTICAL FORMULATION COMPRISING PATEL SATISHCHANDRA
CYCLOSPORIN PROPYLENE GLYCOL ESTER AND NON- PUNAMBHAI,27 YALE
IONIC SURFACTANT COURT,LIVINGSTON,NEW JERSEY
07039,U.S.A
1133/CHENP/2006 03-04-2006 247041 25-03-2011 DRUG CONTAINING (2R)-2-PROPYLOCTANOIC ACID AS ONO PHARMACEUTICAL CO., LTD.
THE ACTIVE INGREDIENT
1511/MUM/2006 21-09-2006 247054 26-03-2011 SUSTAINED RELEASE ANTI-EPILEPTIC COMPOSITIONS INVENTIA HEALTHCARE PRIVATE
LIMITED
3511/KOLNP/2006 24-11-2006 247064 28-03-2011 GLUCAGON RECEPTOR ANTAGONISTS AND ELI LILLY AND COMPANY
PHARMACEUTICAL COMPOSITION THEREOF
1099/KOLNP/2004 03-08-2004 247070 28-03-2011 A 2,4,6 - TRIAMINE-1,3,5-TRIAZINE ASTELLAS PHARMA INC.
2906/DELNP/2006 22-05-2006 247072 28-03-2011 IMIDAZOLE DERIVATIVES UCB&nbsp;S.A
210/DELNP/2005 19-01-2005 247093 28-03-2011 PHARMACEUTICAL COMPOSITION FOR TRANSDERMAL ACRUX DDS PTY. LTD.
DELIVERY RATE CONTROL OF PHYSIOLOGICALLY ACTIVE
AGENT USING AMORPHOUS DEPOSIT

1990/DELNP/2005 10-05-2005 247096 28-03-2011 A PHARMACEUTICAL COMPOUND FOR TREATING TARO PHARMACEUTICAL INDUSTRIES
MOVEMENT DISORDERS LIMITED
811/KOLNP/2005 04-05-2005 247104 28-03-2011 N-SUBSTITUTED CARBAMATE META-BIPHENYL ESTER THE REGENTS OF THE UNIVERSITY OF
AS NOVEL FATTY ACID AMIDE HYDROLASE INHIBITORS CALIFORNIA

1885/KOLNP/2006 06-07-2006 247116 28-03-2011 DERIVATIVES OF N-' (1,5-DIPHENYL-1 H-PYRAZOL-3-YL) SANOFI-AVENTIS


SUPHONAMIDE WITH CB1 RECEPTOR AFFINITY
2621/KOLNP/2005 19-12-2005 247151 29-03-2011 AN ORAL PHARMACEUTICAL COMPOSITION UNITED THERAPEUTICS CORPORATION
6026/DELNP/2005 23-12-2005 247176 29-03-2011 A CONJUGATE MOLECULE CONSISTING OF AN OLIGO- INSTITUT PASTEUR
OR POLYSACCHARIDE
978/DEL/2004 28-05-2004 247177 29-03-2011 AN AZITHROMYCIN COMPOSITION PFIZER PRODUCTS INC.
2347/DELNP/2006 27-04-2006 247226 30-03-2011 SPIROCYCLIC HETEROCYLIC COMPOUND ADOLOR CORPORATION
2103/MUM/2006 22-12-2006 247344 31-03-2011 ( 1-H-PYRAZOL-1-YL)ALKYLAMINE COMPOUNDS OF AVENTIS PHARMA S.A.
FORMULA (III)
1279/MUM/2005 11-10-2005 247285 31-03-2011 NOVEL ANTI-MALARIAL COMBINATION AND METHODS IPCA LABORATORIES LTD.
OF FORMULATION
83/MUM/2006 18-01-2006 247313 31-03-2011 MODIFIED RELEASE ORAL DOSAGES FORM USING CO- ASTRON RESEARCH LIMITED
POLYMER OF POLYVINYI ACETATE
1125/MUM/2004 20-10-2004 247325 31-03-2011 DRUGS LOADED INTRANASAL NASOADHESIVE AMBIKANANDAN MISRA
MICROEMULSIONS FOR BRAIN TARGETED DELIVERY IN
MIGRAINE
1269/CHENP/2006 13-04-2006 247373 04-04-2011 A COMPOSITION FOR ASSISTING MUCUS CLEARANCE IN VECTURA LIMITED
THE RESPIRATORY TRACT
00590/DELNP/2004 09-03-2004 247381 04-04-2011 A NOVEL COMPOUND OF FORMULA (1) BRISTOL - MYERS SQUIBB COMPANY
1882/KOLNP/2006 06-07-2006 247403 05-04-2011 SUBSITUTED PIPERAZINES CHEMOCENTRYX, INC.
1921/DELNP/2005 06-05-2005 247426 06-04-2011 DERMASTICK THICKENED OINTMENT JAGOTEC AG
3762/KOLNP/2006 13-12-2006 247490 12-04-2011 CAPSULES COMPRISING A MICRO-ORGANISM, A FIRMENICH SA
MATRIX COMPONENTS AND AT LEAST ONE
ENCAPSULATABLE MATERIAL AND PROCESS FOR ITS
PREPARATION
1208/KOLNP/2006 09-05-2006 247495 12-04-2011 PYRAZOLYL DERIVATIVES IN THE FORM OF DRUGS FOR AVENTIS PHARMA S.A.
TREATING ACUTE OR CHRONIC NEURONAL
REGRESSIONS
3481/KOLNP/2006 22-11-2006 247501 12-04-2011 PROPANE-1,3-DIONE DERIVATIVE OR SALT THEREOF ASTELLAS PHARMA INC.

132/KOLNP/2007 10-01-2007 247503 12-04-2011 2-(PYRIDIN-2-YL)-PYRIMIDINES AND THEIR USE FOR BASF AKTIENGESELLSCHAFT
CONTROLLING HARMFUL FUNGI
2286/KOLNP/2006 10-08-2006 247504 12-04-2011 TRIAZOLOPYRIMIDINES BASF AKTIENGESELLSCHAFT
405/DELNP/2005 02-02-2005 247532 18-04-2011 AZABICYCLO DERIVATIVES AS MUSCARINIC RECEPTOR RANBAXY LABORATORIES LIMITED
ANTAGONISTS
1406/DELNP/2005 07-04-2005 247540 18-04-2011 A PHARMACEUTICAL COMPOSITION COMPRISING AN OREXO AB
ACID SUSCEPTIBLE PROTON PUMP INHIBITOR AND AN
H2 RECEPTOR ANTAGONIST
2482/CHENP/2006 06-07-2006 247551 19-04-2011 TETRAPEPTIDE LYSYL-GLUTAMYL-ASPARTYL- ACCESS BIOSCIENCE CJSC
TRYPTOPHANE AMIDE
233/MUM/2003 27-02-2003 247575 25-04-2011 HERBAL SKIN-CARE COMPOSITION THE KELKAR EDUCATION TRUST'S
SCIENTIFIC RESEARCH CENTRE
1411/MUM/2006 04-09-2006 247582 25-04-2011 A SYSTEM FOR SPATIALLY AND TEMPORALLY PANACEA BIOTEC LTD.
PROGRAMMABLE DELIVERY OF AN ACTIVE AGENT
4915/DELNP/2005 26-10-2005 247600 26-04-2011 MAYTANSINOID CELL-BINDING CONJUGATES AND THE IMMUNOGEN , INC.
PREPARATION THEREOF
1310/CHENP/2006 17-04-2006 247612 27-04-2011 TASTE - MASKED FORMULATION COMPRISING NOVARTIS AG
CLARITHROMYCIN
858/DEL/2004 11-05-2004 247615 27-04-2011 A POLYHERBAL COMPOSITION FOR THE TREATMENT OF OHARI, VIJAY KUMAR
VIRAL HEPATITIS
2954/KOLNP/2006 12-10-2006 247675 02-05-2011 COMBINATION OF PENTRAXIN PTX3 AND AN SIGMA-TAU INDUSTRIE
ANTIFUNGAL AGENT FARMACEUTICHE RIUNITE S.P.A.
IN/PCT/2002/00585/DEL 06-06-2002 247731 09-05-2011 A COMPOSITION USEFUL FOR TREATING OR CHEMGEN CORPORATION
AMELIORATING THE RISK OF DIGESTIVE TRACT
INFECTION
156/MUM/2005 14-02-2005 247743 10-05-2011 WATER SOLUBLE ANTI-DANDRUDFF COMPOUNDS AND GALAXY SURFACTANTS LIMITED
COMPOSITIONS THEREOF
2576/DELNP/2006 08-05-2006 247748 11-05-2011 PHARMACEUTICAL COMPOSITION COMPRISING RIEMSER ARZNEIMITTEL AG.
OXOPLATIN, THE SALTS AND DERIVATIVES THEREOF
1388/DEL/1999 20-10-1999 247750 11-05-2011 A SUSTAINED-RELEASE FORMULATION FOR ORAL PFIZER RESEARCH AND DEVELOPMENT
ADMINISTRATION FOR THE TREATMENT OR COMPANY, N.V./S.A.,
PREVENTION OF SEXUAL DYSFUNCTION
187/DEL/2002 01-03-2002 247754 11-05-2011 4-(AMINOMETHYL)-PIPERIDINE BENZAMIDE JANSSEN PHARMACEUTICA N.V
COMPOUNDS
462/MUM/2004 16-04-2004 247764 16-05-2011 ANTIINFECTIVE QUINOLONE COMPOUNDS AND CADILA HEALTHCARE LIMITED
PROCESS FOR PREPARATION THEREOF
3818/KOLNP/2006 18-12-2006 247808 24-05-2011 A COMPOSITION FOR TREATING AND PREVENTING BRIGHT FUTURE PHARMACEUTICAL
SLEEP DISORDER LABORATORIES LIMITED
52/DELNP/2006 03-01-2006 247821 25-05-2011 6-(1,1-DIFLUOROALKYL)-4-AMINOPICOLINATES AND DOW AGROSCIENCES LLC
THEIR USE AS HERBICIDES
179/DELNP/2006 10-01-2006 247860 27-05-2011 ISETHIONATE SALT OF A SELECTIVE CDK4 INHIBITOR WARNER-LAMBERT COMPANY LLC,

6241/DELNP/2006 25-10-2006 247890 31-05-2011 AN ORAL MODIFIED RELEASE PHARMACEUTICAL ASTRAZENECA AB


COMPOSITION
971/MUMNP/2006 21-08-2006 247891 31-05-2011 ENTERIC COATINGS FOR ORALLY INGESTIBLE BPSI HOLDINGS,INC.
SUBSTRATES
2478/KOLNP/2006 22-08-2006 247909 01-06-2011 A FLUORO SUBSTITUTED COMPOUND OF FORMULA ELI LILLY AND COMPANY
(1A) USEFUL AS SELECTIVE ESTROGEN RECEPTOR
MODULATORS AND PHARMACEUTICAL COMPOSITION
THEREOF
485/CAL/2001 29-08-2001 247910 01-06-2011 A STERILE OPHTHALMIC DROP PREPARATION DR. GERHARD MANN CHEMISCH-
PHARMAZEUTISCHE FABRIK GMBH
922/MUM/2002 23-10-2002 247913 02-06-2011 NOVEL TRICYCLIC COMPOUNDS AS PDE4 INHIBITORS GLENMARK PHARMACEUTICALS
LIMITED
811/MUMNP/2003 28-08-2003 247914 02-06-2011 A COMPOUND OF FORMULA I AND BAYER HEALTHCARE LLC
PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF IN
TREATING RAF MEDIATED DISEASES
5515/DELNP/2005 29-11-2005 247944 06-06-2011 STABILIZED PHARMACEUTICAL PEPTIDE NOVO NORDISK A/S
COMPOSITIONS.
2479/KOLNP/2006 31-08-2006 247943 06-06-2011 A BENZAZEPINE COMPOUND ELI LILLY AND COMPANY
3137/DELNP/2005 14-07-2005 247967 07-06-2011 ORAL CARE COMPOSITION COLGATE-PALMOLIVE COMPANY
13/MUMNP/2007 02-01-2007 247984 08-06-2011 CRYSTALLINE FORM OF A TRIAZOLO (4,5-D)PYRIMIDINE ASTRAZENECA AB
COMPOUND
1891/MUM/2006 15-11-2006 248024 09-06-2011 A LIQUID FORMULATION FOR HYGIENE AND JOSHI, VINAYAK NARAHAR
TREATMENT OF AILMENTS OF THROAT AND MOUTH

890/MUM/2004 16-08-2004 248023 09-06-2011 A CONTROLLED RELEASE ANTIDIABETIC FORMULATION IPCA LABORATORIES LIMITED
COMPRISING GLICLAZIDE
1112/DEL/2002 06-11-2002 248025 09-06-2011 NOVEL 4-ETHYL-5ALKOXYPRIMAQUINE COMPOUNDS NATIONAL INSTITUTE OF
PHARMACEUTICAL EDUCATION AND
RESEARCH (NIPER)
844/DELNP/2005 04-03-2005 248026 09-06-2011 S-(-)- AMLODIPINE NICOTINATE AND PROCESS FOR THE HANLIM PHARMACEUTICAL CO., LTD.
PREPARATION THEREOF
456/DEL/2000 25-04-2000 248090 16-06-2011 GLUCOCORTICOID RECEPTOR MODULATORS PFIZER PRODUCTS IN
58/MUM/2005 19-01-2005 248096 16-06-2011 HERBAL CONTRACEPTIVE FORMULATIONS SINGH KAMALINDER KAUR
02044/DELNP/2003 28-11-2003 248107 17-06-2011 PHARMACEUTICAL FORMULATION FOR THE EFFICIENT AXON BIOCHEMICALS B.V.
ADMINISTRATION OF APOMORPHINE 6AR-(-)-N-PROPYL-
NORAPOMORPHINE AND THEIR DERIVATIVES AND PRO-
DRUGS THEREOF
768/DELNP/2005 25-02-2005 248186 27-06-2011 A HEMIACETAL COMPOUND KISSEI PHARMACEUTICAL CO.,LTD.,
1556/KOLNP/2006 06-06-2006 248227 28-06-2011 PYRAZINES VERTEX PHARMACEUTICALS
INCORPORATED
1193/KOLNP/2003 18-09-2003 248253 29-06-2011 AN INVITRO ASSAY FOR IDENTIFYING A CANDIDATE CHIRON CORPORATION
AGENT THAT REDUCES GROWTH OF A CANCEROUS
CELL
IN/PCT/2002/00769/DEL 06-08-2002 248284 01-07-2011 AN AQUEOUS PREPARATION OF PROPOFOL WITH MAELOR PHARMACEUTICALS LIMITED
IMPROVED SOLUBILITES
1891/DELNP/2004 01-07-2004 248287 01-07-2011 PURIFICATION OF ONIUM HYDROXIDES BY SACHEM, INC
ELECTRODIALYSIS
666/DELNP/2005 21-02-2005 248348 06-07-2011 A SUBSTITUTED PYRAZOLE COMPOUND AND KISSEI PHARMACEUTICAL CO. LTD
PHARMACEUTICAL COMPOSITION THEREOF
2248/KOLNP/2006 08-08-2006 248349 06-07-2011 NOVEL COMPOUNDS AS FAAH INHIBITORS SANOFI AVENTIS
1334/DELNP/2005 04-04-2005 248353 06-07-2011 A SPOT-ON FORMULATION USEFUL FOR THE MERIAL LIMITED
TREATMENT OF PARASITE INFESTATION
6786/DELNP/2006 15-11-2006 248361 07-07-2011 A PHARMACEUTICAL COMPOSITION FOR EFFECTIVE WARNER CHILCOTT COMPANY,LLC
ABSORPTION
1135/CHENP/2006 03-04-2006 248395 12-07-2011 PYRAZOLO AND IMIDAZO-PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG

2240/KOLNP/2006 08-08-2006 248401 12-07-2011 THIOAMIDES AND SALTS THEREOF AND CYTOKINE ISHIHARA SANGYO KAISHA, LTD.
PRODUCTION INHIBITORS CONTAINING BOTH
491/DELNP/2007 18-01-2007 248459 18-07-2011 A COMPOUND REPRESENTED BY FORMULA (I) MEIJI SEIKA KAISHA&nbsp; LTD.
583/MUMNP/2004 19-10-2004 248542 25-07-2011 PHARMACEUTICAL FORMULATION COMPRISING NEURIM PHARMACEUTICALS (1991)
MELATONIN LTD.
5666/DELNP/2006 28-09-2006 248545 25-07-2011 FLAVOPEREIRINE DERIVATIVES FOR CANCER THERAPY DABUR PHARMA LTD

2504/DEL/2004 16-12-2004 248560 25-07-2011 ANTICIGARETTE HERBAL FORMULATION AS AN ANTI- COUNCIL OF SCIENTIFIC & INDUSTRIAL
DOTE TO TOBACCO RESEARCH
327/DELNP/2004 12-02-2004 248615 28-07-2011 A COSMETIC COMPOSITION HAVING A SKIN LVMH RECHERCHE
TIGHTENNING EFFECT
1480/MUM/2005 29-11-2005 248622 28-07-2011 PREPARATION OF DIGESTIVE ENZYMES CONTAINING MERCURY LABORATORIES LIMITED
DRY SYRUP
3239/DELNP/2005 21-07-2005 248632 29-07-2011 AZABICYCLIC HETEROCYCLIC COMPOUND NOVEXEL
539/DELNP/2004 04-03-2004 248635 29-07-2011 BENZOTHIAZEPINE AND BENZOTHIADIAZEPINE ASTRAZENECA AB
DERIVATIVES WITH LLEAL BILE ACID TRANSPORT (IBAT)
INHIBITORY ACTIVITY FOR THE TREATMENT OF
HYPERLIPIDAEMIA
685/DEL/2002 26-06-2002 248660 02-08-2011 A SYNERGISTIC PHARMACEUTICAL COMPOSITION OF NATIONAL INSTITUTE OF
CELECOXIB WITH IMPROVED AQUEOUS SOLUBILITY PHARMACEUTICAL EDUCATION AND
RESEARCH (NIPER)
583/MUM/2007 29-03-2007 248729 12-08-2011 MODIFIED DOSAGE FORMS OF TACROLIMUS PANACEA BIOTEC LIMITED
775/MUM/2004 21-07-2004 248777 24-08-2011 PHARMACEUTICAL COMPOSITION CONTAINING MACLEODS PHARMACEUTICALS
COMBINATION OF PROTON PUMP INHIBITOR WITH LIMITED
MODIFIED RELEASE DOMPERIDONE
2507/DEL/2004 16-12-2004 248784 24-08-2011 DEVELOPMENT OF HARBAL NUTRITIOUS CHOCAEATE COUNCIL OF SCIENTIFIC AND
AND ITS PROCESSING INDUSTRIAL RESEARCH
4656/DELNP/2005 13-10-2005 248794 25-08-2011 A COMPOSITION CONTAINING L-LACTIC ACID OR L- INNOGENE KALBIOTECH PTE LTD
LACTATE AND USES THEREOF
1535/DEL/2004 18-08-2004 248796 25-08-2011 AN ANALGESIC PREPARATION CONTAINING MORPHINE ALL INDIA INSTITUTE OF MEDICAL
AND NIMODIPINE AND A PROCESS FOR PREPARATION SCIENCE
THEREOF
2426/DEL/2005 09-09-2005 248802 25-08-2011 A SUSTAINED RELEASE MULTILAYERED TABLET DELHI INSTITUTE OF PHARMACEUTICAL
COMPOSITION FOR UNSTABLE DRUG SCIENCES & RESEARCH

147/DEL/2005 24-01-2005 248830 29-08-2011 A RELEASE PHARMACEUTICAL PREPARATION FOR JAMIA HAMDARD (HAMDARD
COLON DELIVERY UNIVERSITY)
2403/KOLNP/2006 24-08-2006 248843 30-08-2011 ANTITHROMBOTIC COMPOUND SANOFI-AVENTIS
74/MUM/2005 24-01-2005 248852 31-08-2011 NOVEL OPTHALMIC COMBINATION OF GATIFLOXACIN CIPLA LIMITED
AND PREDNISOLONE
1197/MUM/2006 28-07-2006 248853 31-08-2011 TOPICAL COMPOSITION FOR MINIMIZING HAIR LOSS HINDUSTAN UNILEVER LIMITED

1643/DELNP/2005 21-04-2005 248867 02-09-2011 AMIDE COMPOUNDS OF GENERAL FORMULA I AS MCH BOEHRINGER INGELHEIM PHARMA
ANTAGONISTS GMBH & CO. KG.
3162/DELNP/2007 27-04-2007 248904 07-09-2011 QUINOLINE DERIVATIVES. F.HOFFMANN-LA ROCHE AG
1353/MUM/2006 28-08-2006 248977 19-09-2011 LIPIDIC NANOPARTICULATE BASED DOSAGE FORMS OF PATRAVALE VANDANA BHARAT
ANTIPARASITICS AND ANTIINFECTIVES
2669/KOLNP/2007 18-07-2007 248983 19-09-2011 A SUBSTITUTED THIAZOLOPYRIDINONE COMPOUND ELI LILLY AND COMPANY
USEFUL AS MELANIN CONCENTRATING HERMONE
(MCH) ANTAGONISTS AND PHARMACEUTICAL
COMPOSITION THEREOF
3008/DELNP/2007 23-04-2007 248995 20-09-2011 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR WAKUNAGA PHARMACEUTICAL CO.,
SALTS THEREOF LTD
2282/KOLNP/2006 10-08-2006 248998 20-09-2011 DERIVATIVES OF ALKYLPIPERAZINE- AND SANOFI-AVENTIS
ALKYLHOMOPIPERAZINE- CARBOXYLATES,
PREPARATION METHOD THEREOF AND USE OF SAME
AS FAAH ENZYME INHIBITORS
4047/DELNP/2004 20-12-2004 249008 21-09-2011 A PHARMACEUTICAL COMPOSITION COMPRISING A PFIZER PRODUCTS INC.
TABLET CORE OR CAPSULE FILL
2997/KOLNP/2006 17-10-2006 249090 29-09-2011 PIPERAZINYLPIPERIDINE DERIVATIVES AS CYTOKINE INCYTE CORPORATION
RECEPTOR ANTAGONISTS
3884/DELNP/2005 31-08-2005 249112 30-09-2011 AN ORALLY ADMINISTERED PHARMACEUTICAL MCNEIL AB
FORMULATION
478/MUM/2006 29-03-2006 249133 03-10-2011 HERBAL COMPOSITION COMPRISING EXTRACT OF ROOT PIRAMAL LIFE SCIENCES LIMITED
OF MURRAYA KOENIGII FOR TREATMENT OF
INFECTIONS CAUSED BY DERMATOPHYTES
4188/DELNP/2005 16-09-2005 249157 05-10-2011 OXIDATIVE REDUCTIVE POTENTIAL WATER SOLUTION OCULUS INNOVATIVE SCIENCES, INC.
AND PROCESSES FOR PRODUCING SAME
3208/DELNP/2006 05-06-2006 249171 10-10-2011 A PHARMACEUTICAL FORMULATION ADAPTED FOR BIONUMERIK PHARMACEUTICALS, INC.
ADMINISTRATION TO HUMAN PATIENTS
1698/MUM/2007 05-09-2007 249181 10-10-2011 STABLE SOLID ORAL PHARMACEUTICAL COMPOSITIONS IPCA LABORATORIES LIMITED
OF ISOTRETINOIN AND PROCESS THEREOF

4048/DELNP/2005 09-09-2005 249175 10-10-2011 AN ORAL PHARMACEUTICAL PREPARATION PIERRE FABRE MEDICAMENT
688/MUM/2005 08-06-2005 249183 10-10-2011 A TOPICAL SEMISOLID SILVER NANOPARTICLE SANJEEV KHANDELWAL
DISPERSION FORMULATION
215/DEL/2006 25-01-2006 249180 10-10-2011 A HERBAL COMPOSITION EFFECTIVE AGAINST DIRECTOR, CENTRAL COUNCIL FOR
NAZFUDDAM AND A PROCESS FOR THE PREPARATION RESEARCH IN UNANI MEDICINE
THEREOF"
218/DEL/2006 25-01-2006 249186 10-10-2011 A NOVEL HERBAL COMPOSITION EFFECTIVE AGAINST DIRECTOR, CENTRAL COUNCIL FOR
CORYZA AND A PROCESS FOR PREPARING THEREOF RESEARCH IN UNANI MEDICINE

1230/MUM/2006 03-08-2006 249226 12-10-2011 ION EXCHANGE RESIN BASED EXTENDED RELEASE AMIN, PURNIMA DHANRAJ
GASTRO-RETENTIVE DOSAGE FORMS
5691/DELNP/2006 29-09-2006 249232 12-10-2011 MICROFLUIDIZED OIL-IN-WATER EMULSIONS AND PFIZER PRODUCTS INC.
VACCINE COMPOSITIONS
1012/MUM/2006 27-06-2006 249243 12-10-2011 THE THROMBOCHEK TEST KIT DILIP SHRINIVAS VELASKAR
2128/MUM/2006 26-12-2006 249299 17-10-2011 A SYNERGISTIC HERBAL FORMULATION FOR THE PATANKAR SURESH
TREATMENT OF RENAL CONDITION
2114/MUM/2006 22-12-2006 249293 17-10-2011 A MEDICAMENT FOR THE TREATMENT OF HIV SAYYED BAWA ABDUL KAREEM
INFECTION,
3734/DELNP/2005 23-08-2005 249316 17-10-2011 AN AMINO-PYRIDINE COMPOUND OF FORMULA I SUGEN, INC.,
2254/DELNP/2003 24-12-2003 249325 17-10-2011 A COMPOUND OF FORMULA (I) BAOSHUN LIU
515/MUMNP/2007 09-04-2007 249345 18-10-2011 CONVENIENTLY IMPLANTABLE SUSTAINED RELEASE RAMSCOR INC.
DRUG COMPOSITIONS
2492/KOLNP/2006 31-08-2006 249558 25-10-2011 PHYSIOLOGICAL COOLING COMPOSITIONS CONTAINING MILLENNIUM SPECIALTY CHEMICALS
HIGHLY PURIFIED ETHYL ESTER OF N-[[5-METHYL-2-(1-
METHYLETHYL)CYCLOHEXYL)CARBONYL]GLYCINE

3827/KOLNP/2006 19-12-2006 249525 25-10-2011 NOVEL ARYLAMIDINE COMPOUND HAVING M/S TOYAMA CHEMICAL CO., LTD.
ANTIFUNGAL AND ANTIPROTOZOAL ACTIVITY
1961/KOLNP/2006 12-07-2006 249527 25-10-2011 A PHARMACEUTICAL COMPOSITION RICHTER GEDEON VEGYESZETI GYAR RT

7358/DELNP/2006 06-12-2006 249562 27-10-2011 A FORMULATION PROVIDING ENHANCED ULTRASOUND ACUSPHERE&nbsp; INC
CONTRAST IMAGES AND A METHOD FOR MAKING THE
SAME
4201/CHENP/2006 14-11-2006 249605 31-10-2011 A COMPOUND OF FORMULA I AS PPAR MODULATORS IRM LLC

1054/KOLNP/2007 26-03-2007 249614 31-10-2011 OPTICALLY ACTIVE 4,4-DI-SUBSTITUTED OXAZOLIDINE SANKYO COMPANY LIMITED
DERIVATIVE AND PROCEDURES FOR THEIR
PREPARATION
497/KOLNP/2006 03-03-2006 249626 31-10-2011 A NON-TRANSLUCENT OIL IN WATER EMULSION FOAMIX LTD.
1944/KOLNP/2006 11-07-2006 249627 31-10-2011 ARYLOXYALKYLCARBAMATE COMPOUNDS, SANOFI-AVENTIS
PREPARATION METHOD THEREOF AND COMPOSITION
COMPRSING THEM
1290/CHENP/2006 13-04-2006 249666 01-11-2011 IMIDAZOPYRAZINE TYROSINE KINASE INHIBITORS OSI PHARMACEUTICALS, INC.
2932/KOLNP/2006 11-10-2006 249679 02-11-2011 THIOAMIDE DERIVATIVES AS PROGESTERONE WYETH
RECEPTOR MODULATORS
2938/KOLNP/2006 11-10-2006 249735 08-11-2011 CYANOPYRROLE CONTAINING CYCLIC CARBAMATE AND WYETH
THIOCARBAMATE BIARYLS AND METHODS FOR
PREPARING THE SAME
8001/DELNP/2006 29-12-2006 249742 08-11-2011 2-QUINAZOLINYLAMINOC1-6ALKANEDIYL COMPOUND JANSSEN PHARMACEUTICA N.V.
AS PARP INHIBITORS
3206/KOLNP/2006 02-11-2006 249747 08-11-2011 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES AS ARENA PHARMACEUTICALS, INC.
MODULATORS OF METABOLISM AND THE PROPHYLAXIS
AND TREATMENT OF DISORDERS RELATED THERETO.

2984/KOLNP/2006 16-10-2006 249754 08-11-2011 PURIFICATION OF PROGESTERONE RECEPTOR WYETH


MODULATORS
1960/KOLNP/2006 12-07-2006 249758 08-11-2011 CYSTEINE PROTEASE INHIBITORS MEDIVIR AB
4509/DELNP/2005 04-10-2005 249774 09-11-2011 A TWO-PART BICARBONATE CONTAINING SOLUTION. BAXTER INTERNATIONAL INC.

1960/MUM/2006 29-01-2007 249777 10-11-2011 PHARMACEUTICAL DERMAL COMPOSITION USEFUL IN VLIFE SCIENCES TECHNOLOGIES PVT.
TREATMENT OF DIABETIC COMPLICATIONS LTD.
404/KOLNP/2007 05-02-2007 249810 14-11-2011 ACID AMIDE DERIVATIVE AND FUNGICIDAL ISHIHARA SANGYO KAISHA, LTD.
COMPOSITION COMPRISING IT
194/KOLNP/2007 16-01-2007 249822 15-11-2011 N-(1H-INDOLYL)-1H-INDOLE-2-CARBOXAMIDE SANOFI-AVENTIS
DERIVATIVES AND THEIR PREPARATION
1517/CHENP/2006 03-05-2006 249834 16-11-2011 STABLE PHARMACEUTICAL COMPOSITION COMPRISING LEK PHARMACEUTICALS d.d.
GRANULOCYTE-COLONY STIMULATING FACTOR

1080/DELNP/2006 01-03-2006 249872 17-11-2011 MELT-FORMULATED, MULTIPARTICULATE ORAL GRUNENTHAL GMBH


DOSAGE FORM
IN/PCT/2000/322/KOL 18-09-2000 249892 21-11-2011 INHIBITORS OF CASPASES VERTEX PHARMACEUTICALS
INCORPORATED
1963/KOLNP/2006 13-07-2006 249917 23-11-2011 NOVEL FUSED PYRROLOCARBAZOLES CEPHALON, INC
3798/KOLNP/2006 18-12-2006 249919 23-11-2011 FUSED HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY
LIMITED
2761/KOLNP/2006 21-09-2006 249922 23-11-2011 NON-CYCLIC KETONES AND PERFUMING COMPOSITION FIRMENICH S.A.
COMPRISING THEM
385/MUM/2007 28-02-2007 249929 23-11-2011 NOVEL COSMETIC CREAM COMPOSITIONS HINDUSTAN UNILEVER LIMITED
2544/DELNP/2004 31-08-2004 249968 25-11-2011 ACYLAMINOPIPERIDINE-1-CARBOXAMIDINE KALVISTA PHARMACEUTICALS LIMITED
COMPOUND OF FOUMULA 1
5385/DELNP/2005 23-11-2005 250040 30-11-2011 A PHARMACEUTIACAL COMPOSITION OF PHARMA MAR S.A.U.
ECTEINASCIDIN 743 (ET-743) IN COMBINATION WITH A
PLATINUM COMPOUND WITHOUT INCREASING THE
TOXICITY OF EACH DRUG
144/DELNP/2007 05-01-2007 250050 30-11-2011 AN ENANTIOMERICALLY PURE AMINOPYRIDINE PFIZER INC
COMPOUND OF FORMULA (I)
3494/DELNP/2006 19-06-2006 250055 01-12-2011 AN OPHTHALMICALLY ACCEPTABLE COMPOSITION ALLERGAN, INC.
6179/DELNP/2006 23-10-2006 250059 01-12-2011 ”BIOCOMPATIBLE COMPOSITE PARTICLE OR NANOBIOTIX
NANOPARTICLE AGGREGATE CAPABLE OF GENERATING
FREE RADICALS OR HEAT”
1375/MUMNP/2006 16-11-2006 250088 05-12-2011 NOVEL TETRAHYDROCARBAZOLE DERIVATIVES WITH ZENTARIS GMBH
IMPROVED BIOLOOGICAL ACTION AND IMPROVED
SOLUBILITY AS LIGANDS FOR G-PROTEIN COUPLED
RECEPTORS (GPCRS)
2121/MUM/2007 26-10-2007 250095 07-12-2011 A STABLE ORAL FORMULATION CONTAINING A PROTON CADILA HEALTHCARE LIMITED
PUMP INHIBITOR
2150/DELNP/2004 23-07-2004 250133 09-12-2011 A 4-(ARYLMETHYLOXY)-PYRIDIN-2-ONE COMPOUND" PHARMACIA CORPORATION
1340/MUM/2007 12-07-2007 250130 09-12-2011 A SUSTAINED RELEASE ANTIMALARIAL TABLET IPCA LABORATORIES LIMITED
COMPOSITION COMPRISING PRIMAQUINE PHOSPHATE
AND A PROCESS FOR PREPARING THE SAME

1233/KOLNP/2006 11-05-2006 250181 14-12-2011 MODULATORS OF CELLULAR ADHESION SARCODE CORPORATION


580/MUM/2003 06-06-2003 250249 19-12-2011 MODIFIED RELEASE PHARMACEUTICAL FORMULATION CADILA HEALTHCARE LIMITED
CONTAINING FLUVASTATIN SODIUM

3348/DELNP/2007 04-05-2007 250251 20-12-2011 EYE DROP COMPRISING HOMOPIPERAZINE AND KOWA CO.,LTD
PHOSPHORIC ACID OR THEIR SALTS THEREOF
2140/DELNP/2006 19-04-2006 250309 22-12-2011 COMPOUND USEFUL AS CCR-2 ANTAGONIST SALT MERCK SHARP & DOHME CORP.
4311/DELNP/2006 26-07-2006 250334 27-12-2011 AN AMINE SALT OF A 2-QUINOLINE DERIVATIVE OTSUKA PHARMACEUTICAL CO., LTD
6170/DELNP/2007 07-08-2007 250384 30-12-2011 RINSE-OFF/WIPE-OFF SKIN CLEANSING COMPOSITION THE PROCTER & GAMBLE COMPANY

5178/DELNP/2007 05-07-2007 250392 30-12-2011 N-[(1S)-2-(DMETHYLAMINO)-1-PHENYLETHYL]-6,6- PFIZER INC.


DIMITHYL-3-[(2-METHYLTHIENO[3,2-D]PYRIMDIN-4-
YL)AMINO]-4,6-DIHYDROPYRROLO[3,4-C]PYRAZOLE-
5(1H) CARBOXAMIDE
3130/KOLNP/2006 27-10-2006 250430 03-01-2012 AMIDO COMPOUNDS AND THEIR USE AS INCYTE CORPORATION
PHARMACEUTICALS
2112/KOLNP/2006 26-07-2006 250432 03-01-2012 FUSED CYCLIC SYSTEMS USEFUL AS INHIBITORS OF TEC VERTEX PHARMACEUTICALS
FAMILY PROTEIN KINASES INCORPORATED
3348/KOLNP/2006 14-11-2006 250453 04-01-2012 PYRROLE COMPOUNDS VERTEX PHARMACEUTICALS
INCORPORATED
2395/KOLNP/2006 23-08-2006 250461 04-01-2012 LYSINE BASED COMPOUNDS AMBRILIA BIOPHARMA INC.
3049/KOLNP/2006 20-10-2006 250462 04-01-2012 SUBSTITUTED AZEPINE DERIVATIVES AS SEROTONIN ATHERSYS, INC.
RECEPTOR MODULATORS
2683/KOLNP/2005 23-12-2005 250464 04-01-2012 ABUSE RESISTANT AMPHETAMINE COMPOUNDS NEW RIVER PHARMACEUTICALS INC
4483/KOLNP/2007 21-11-2007 250478 05-01-2012 PHARMACEUTICAL COMBINATION COMPRISING AN ADVANCED SCIENTIFIC DEVELOPMENTS
ANTIFUNGAL AGENT AND AN ACTIVE SUBSTANCE
SELECTED FROM CARVEOL, EUGENOL, THYMOL,
BORNEOL, CARVACROL, AND ALPHA- AND BETA-
IONONES
3074/DELNP/2004 07-10-2004 250486 05-01-2012 "HYPERFORIN AND ADHYPERFORIN DERIVATIVES FOR INDENA S.P.A
USE IN THE TREATMENT OF DEPRESSION AND
ALZHEIMER'S DISEASE"
5093/DELNP/2007 02-07-2007 250488 05-01-2012 "2-CYCLOPENTEN-1-ONE OXIME DERIVATIVES AMOREPACIFIC CORPORATION
INHIBITING PRODUCTION OF TNF-ALPHA"
2498/DEL/2006 20-11-2006 250538 09-01-2012 "A NOVEL HETEROCYCLEC CMPOUND XANTHONOXY HAMDARD UNIVERSITY
PROPANOLAMINES"
6487/DELNP/2006 02-11-2006 250549 10-01-2012 "INDENE DERIVATIVES AND PROCESS FOR THE KOREA RESEARCH INSTITUTE OF
PREPARATION THEREOF" CHEMICAL TECHNOLOGY
2027/KOLNP/2005 17-10-2005 250551 10-01-2012 NOVEL PHOSPHONIC ACID COMPOUNDS AS INHIBITORS ORTHO-MCNEIL PHARMACEUTICAL,
OF SERINE PROTEASES INC.
3178/KOLNP/2006 31-10-2006 250552 10-01-2012 NEUROLOGICALLY-ACTIVE COMPOUNDS PRANA BIOTECHNOLOGY LIMITED
2947/KOLNP/2006 12-10-2006 250556 10-01-2012 NOVEL COMPOUNDS (CAMPTOTHECIN DERIVATIVES SIGMA-TAU INDUSTRIE
CONJUGATED IN POSITION 7 TO ANTI-INTEGRIN CYCLIC FARMACEUTICHE RIUNITE S.P.A.
PEPTIDES) AS CYTOSTATIC AGENTS

2107/MUMNP/2008 01-10-2008 250583 11-01-2012 SUBSTITUTED PYRROLIDINONES AS INHIBITORS OF 11- ELI LILLY AND COMPANY
BETA-HYDROXYSTEROID DEHYDROGENASE 1
2793/KOLNP/2006 25-09-2006 250594 11-01-2012 NOVEL COMPOUNDS AND COMPOSITION THEREOF AS ARYX T HERAPEUTICS
ANTICOAGULANT
1653/DELNP/2006 27-03-2006 250598 11-01-2012 "A BODY-ABSORBABLE COMPOSITION" ORTHOCON, INC
3187/DEL/1998 29-10-1998 250614 12-01-2012 " MUTILIN 14-(EXO-8-METHYL-8-AZABICYCLO[3.2.1]OCT- SMITHKLINE BEECHAM LIMITED
3-YLSULFANYL)-ACETATE AND ITS SALT"

1343/KOLNP/2005 12-07-2005 250653 16-01-2012 HYDROXAMIC ACID COMPOUND NOVARTIS VACCINES AND DIAGNOSTICS
INC.
2955/KOLNP/2006 12-10-2006 250673 18-01-2012 7-T-BUTOXYIMINOMETHYLCAMPTOTHECIN SIGMA-TAU INDUSTRIE
CONJUGATED IN POSITION 20 WITH INTEGRIN FARMACEUTICHE RIUNITE S.P.A.
ANTAGONISTS
6268/DELNP/2006 25-10-2006 250681 18-01-2012 "SOFTGEL ENCAPSULATED PHARMACEUTICAL THE PROCTER & GAMBLE COMPANY
COMPOSITIONS COMPRISING CONCENTRATED ACTIVE
INGREDIENTS"
216/DEL/2006 25-01-2006 250700 20-01-2012 ""A HERBAL COMPOSITION EFFECTIVE AGAINST DIRECTOR, CENTRAL COUNCIL FOR
ARTHRITIS AND TO PROCESS FOR THE PREPARATION RESEARCH IN UNANI MEDICINE
THEREOF".
1321/CHENP/2007 30-03-2007 250702 20-01-2012 HYDROXYLAMINE ESTERS AS POLYMERIZATION CIBA HOLDING INC.
INITIATORS
828/CAL/1999 06-10-1999 250728 23-01-2012 A COMPOUND OF PYRIDINIUM SERIES TORRENT PHARMACEUTICALS LTD.
901/MUM/2004 20-08-2004 250735 23-01-2012 NOVEL ANTIDIABETIC COMPOUNDS CADILA HEALTHCARE LIMITED
337/MUMNP/2007 06-03-2007 250747 23-01-2012 PURINE DERIVATIVES AS A3 AND A1 ADENOSINE GOVERNMENT OF THE UNITED STATES
RECEPTOR AGONISTS OF AMERICA REPRESENTED BY THE
SECRETARY, DEPARTMENT OF HEALTH
AND HUMAN SERVICES
406/DELNP/2005 02-02-2005 250752 24-01-2012 "3,6-DISUBSTITUTED AZABICYCLO [3.1.0]HEXANE RANBAXY LABORATORIES LIMITED
DERIVATIVES USEFUL AS MUSCARINIC RECEPTOR
ANTAGONISTS"
IN/PCT/2001/00758/DEL 24-08-2001 250754 24-01-2012 "A PHARMACEEUTICAL COMPOSITION" TRIANGLE PHARMACEUTICALS, INC.
5055/DELNP/2006 01-09-2006 250758 24-01-2012 TETRAHYDROCARBAZOLE COMPOUNDS F. HOFFMANN-LA ROCHE AG
3183/DELNP/2006 02-06-2006 250807 30-01-2012 "HETEROCYCLIC INHIBITORS OF MEK AND METHODS OF ARRAY BIOPHARMA INC.
USE THEREOF"
1511/CHENP/2006 03-05-2006 250824 31-01-2012 AQUEOUS SOLUTION OF CHROMIUM SALT AND NIPPON CHEMICAL INDUSTRIAL CO.,
METHOD FOR PRODUCING SAME LTD
3339/DELNP/2007 03-05-2007 250842 01-02-2012 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 SYNTA PHARMACEUTICALS CORP.
ACTIVITY
2301/DELNP/2007 23-03-2007 250843 01-02-2012 "LIPOSOMAL COMPOSITIONS OF GLUCOCORTICOID YISSUM RESEARCH DEVELOPMENT
AND GLUCOCORTICOID DERIVATIVES" COMPANY OF THE HERBREW
UNIVERSITY OF JERUSALEM
2488/CHENP/2006 06-07-2006 250853 02-02-2012 DIAZA-SPIROPIPERIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG
2284/DEL/2004 17-11-2004 250857 02-02-2012 "2-ETHYL-4,6-DIMETHYLPHENYL-SUBSTITUTED BAYER CROPSCIENCE AG,
SPIROCYCLIC TETRAMIC ACID COMPOUNDS"
419/DEL/2002 28-03-2002 250881 03-02-2012 "A HERBAL OPHTHALMIC FORMULATION OF CURCUMA ALL INDIA INSTITUTE OF MEDICAL
LONGA FOR DELAYING THE ONSET AND PROGRESSION SCIENCES,
OF CATARACT"
1139/CHENP/2006 03-04-2006 250918 07-02-2012 ALKOXY SUBSTITUTED IMIDAZOQUINOLINES 3M INNOVATIVE PROPERTIES
COMPANY
2872/CHENP/2006 04-08-2006 250919 07-02-2012 MICROEMULSION FORMULATIONS COMPRISING NOVARTIS AG
PARTICULAR SUBSTANCE P ANTAGONISTS
3870/CHENP/2007 05-09-2007 250923 07-02-2012 ANALOGUES OF GLP-1 IPSEN PHARMA S.A.S
2395/CHENP/2007 04-06-2007 250971 14-02-2012 A COMPOSITION COMPRISING A SEQUESTERING AND A ALPHARMA, INC.
THERAPEUTIC SUBUNIT
3320/CHENP/2006 13-09-2006 250977 14-02-2012 A METHOD OF DEACTIVATING DUST MITE ALLERGENS RECKITT BENCKISER (UK) LIMITED
DER P AND DER F BY HOTPLATE EMANATION

2391/DEL/2004 30-11-2004 250983 14-02-2012 "A PHARMACEUTICAL COMPOSITION FOR JAMIA HAMDARD (HAMDARD
TRANSDERMAL/TRANSMUCOSAL DELIVERY" UNIVERSITY)
1012/DELNP/2006 27-02-2006 251016 16-02-2012 "A PHARMACEUTICAL COMPOSITIONS SUITABLE FOR STIEFEL LABORATORIES, INC.
TOPICAL ADMINISTRATION"
275/MUM/2004 07-03-2004 251029 17-02-2012 ORAL DROP FORMULATION CONTAINING SIMETHICONE SANJEEV KHANDELWAL
AND CAMYLOFIN DIHYDRAOCHLORIDE

6498/DELNP/2007 22-08-2007 251035 17-02-2012 "A BENZOIMIDAZOLE COMPOUND AND DAEWOONG PHARMACEUTICAL CO.,
PHARMACEUTICAL COMPOSITION COMPRISING THE LTD.
SAME"
1291/MUMNP/2006 03-11-2006 251055 20-02-2012 DERIVATIVES OF 14.15-DIHYDRO 20.21- BIOCORTECH
DINOREBURNAMENIN-14-OL FOR TREATMENT OF
DIPRESSIUON
2496/MUM/2007 18-12-2007 251063 21-02-2012 NOVEL SUBSTITUTED ARALKYL DERIVATIVES HAVING CADILA HEALTHCARE LIMITED
ANTIDIABETIC HYPOLIPIDEMIC,HYPOCHOLESTEREMIC
ACTIVITIES, PROCESS FOR THEIR PREPARATION AND
PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
AND THEIR USE IN MEDICINE

3740/DELNP/2005 23-08-2005 251084 22-02-2012 "A PHARMACEUTICAL FORMULATION" CHIESI FARMACEUTICI S.P.A.
1117/DELNP/2006 02-03-2006 251092 22-02-2012 "A COMPOSITION OF AT LEAST TWO AMIDE-BASED NEW JAPAN CHEMICAL CO., LTD.
COMPOUNDS REPRESENTED BY GENERAL FORMULA I"

1402/MUM/2006 01-09-2006 251100 22-02-2012 A NOVEL FORMULATION OF SEVELAMER USV LIMITED


HYDROCHLORIDE
4715/DELNP/2007 19-06-2007 251113 24-02-2012 "MATRIX TYPE SUSTAINED-RELEASE PREPARATION EISAI R & D MANAGEMENT CO.,LTD
CONTAINING BASIC DRUG OR SALT THEREOF, AND
METHOD FOR MANUFACTURING THE SAME"
1867/DELNP/2007 09-03-2007 251123 24-02-2012 "A MIXTURE OF FISH OIL FATTY ACID ESTER(S) OF ENZYMOTEC LTD.
PHYTOSTEROLS AND 1,3-DIGLYCERIDE(S) (DAG)"
745/MUM/2004 12-07-2004 251135 27-02-2012 NOVEL HETEROCYCLIC COMPOUNDS CADILA HEALTHCARE LIMITED
304/KOLNP/2007 25-01-2007 251140 27-02-2012 A COMPOSITION FOR A CAPSULE COATING WAKUNAGA PHARMACEUTICAL CO.,
LTD.
2013/DELNP/2007 15-03-2007 251142 27-02-2012 "A CYCLIC AMINE DERIVATIVE OR SALT THEREOF AND ASTELLAS PHARMA INC.
ITS PHARMACEUTICAL COMPOSITION"
177/MUMNP/2007 05-02-2007 251154 28-02-2012 NEW SELENOHYDROXY ACIDS AND THEIR DERIVATIVES TETRAHEDRON
APPLICATIONS IN NUTRITION, COSMETICS AND
PHARMACEUTICS
2418/MUM/2007 10-12-2007 251161 28-02-2012 NOVEL OMEGA -3 FATTY ACID COMPOSITION WITH OMNIACTIVE HEALTH TECHNOLOGIES
SIGNIFICANTLY REDUCED OFFENSIVE ODOUR AND PVT. LTD.
PROCESS FOR ITS PREPARATION
1976/MUMNP/2008 16-09-2008 251162 28-02-2012 BICYCLOHETEROARYL COMPOUNDS AS P2X7 RENOVIS, INC.
MODULATORS AND USES THEREOF
1378/MUMNP/2006 16-11-2006 251169 28-02-2012 GUANYLHYDRAZONE SALTS, COMPOSITIONS, CYTOKINE PHARMASCIENCES INC.
PROCESSES OF MAKING AND METHODS OF USING
1638/CHENP/2006 11-05-2006 251191 29-02-2012 ORTHO-SUBSTITUTED PENTAFLUORIDE SULFANYL- SANOFI-AVENTIS DEUTSCHLAND GMBH
BENZENES, METHOD FOR THE PRODUCTION THEREOF
AND THE THEREOF
2118/CHENP/2006 15-06-2006 251196 29-02-2012 COMPOSITION FOR COUPLING FILLER AND ELASTOMER CIBA HOLDING INC.

610/CHE/2006 03-04-2006 251197 29-02-2012 NOVEL DIPEPTIDYL PEPTIDASE IV INHIBITORS, MATRIX LABORATORIES LTD.
PROCESSES FOR THEIR PREPARATION AND
PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

7041/DELNP/2007 12-09-2007 251204 29-02-2012 "A HETEROCYCLIC COMPOUND REPRESENTED BY THE OTSUKA PHARMACEUTICAL CO., LTD.
FORMULA(1)"
3795/DELNP/2004 01-12-2004 251219 01-03-2012 "BASIC NON-PEPTIDE BRADYKININ ANTAGONISTS MENARINI RICERCHE S.P.A.
CONTAINING QUINOLINE AND A NITROGEN
HETEROCYCLE"
1331/CHENP/2003 25-08-2003 251226 02-03-2012 SALTS OF AVERMECTINS SUBSTITUTED IN THE 4"- SYNGENTA PARTICIPATIONS AG
POSITION AND HAVING PESTICIDAL PROPERTIES"
712/DELNP/2006 13-02-2006 251234 02-03-2012 "AN &#945;-2A/&#945;-1A SELECTIVE AGONIST, 1-(2,3- ALLERGAN, INC.
DIMETHYL-PHENYL)-ETHYL-1,3-DIHYDRO-IMIDAZOLE-2-
THIONE COMPOUND"
1838/CHENP/2004 18-08-2004 251236 02-03-2012 PHARMACEUTICAL FORMULATIONS OF SCHERING CORPORATION
TEMOZOLOMIDE
2130/KOLNP/2007 12-06-2007 251257 05-03-2012 POTENTIATORS OF GLUTAMATE RECEPTORS ELI LILLY AND COMPANY
1734/CHE/2007 07-08-2007 251268 05-03-2012 SOLID DOSAGE FORM OF ENTERIC SOLID DISPERSION SHIN-ETSU CHEMICAL CO., LTD
AND METHOD FOR PRODUCING THE SAME

1835/CHENP/2007 30-04-2007 251278 05-03-2012 PYRIMIDONE COMPOUND MITSUBISHI PHARMA CORPORATION,


SANOFI- AVENTIS
1170/DEL/1998 01-05-1998 251314 06-03-2012 "PHARMACEUTICAL COMPOSITION WITH FDXED FERRER INTERNACIONAL S.A.
QUANTITIES OF AN EPNALARIL AND NITRENDIPINE AND
METHOD FOR OBTAINING THE SAME"
710/CHENP/2007 19-02-2007 251320 06-03-2012 3-SUBSTITUTED-5-AND 6-AMINOALKYL INDOLE-2- AVENTIS PHARMACEUTICALS, INC
CARBOXYLIC ACID AMIDES AND RELATED ANALOGS AS
INHIBITORS OF CASEIN KINASE Ie
3006/DELNP/2004 01-10-2004 251447 16-03-2012 "A PHARMACEUTICAL COMPOSITION USEFUL FOR SINCLAIR PHARMACEUTICALS LIMITED
TOPICAL ADMINISTRATION COMPRISING AS ACTIVE
INGREDIENTS PROANTHOCYANIDINS"
3359/DELNP/2004 29-10-2004 251451 16-03-2012 "HYDROXAMIC ACID COMPOUNDS COMPRISING A TOPOTARGET UK (LIMITED)
PIPERAZINE LINKAGE AS HDAC INHIBITORS"
1862/DEL/2006 21-08-2006 251453 16-03-2012 "A NOVEL HERBAL COMPOSITION AND A PROCESS FOR CENTRAL COUNCIL FOR RESEARCH IN
PREPARATION THEREOF EFFECTIVE AGAINST UNANI MEDICINE
CONSTIPATION"
15/MUMNP/2005 10-01-2005 251454 16-03-2012 FLAVONE DERIVATIVES AS INHIBITORS OF CYCLIN- NICHOLAS PIRAMAL INDIA LIMITED
DEPENDENT KINASES
1374/DEL/2007 27-06-2007 251457 16-03-2012 "NAPHTHALENE COMPOUNDS OF FORMULA (I)" LES LABORATOIRES SERVIER
2269/CHENP/2006 22-06-2006 251463 19-03-2012 A PHARMACEUTICAL COMPOSITION COMPRISING AN LEK PHARMACEUTICALS D.D.
ACTIVE PRINCIPLE AND SULPHOBETAINE
431/CAL/1999 10-05-1999 251480 20-03-2012 INHIBITORS OF p38 VERTEX PHARMACEUTICALS
INCORPORATED
8276/DELNP/2007 26-10-2007 251484 20-03-2012 "PYRROLIDINE COMPOUND OF GENERAL FORMULA(I)" OTSUKA PHARMACEUTICAL CO., LTD.,

1850/KOLNP/2005 16-09-2005 251492 20-03-2012 A NASAL PHARMACEUTICAL FORMULATION MERCK PATENT GMBH
1192/DEL/2002 27-11-2002 251502 21-03-2012 "A COMPOSITION COMPRISING COMPONENT A AND ROHM AND HAAS COMPANY
COMPONENT B"
2104/MUMNP/2008 30-09-2008 251513 21-03-2012 BIPHENYL AMIDELACTAM DERIVATIVES AS INHIBITORS ELI LILLY AND COMPANY
OF 11 - BETA - HYDROXYSTEROID DEHYDROGENASE 1

1684/MUM/2008 08-08-2008 251524 21-03-2012 A NOVEL PHARMACEUTICAL COMPOSITION OF TOPICAL MRS. ANURADHA MAJUMDAR
METHOTREXATE GEL IN CHRONIC INFLAMMATORY
CONDITION
4926/KOLNP/2007 19-12-2007 251525 21-03-2012 HISTAMINE H3 RECEPTOR AGENTS, PREPARATION AND ELI LILLY AND COMPANY
THERAPEUTIC USES
1885/DEL/2005 20-07-2005 251564 23-03-2012 "COMPOSITIONS WITH CYCLOPROPENES AND METAL- ROHM AND HAAS COMPANY
COMPLEXING AGENTS"
1796/KOLNP/2007 21-05-2007 251577 26-03-2012 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT TOYAMA CHEMICAL CO., LTD.
THEREOF
3158/DEL/2005 25-11-2005 251579 26-03-2012 "NOVEL LOGANIN ANALOGUES AND A PROCESS FOR COUNCIL OF SCIENTIFIC & INDUSTRIAL
THE PREPARATION THEREOF" RESEARCH
5293/DELNP/2006 13-09-2006 251580 26-03-2012 "COMPOSITIONS AND METHODS FOR REDUCING OR NESTEC S.A.
PREVENTING OBESITY"
IN/PCT/2002/00308/MUM 13-03-2002 251589 26-03-2012 CICLESONIDE CONTAINED PHARMACEUTICAL NYCOMED GMBH,
COMPOSITION FOR APPLICATION TO MUCOSA
1770/MUM/2008 22-08-2008 251593 26-03-2012 A MICROEMULSION BASED INTRANASAL DRUG AMRITA BAJAJ
DELIVERY SYSTEM AND METHOD FOR PREPARATION
THEREOF
1701/MUMNP/2008 07-08-2008 251601 26-03-2012 MICROTABLET-BASED PHARMACEUTICAL PREPARATION BIOGENERICS PHARMA GMBH

2876/KOLNP/2007 07-08-2007 251605 26-03-2012 SUBSTITUTED THIOPHENES AS GLUCAGON RECEPTOR ELI LILLY AND COMPANY
ANTAGONISTS
2238/CHENP/2006 21-06-2006 251654 27-03-2012 A PHARMACEUTICAL COMPOSITION AND A METHOD DAIICHI SANKYO COMPANY, LIMITED
FOR PROLIFERATING CARDIOMYOCYTES
5502/DELNP/2007 17-07-2007 251668 27-03-2012 "A 4"-SUBTITUTED 8A OR 9A-LACTAM 15-MEMBERED GLAXO GROUP LIMITED.
MACROLIDE COMPOUND OF FORMULA (I)"

2966/DELNP/2007 20-04-2007 251671 27-03-2012 ALKIL-PYRIDINE COMPOUNDS F.HOFFMANN-LA ROCHE AG


2626/MUMNP/2008 10-12-2008 251679 28-03-2012 HETEROCYCLIC NON-NUCLEOSIDE COMPOUNDS, SHANGHAI INSTITUTE OF MATERIA
MEDICA CHINESE ACADEMY OF
SCIENCES
5889/DELNP/2007 27-07-2007 251739 30-03-2012 "A QUINAZOLINE DERIVATIVE" HANMI HOLDINGS CO., LTD.
2970/KOLNP/2007 14-08-2007 251793 03-04-2012 SUBSTITUTED IMIDAZO[1,2-b] PYRIDAZINE COMPOUND ELI LILLY AND COMPANY

7324/DELNP/2006 05-12-2006 251800 03-04-2012 "3-{(3R,4R)-4-METHYL-3-[METHYL-(7H-PYRROLO[2,3- PFIZER PRODUCTS INC


D]PYRIMIDIN-4-YL)-AMINO]-PIPERIDIN-1-YL}-3-OXO-
PROPIONITRILE MONO CITRATE SALT AND ITS METHOD
OF PREPARATION"
781/DEL/2003 05-06-2003 251801 04-04-2012 "A FEXOFENADINE-CARBOMER COMPLEX" M/S. IND-SWIFT LIMITED
910/MUMNP/2008 06-05-2008 251804 04-04-2012 NERAMEXANE MODIFIED RELEASE MATRIX TABLET MERZ PHARMA GMBH & CO. KGAA
613/MUMNP/2009 30-03-2009 251805 04-04-2012 1, 5-DIPHENYL-3-PYRIDINYLAMINO-1, 5- ELI LILLY AND COMPANY
DIHYDROPYRROLIDIN-2-ONE AS CB1 RECEPTOR
MODULATOR
203/CHENP/2008 11-01-2008 251826 10-04-2012 INDOL-3-CARBONYL-SPIRO-PIPERIDINE DERIVATIVES AS F. HOFFMANN-LA ROCHE AG
VIA RECEPTOR ANTAGONISTS
8313/DELNP/2007 29-10-2007 251828 10-04-2012 "MOTILIDE COMPOUNDS" PFIZER INC.
949/MUMNP/2006 10-08-2006 251841 11-04-2012 EXTENDED RELEASE COATED MINITABLETS OF ALEMBIC LIMITED
VENLAFAXINE HYDROCHLORIDE
2474/KOLNP/2006 30-08-2006 251854 12-04-2012 CASPASE INHIBITORS AND USES THEREOF VERTEX PHARMACEUTICALS
INCORPORATED
1816/KOLNP/2007 22-05-2007 251857 12-04-2012 A LUBRICANT COMPOSITION HCB HAPPY CHILD BIRTH HOLDING AG.

5334/DELNP/2006 14-09-2006 251863 12-04-2012 "PHARMACEUTICAL COMPOSITION AND PROCESS FOR SOLVAY PHARMACEUTICALS GMBH.
THEIR PREPARATION"
4253/CHENP/2006 17-11-2006 251875 12-04-2012 NOVEL CIS-IMIDAZOLINES HAVING ANTIPROLIFERATIVE F. HOFFMANN-LA ROCHE AG
ACTIVITY
IN/PCT/2000/00792/MUM 29-12-2000 251878 13-04-2012 C-TERMINAL MODIFIED OXAMYL DIPEPTIDES AS IDUN PHARMACEUTICALS, INC.,
INHIBITORS OF THE ICE/CED-3 FAMILY OF CYSTEINE
PROTEASES
5209/DELNP/2007 06-07-2007 251908 17-04-2012 "SUBSTITUTED TRIAZOLE COMPOUNDS AS OXYTOCIN PFIZER LIMITED
ANTAGONISTS"
IN/PCT/2002/484/KOL 18-04-2002 251919 17-04-2012 QUINOLINE DERIVATIVES FOR THE TREATMENT OF ACTIVE BIOTECH AB
MALIGNANT TUMORS
305/KOLNP/2007 25-01-2007 251921 17-04-2012 INHIBITORS OF VEGF RECEPTOR AND HGF RECEPTOR METHYLGENE, INC.
SIGNALING
3362/DELNP/2007 04-05-2007 251922 17-04-2012 "A BOTANICAL DRUG SUBSTANCE OBTAINABLE FROM GW PHARMA LIMITED
BOTANICAL RAW MATERIAL"
7575/DELNP/2007 03-10-2007 251929 18-04-2012 A PHARMACUTICAL COMPOSITION CONTAINING WARNER CHILCOTT COMPANY,LLC
RISEDRONATE
2888/KOLNP/2006 06-10-2006 251939 18-04-2012 SUBSTITUTED ORGANOSULFUR COMPOUNDS AND ACEA BIOSCIENCES INC.
PHARMACEUTICAL COMPOSITION COMPRISING THEM

4769/KOLNP/2007 10-12-2007 251944 18-04-2012 FORMULATION OF A THIENOPYRIDINE PLATELET ELI LILLY AND COMPANY
AGGREGATION INHIBITOR
2052/KOLNP/2006 21-07-2006 251946 18-04-2012 NOVEL FUSED PYRROLOCARBAZOLES CEPHALON, INC.
436/KOLNP/2007 07-02-2007 251952 18-04-2012 METHOD AND COMPOSITION FOR HIGH LEVEL NANOSONICS PTY LIMITED
DISINFECTION EMPLOYING QUATERNARY AMMONIUM
COMPOUNDS
232/KOLNP/2007 18-01-2007 251957 18-04-2012 "NEW 4-BENZYLIDENE-PIPERIDIN DERIVATIVES" RICHTER GEDEON VEGYÉSZETI GYÁR RT.

1308/KOLNP/2008 01-04-2008 251964 18-04-2012 CYCLIC AMINE COMPOUNDS AND PESTICIDAL NIPPON SODA CO., LTD.
COMPOSITION COMPRISING THEM
5059/DELNP/2006 01-09-2006 251968 18-04-2012 "A FUSED HETEROCYCLE DERIVATIVE AND KISSEI PHARMACEUTICAL CO., LTD
PHARMACEUTICAL COMPOSITION COMPRISING THE
SAME"
3400/DELNP/2007 07-05-2007 251979 19-04-2012 "HETEROCYCLIC COMPOUNDS SUITABLE FOR TREATING ABBOTT GMBH & CO. KG
DISORDERS THAT RESPOND TO MODULATION OF THE
DOPAMINE D3 RECEPTOR"
4247/DELNP/2006 24-07-2006 251981 19-04-2012 A STABLE SOLID PHARMACEUTICAL COMPOSITION ACTIVE BIOTECH AB
CONTAINING QUINOLINE COMPOUNDS AND PROCESS
THEREOF
2453/KOLNP/2006 29-08-2006 251984 19-04-2012 CHEMICALLY STABLE COMPOSITIONS OF 4- HYDROXY LABORATOIRES BESINES
TAMOXIFEN INTERNATIONAL
3547/DELNP/2006 20-06-2006 251990 19-04-2012 "AN AZABICYCLO-INDAZOLE COMPOUND" MEMORY PHARMACEUTICALS
CORPORATION
6842/DELNP/2006 16-11-2006 252033 23-04-2012 "COMPOUNDS AND COMPOSITIONS AS PROTEIN IRM LLC
KINASE INHIBITORS"
1943/KOLNP/2006 11-07-2006 252043 23-04-2012 ACYLAMINOTHIAZOLE DERIVATIVES AND USE THEREOF SANOFI-AVENTIS
AS BETA-AMYLOID INHIBITORS
2332/KOLNP/2006 17-08-2006 252044 23-04-2012 "DERIVATIVES OF PIPERIDINYLALKYLCARBAMATES, SANOFI AVENTIS
PREPARATION METHOD THEREOF AND USE OF SAME
AS FAAH ENZYME INHIBITORS"
2877/DELNP/2006 22-05-2006 252046 23-04-2012 "A COMPOUND OF 1-BENZYLAMINO-2CARBAMOYL- NEWRON PHARMACEUTICALS S.P.A
CYELOPENTANE DERIVATIVES OF FORMULA 1"
1462/KOLNP/2005 27-07-2005 252078 25-04-2012 A MEDICAMENT FOR THE PROPHYLAXIS AND DAIICHI SANKYO COMPANY LIMITED
TREATMENT OF ARTERIOSCLEROSIS AND
HYPERTENSION
3325/KOLNP/2006 13-11-2006 252091 25-04-2012 PHARMACEUTICAL TABLETS HAVING A RELATIVELY ACCU-BREAK TECHNOLOGIES INC.
INACTIVE SEGMENT
605/KOLNP/2007 20-02-2007 252108 25-04-2012 2-DEOXY-2-FLUORO-2-METHYL-D-RIBONOLACTONE PHARMASSET, INC.
DERIVATIVES AND PROCESS FOR PREPARATION OF THE
SAME
2306/KOLNP/2007 22-06-2007 252109 25-04-2012 NOVEL RECEPTOR ANTAGONISTS OF MELANIN ELI LILLY AND COMPANY
CONCENTRATING HORMONE
1646/CHENP/2006 11-05-2006 252114 26-04-2012 PENTAFLUOROSULFANYL BENZOYLGUANIDINES, SANOFI-AVENTIS DEUTSCHLAND GMBH
METHOD FOR THEIR PRODUCTION, THEIR USE AS
MEDICAMENTS OR DIAGNOSTIC AGENTS AND
MEDICAMENT CONTAINING THE SAME
2774/DELNP/2006 17-05-2006 252120 26-04-2012 "NOVEL PHENOL DERIVATIVES AND ARIGEN PHARMACEUTICALS INC.,
ANTITRYPANOSOMA PREVENTIVE/THERAPEUTIC AGENT
COMPRISING THE SAME AS ACTIVE INGREDIENT"

1825/MUMNP/2009 01-10-2009 252131 27-04-2012 TRIAZOLYL AMINOPYRIMIDINE COMPOUNDS ELI LILLY AND COMPANY
7959/DELNP/2006 28-12-2006 252132 27-04-2012 "A SUBSTITUTED 2-ALKYL QUINAZOLINONE DERIVATIVE JANSSEN PHARMACEUTICA N.V
OF FORMULA (I)"
702/MUMNP/2009 13-04-2009 252133 27-04-2012 TETRAHYDROCYCLOPENTA[B] INDOLE COMPOUNDS AS ELI LILLY AND COMPANY
ANDROGEN RECEPTOR MODULATORS

2825/DELNP/2004 22-09-2004 252137 27-04-2012 "THIOXANTHINE DERIVATIVES AS MYELOPEROXIDASE ASTRAZENECA AB


INHIBITORS"
4429/DELNP/2006 01-08-2006 252144 30-04-2012 "N-DEACETYLTHIOCOLCHICINE DERIVATIVES, THEIR USE INDENA S.P.A.
AND PHARMACEUTICAL FORMULATIONS CONTAINING
THEM"
4298/DELNP/2005 22-09-2005 252150 30-04-2012 "PYRROLE COMPOUNDS AS MODULATORS OF MERCK & CO. INC.
METABOTROPIC GLUTAMATE RECEPTOR-5"
5054/DELNP/2006 01-09-2006 252159 30-04-2012 PYRAZOLYL INDOLYL COMPOUNDS F. HOFFMANN-LA ROCHE AG
1863/DEL/2006 21-08-2006 252163 30-04-2012 "A NOVEL HERBAL COMPOSITION AND A PROCESS FOR CENTRAL COUNCIL FOR RESEARCH IN
PREPARATION THEREOF EFFECTIVE AGAINST UNANI MEDICINE
ABDOMINAL WORM ."
2724/DEL/2005 10-10-2005 252167 30-04-2012 OXY SUBSTITUTED CHALCONES AS COUNCIL OF SCIENTIFIC AND
ANTIHYPERGLYCEMIC AND ANTIDYSLIPIDEMIC AGENTS INDUSTRIAL RESEARCH

1518/DELNP/2005 15-04-2005 252201 01-05-2012 "A PHARMACEUTICAL COMPOSITION" FICAAR INC.


3229/CHENP/2006 05-09-2006 252203 01-05-2012 DIAMINOPYRIMIDINES AS P2X3 AND P2X2/3 F. HOFFMANN-LA ROCHE AG
ANTAGONISTS
2452/CHENP/2006 05-07-2006 252204 01-05-2012 POLYPEPTIDES OF ALICYCLOBACILLUS SP NOVOZYMES A/S
649/MUMNP/2006 06-06-2006 252206 01-05-2012 PHARMACEUTICAL COMPOSITION CONTAINING Senju Pharmaceutical Co.Ltd.
PROSTAGLANDIN
3263/DEL/2005 05-12-2005 252211 01-05-2012 "NATURAL CALCLUM CARBONATE TOOTHPOWDER COLGATE-PALMOLIVE COMPANY
COMPOSITIONS"
188/DELNP/2003 19-02-2003 252221 02-05-2012 " HARD CAPSULE PREPARED FROM POLYMERIZABLE NISSHIN KASEI CO., LTD.,
VINYL MONOMER OF FORMULA H2C=C(R1)-COOR2 "

1473/KOLNP/2006 31-05-2006 252229 02-05-2012 NOVEL NITROPHENYL MUSTARD AND AUCKLAND UNISERVICES LIMITED
NITROPHENYLAZIRIDINE ALCOHOLS AND THEIR
CORRESPONDING PHOSPHATES AND THEIR USE AS
TARGETED CYTOTOXIC AGENT
3549/DELNP/2006 20-06-2006 252268 04-05-2012 "COBALAMINE DERIVATIVES USEFUL FOR DIAGNOSIS SOLIDAGO AG.
AND TREATMENT OF ABNORMAL CELLULAR
PROLIFERATION "
2201/CHENP/2006 19-06-2006 252274 04-05-2012 IMMUNOSTIMULANT COMPOSITION COMPRISING AT SANOFI PASTEUR
LEAST ONE TOLL-LIKE RECEPTOR 7 OR TOLL-LIKE
RECEPTOR 8 AGONIST AND A TOLL-LIKE RECEPTOR 4
AGONIST
1267/CHENP/2006 13-04-2006 252299 08-05-2012 AMINOALKANOL DERIVATIVES NOVARTIS AG
1661/KOLNP/2006 15-06-2006 252305 08-05-2012 A PHARMACEUTICAL COMPOSITION MERCK EPROVA AG
1295/KOLNP/2007 12-04-2007 252311 08-05-2012 NOVEL COMPOUNDS AS BRADYKININ RECEPTOR ISTITUTO LUSO FARMACO D'ITALIA
ANTAGONIST AND COMPOSITION THEREFROM S.P.A.
3127/DEL/2005 23-11-2005 252316 08-05-2012 "A HERBAL HEALTH FORMULATION" Three-N-Products Pvt. Ltd.
1980/KOLNP/2007 01-06-2007 252351 09-05-2012 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AND FERRER INTERNACIONAL S.A.
COMPOSITIONS
352/CHENP/2008 22-01-2008 252366 10-05-2012 IMPROVED POLYSACCHARIDE-BASED SOLID GRANULES RHODIA OPERATIONS

1724/CHENP/2006 17-05-2006 252367 10-05-2012 DIPEPTIDYL PEPTIDASE IV INHIBITORS COMPOSITION NOVARTIS AG

2319/DELNP/2007 26-03-2007 252371 10-05-2012 INDOZOLONE DERIVATIVES AS 11B-HSD 1 INHIBITORS H.HOFFMANN-LA ROCHE AG

3432/CHENP/2006 19-09-2006 252374 11-05-2012 A PEPTIDE COMPOSITION FOR IMMUNE DIAGNOSTIC ISTITUTO NAZIONALE PER LE MALATTIE
ASSAY TO DIAGNOSE AND MONITOR TUBERCULOSIS INFETTIVE "LAZZARO SPALLANZANI"
INFECTION IRCCS
2247/KOLNP/2006 08-08-2006 252397 14-05-2012 NOVEL COMPOUNDS FOR INHIBITING FAAH ENZYME, SANOFI AVENTIS
PROCESS FOR THE PREPARATION THEREOF AND
PHARMACEUTICAL COMPOSITION CONTAINING THE
SAME
3563/KOLNP/2006 28-11-2006 252407 14-05-2012 SUBSTITUTED INDAZOLES, COMPOSITIONS AVENTIS PHARMA SA
CONTAINING SAME, PREPARATION AND USE
IN/PCT/2001/31/KOL 09-01-2001 252425 15-05-2012 QUINOLINE DERIVATIVES ACTIVE BIOTECH AB
506/MUMNP/2009 12-03-2009 252432 15-05-2012 SUBSTITUTED THIAZOLE PYRAZOLOPYRIMIDINE ELI LILLY AND COMPANY
COMPOUNDS AS CRF1 RECEPTOR ANTAGONISTS
499/MUMNP/2009 09-03-2009 252439 16-05-2012 “THIOPHENE PYRAZOLOPYRIMIDINE COMPOUNDS” ELI LILLY AND COMPANY

380/MUMNP/2009 18-02-2009 252441 16-05-2012 “COMBINATION OF MODAFINIL AND AN ANTAGONIST BIOPROJET


OR INVERSE AGONIST OF THE H3 RECEPTOR”

3557/DELNP/2006 20-06-2006 252445 16-05-2012 "PHOSPHONATES, MONOPHOSPHONAMIDATES, GILEAD SCIENCES, INC.


BISPHOSPHONAMIDATES FOR THE TREATMNET OF
VIRAL DISEASES "
1282/MUMNP/2007 22-08-2007 252449 16-05-2012 COMPOSITION FOR REDUCING THE EXUDATION OF THE CHOI SEONG-HYUN
SERUM PROTEINS
3624/DELNP/2006 23-06-2006 252466 16-05-2012 HETEROARYL-UREAS AND THEIR USE AS GLUCOKINASE NOVO NORDISK A/S
ACTIVATORS
2448/DEL/2005 12-09-2005 252478 17-05-2012 "SUSTAINED RELEASE SYRUP COMPOSITION AND DELHI INSTITUTE OF PHARMACEUTICAL
PROCESS THEREOF" SCIENCES & RESEARCH

3854/DELNP/2006 05-07-2006 252483 17-05-2012 "MICROCYCLIC PROLINE ANALOGUES AS HCV NS-3 MEDIVIR AB
SERINE PROTEASE INHIBITORS"
7656/DELNP/2007 05-10-2007 252486 17-05-2012 "THE COMPOUND OF 1-METHYL-1H-IMIDAZOLE-4- PFIZER PRODUCTS INC.
CARBOXYLIC ACID (3-AZA-BICYCLO[3.1.0]HEX-6-
YLMETHYL)-(3-CHLORO-4-FLUORO-BENZYL)-AMIDE"
2978/DELNP/2008 10-04-2008 252491 18-05-2012 "IONTOPHORETIC PREPARATION FOR TREATMENT OF KOWA CO. , LTD.
BREAST CANCER AND/OR MASTITIS"
697/DELNP/2004 18-03-2004 252493 18-05-2012 "A COMPOSITION COMPRISING AN ISOMERIC MEXTURE PALADIN LABS INC.
OF A CYCLOSPORINE ANALOGUE'
2702/DELNP/2004 14-09-2004 252499 18-05-2012 "A SUBSTITUTED BENZIMIDAZOLE SULFONAMIDE TIBOTEC PHARMACEUTICALS LTD
COMPOUND AND A PHARMACEUTICAL COMPOSITION
COMPRISING THE SAME"
4837/DELNP/2007 22-06-2007 252509 21-05-2012 PHARMACEUTICAL , THERAPEUTIC, AND DIETARY RENAISSANCE HERBS, INC.
COMPOSITIONS DERIVED FROM LEAVES OF
LAGERSTROEMIA SPECIOSAL I. PLANT
7590/DELNP/2006 15-12-2006 252518 21-05-2012 "AMINOCYCLOHEXANES AS DIPEPTIDYL PEPTIDASE-IV MERCK SHARP & DOHME CORP.
INHIBITORS FOR THE TREATMENT OR PREVENTION OF
DIABETES"
1521/DELNP/2007 26-02-2007 252533 21-05-2012 INDOLE COMPOUNDS COMRISING AN ACETYLENE F. HOFFMANN-LA-ROCHE AG
GROUP AS PPAR ACTIVATORS
8778/DELNP/2007 15-11-2007 252535 21-05-2012 "PHARMACEUTICAL COMPOSITION COMPRISING AN ADVANCED SCIENTIFIC DEVELOPMENTS
ANTIVIRAL AGENT, AN ANTITUMORAL AGENT OR AN
ANTIPARASITIC AGENT, AND AN ACTIVE AGENT
SELECTED AMONG CARVEOL, THYMOL, EUGENOL,
BORNEOL AND CARVACROL"
9905/DELNP/2007 20-12-2007 252541 21-05-2012 "MAO-B INHIBITORS USEFUL FOR TREATING OBESITY" JENRIN DISCOVERY

963/MUMNP/2009 14-05-2009 252549 22-05-2012 “IMIDAZOLIDINONYL AMINOPYRIMIDINE ELI LILLY AND COMPANY
COMPOUNDS"
855/MUM/2006 01-06-2006 252567 23-05-2012 A PROCESS FOR PREPARATION OF A POLYHERBAL CHARAK PHARMA PRIVATE LIMITED
COMPOSITION AND THE PRODUCT THEREOF
1931/MUMNP/2008 08-09-2008 252574 23-05-2012 CAMPTOTHECIN DERIVATIVES SHANGHAI INSTITUTE OF MATERIA
MEDICA, CHINESE ACADEMY OF
SCIENCES
1/DEL/2004 01-01-2004 252589 23-05-2012 "SOLID PHASE BENZOPYRAN COMPOSITION, PROCESS INTERNATIONAL FLAVORS &
FOR PREPARING SAME" FRAGRANCES INC.
1314/DEL/2004 16-07-2004 252592 23-05-2012 A TOPICAL FORMULATION FOR PREVENTION AND THE DIRECTOR GENERAL
MANAGEMENT OF PERIPHERAL VASCULAR DISEASES
AND A PROCESS OF PREPARATION THEREOF

5248/DELNP/2007 06-07-2007 252599 23-05-2012 "ORAL COMPOSITIONS CONTAINING BIPHENOL COLGATE-PALMOLIVE COMPANY
ANTIBACTERIAL COMPOUNDS"
6544/DELNP/2006 06-11-2006 252605 23-05-2012 "A 2-PYRROLIDIN-OR-2-PIPERIDINONE DERIVATIVE OF JANSSEN PHARMACEUTICA N.V.,
FORMULA (I)"
26/MUMNP/2009 02-01-2009 252606 23-05-2012 GLUCOCORTICOID RECEPTOR MODULATOR ELI LILLY AND COMPANY
3402/DELNP/2004 02-11-2004 252607 23-05-2012 "HYDROXY TETRAHYDRO-NAPHTHALENYLUREA XENTION LIMITED.,
DERIVATIVES"
2936/CHENP/2006 10-08-2006 252617 24-05-2012 CHEMOKINE RECEPTOR ANTAGONISTS NOVARTIS AG
999/DELNP/2006 24-02-2006 252629 24-05-2012 "HETEROARYL-TETRAHYDROPIPERIDYL COMPOUNDS EUROCELTIQUE S. A.
USEFUL FOR TREATING OR PREVENTING PAIN"

3727/DELNP/2006 28-06-2006 252647 25-05-2012 "A COMPOSITION CONTAINING A LYOPHILISATE OF BIOTECHMARINE.


DEDIFFERENTIATED PLANT CELLS FOR SKIN
DEPIGMENTATION"
4015/DELNP/2004 16-12-2004 252658 25-05-2012 " A PHARMACEUTICAL COMPOSITION FOR THE FIDELINE
TREATMENT OF STRESS IN AN AVIAN"
7188/DELNP/2006 29-11-2006 252687 28-05-2012 "A PHARMACEUTICAL COMPOSITION COMPRISING M3 ALMIRALL S.A.
ANTAGONIST AND B2-AGONIST FOR USE IN THE
RESPIRATORY DISORDERS"
272/MUMNP/2006 08-03-2006 252689 28-05-2012 6-CYCLOAMINO-2-QUINOLINONE DERIVATIVES AS LIGAND PHARMACEUTICALS
ANDROGEN RECEPTOR MODULATOR COMPOUNDS INCORPORATED
3341/DELNP/2004 27-10-2004 252695 28-05-2012 A COMPOSITION FOR THE TREATMENT OF OBESITY DUKE UNIVERSITY
705/DELNP/2006 13-02-2006 252720 29-05-2012 "CALCIUM CARBONATE GRANULATION" DELAVAU L.L.C
1848/CHENP/2006 25-05-2006 252776 30-05-2012 COMPOUNDS WITH SUBSTITUTED IMIDAZO RING 3M INNOVATIVE PROPERTIES
SYSTEMS COMPANY
951/MAS/2002 18-12-2002 252779 30-05-2012 NOVEL TETRACYCLIC 3-SUBSTITUTED INDOLES HAVING SUVEN PHARMACEUTICALS LTD
SEROTONIN RECEPTOR AFFINITY AND PROCESS FOR
THEIR PREPARATION
332/KOLNP/2007 29-01-2007 252786 30-05-2012 "THIENOPYRAZOLE DERIVATIVE HAVING PDE7 DAIICHI SANKYO CO., LTD.
INHIBITORY ACTIVITY"
2501/DELNP/2004 26-08-2004 252787 30-05-2012 "PHARMACEUTICAL AEROSOL FORMULATION OF CHIESI FARMACEUTICI S.p.A.
FORMOTEROL FUMARATE TO BE ADMINISTERED BY A
PRESSURIZED METERED DOSE INHALER"
2010/DEL/2004 15-10-2004 252796 31-05-2012 "AMIDE DERIVATIVES" ASTRAZENECA AB
1820/DELNP/2006 03-04-2006 252801 31-05-2012 AN ANTHRAPYRIDONE OF THE FORMULA (I) SABIC INNOVATIVE PLASTICS IP B.V.
778/DELNP/2007 31-01-2007 252825 01-06-2012 ARYL-PYRIDINE COMPOUNDS F. HOFFMANN-LA ROCHE AG
607/DELNP/2007 23-01-2007 252833 04-06-2012 "TRIAZOLOPYRIDINYLSULFANYL DERIVATIVES AS P38 PFIZER INC
MAP KINASE INHIBITORS"
9927/DELNP/2007 20-12-2007 252838 04-06-2012 "SULFONAMIDE DERIVATIVES USEFUL AS LIVER F. HOFFMANN-LA ROCHE AG
CARNITINE PALMITOYL TRANSFERASE (L-CPT1)
INHIBITORS"
498/MUMNP/2009 09-03-2009 252845 04-06-2012 “COMPOSITIONS OF CHK1 INHIBITORS” ICOS CORPORATION
381/KOLNP/2007 02-02-2007 252855 05-06-2012 "THIENOPYRIMIDINES USEFUL AS AURORA KINASE SUNESIS PHARMACEUTICALS, INC.
INHIBITORS".
1767/KOLNP/2006 23-06-2006 252877 06-06-2012 "STEREOISOMERIC COMPOUNDS AND METHODS FOR ARYX THERAPEUTICS
THE TREATMENT OF GASTROINTESTINAL AND CENTRAL
NERVOUS SYSTEM DISORDERS"
510/MUMNP/2009 13-03-2009 252901 07-06-2012 “ORAL RECOMBINANT HELICOBACTER PYLORI VACCINE CHONGQING KANG WEI
AND PREPARING METHOD THEREOF” BIOTECHNOLOGY CO. LTD.
489/MUMNP/2007 04-04-2007 252902 07-06-2012 PHARMACEUTICAL COMPOSITION COMPRISING AN CIPLA LIMITED
ISOMER OF A BETAMIMETIC AGENT AND AN ANTI-
CHOLINERGIC AGENT
2916/CHENP/2007 02-07-2007 252910 08-06-2012 BORON-CONTAINING MOLECULAR SIEVE CHA CHEVRON U.S.A INC.
3646/KOLNP/2006 05-12-2006 252936 11-06-2012 COMPOSITIONS AND METHODS TO PREVENT AAV GENZYME CORPORATION
VECTOR AGGREGATION
2089/CHENP/2006 12-06-2006 252964 12-06-2012 SPIROINDOLINE DERIVATIVES HAVING INSECTICIDAL SYNGENTA PARTICIPATIONS AG
PROPERTIES
1268/DEL/2003 14-10-2003 252981 13-06-2012 "TRICYCLIC COMPOUNDS HAVING ANTIOXIDANT NATIONAL INSTITUTE OF
PROPERTIES" PHARMACEUTICAL EDUCATION AND
RESEARCH (NIPER)
3429/DELNP/2006 14-06-2006 252982 13-06-2012 "PYRAZOLE DERIVATIVES AS PROTEIN KINASE ASTEX THERAPEUTICS LIMITED
MODULATORS"
2451/KOLNP/2006 28-08-2006 252989 13-06-2012 2H OR 3H-BENZO[E]INDAZOL-1-YLE CARBAMATE SANOFI AVENTIS
DERIVATIVES, AND THEIR PREPARATION
1851/CHENP/2006 26-05-2006 252990 13-06-2012 NOVEL ANALGESIC COMPOUNDS, EXTRACTS GRIFFITH UNIVERSITY
CONTAINING SAME AND METHODS OF PREPARATION

2888/DELNP/2006 22-05-2006 253024 15-06-2012 "A COMPOSITION, FOR THE TREATMENT OF AN INDENA S.P.A.
AFECTION OF THE ORAL CAVITY AND UPPER
RESPIRATORY TRACT"
1939/MUM/2006 24-11-2006 253029 15-06-2012 CCR5 MODULATOR COMPOUNDS PHIVCO-1 LLC
443/MUMNP/2006 18-04-2006 253030 15-06-2012 SUBSTITUTED DIAZABICYCLOALKANE DERIVATIVES AS ABBOTT LABORATORIES
LIGANDS AT ALPHA 7 NICOTINIC ACETY LCHOLINE
RECEPTORS.
2180/DELNP/2007 21-03-2007 253033 18-06-2012 "A COMPOSITION FOR PREVENTING OR IMPROVING OTSUKA PHARMACEUTICAL CO., LTD.,
PIGMENTATION"
4720/DELNP/2006 17-08-2006 253042 19-06-2012 "A DIKETOPIPERAZINE" NEREUS PHARMACEUTICALS, INC.
145/CHENP/2008 09-01-2008 253053 20-06-2012 COMPOUND EXHIBITING GLUCOKINASE ACTIVATION MITSUBISHI TANABE PHARMA
AND ITS PREPARATION THEREOF CORPORATION
1331/CAL/1998 29-07-1998 253099 25-06-2012 4-OXO-3,5-DIHYDRO-4H-PYRIDAZINO[4,5-b] INDOLE-1- SANOFI AVENTIS
ACETAMIDE-DEIVATIVES
393/MUMNP/2008 29-02-2008 253106 26-06-2012 A COMPOSITION COMPRISING PHARMACEUTICAL- GLOBOASIA LLC
GRADE FERRIC CITRATE EFFECTIVE IN REDUCING
SERUM PHOSPHATE LEVEL
3268/KOLNP/2006 08-11-2006 253108 26-06-2012 AZASUGAR DERIVATIVES, HEPARANASE INHIBITORS SANOFI-AVENTIS
AND PHARMACEUTICAL COMPOSITIONS THEREOF
4470/DELNP/2006 02-08-2006 253109 26-06-2012 "TETRAZOLE COMPOUND AND COMPOSITION ASTRAZENECA AB
THEREOF"
3685/CHENP/2006 05-10-2006 253139 27-06-2012 HYALURONIC ACID-METHOTREXATE CONJUGATE DENKI KAGAKU KOGYO KABUSHIKI
KAISHA
571/DEL/2007 16-03-2007 253149 28-06-2012 "A COMPOUND USEFUL AS PHARMACEUTICALS, WHITE FLOWER ASSOCIATES LLP
AVERSIVE AGENTS AND/OR ANTIFOULANTS"
5184/DELNP/2006 08-09-2006 253159 28-06-2012 "A COMPOSITION COMPRISING GLYPHOSPHATE AND FMC CORPORATION
AT LEAST ONE TAURATE SALT"
2120/DELNP/2006 19-04-2006 253168 29-06-2012 "SOLID PHARMACEUTICAL COMPOSITION" BAYER ANIMAL HEALTH GMBH
4557/DELNP/2005 06-10-2005 253179 29-06-2012 "ORAL FORMULATIONS OF CLADRIBINE" ARES TRADING S.A.,
644/KOLNP/2007 22-02-2007 253193 04-07-2012 COMPOUND OF FORMULA (I) FOR TREATMENT OF IVAX DRUG RESEARCH INSTITUTE LTD.
INFLAMMATORY DISEASES OF THE AIRWAY
764/CHENP/2008 14-02-2008 253217 04-07-2012 PIPERIDINE AND PIPERAZINE DERIVATIVES AS P2X3 F. HOFFMANN-LA ROCHE AG
ANTAGONISTS
2870/DELNP/2006 19-05-2006 253261 09-07-2012 PYRAZOLE DERIVATIVES AS INHIBITORS OF RECEPTOR ASTRAZENECA AB
TYROSYNE KINASES
511/KOLNP/2007 12-02-2007 253273 10-07-2012 SUBSTITUTED QUINOLONES AICURIS GMBH & CO. KG,
982/KOLNP/2007 20-03-2007 253276 10-07-2012 POLYPHOSPHATE DERIVATIVE OF A 1,3,5-TRIAZINE CHEMISCHE FABRIK BUDENHEIM KG.
COMPOUND, A PROCESS FOR THE PRODUCTION
THEREOF
3937/KOLNP/2006 28-12-2006 253283 10-07-2012 "TRICYCLIC INDENO-PYRROLE DERIVATIVES AS ATHERSYS, INC.
SEROTONIN RECEPTOR MODULATORS"
1484/KOLNP/2007 25-04-2007 253285 10-07-2012 COMPOSITION COMPRISING AN ACTIVE CORE CADBURY ADAMS USA LLC.
ENCAPSULATED BY MATRIX INCLUDING POLYMER AND
SUCRALOSE AND METHOD OF PREPARATION THEREOF

2681/DELNP/2006 12-05-2006 253290 11-07-2012 "A SUBSTITUTED AMIDE DERIVATIVE HAVING POTENT ASTRAZENECA AB
CYTOKINE INHIBITORY ACTIVITY"
2698/KOLNP/2007 20-07-2007 253297 11-07-2012 TRIOXEPANE COMPOSITION AND PROCESS FOR AKZO NOBEL N.V.
PREPARING TRIOXEPANE COMPOSITION
1574/KOLNP/2006 07-06-2006 253308 11-07-2012 A COMBINATION OF DEXAMETHASONE AND 4-AMINO- NOVARTIS VACCINES &amp;
5-FLUORO-3-[6-(4-METHYLPIPERAZIN-1-YL)-1H- DIAGNOSTICS S.R.L.,
BENZIMIDAZOL-2-YL]QUINOLIN-2(1H)-ONE A
TAUTOMER OR A PHARMACEUTICALLY ACCEPTABLE
SALT THEREOF
2096/MUMNP/2007 10-12-2007 253338 13-07-2012 PYRIMIDINE COMPOUNDS TAIGEN BIOTECHNOLOGY CO., LTD.
3684/CHENP/2006 05-10-2006 253384 17-07-2012 4-BENZYL-[1,2,4]THIADIAZOLIDINE-3,5-DIONE NOSCIRA S A
DERIVATIVES AS GSK-3 INHIBITORS
4138/DELNP/2007 31-05-2007 253414 18-07-2012 "A PIPERIDINYL INDOLE COMPOUND" EURO-CELTIQUE, S.A
621/KOLNP/2007 20-02-2007 253465 24-07-2012 "VACCINE FOR PREVENTION AND TREATMENT OF HIV- GLAXOSMITHKLINE BIOLOGICALS S.A.
INFECTION"
144/KOLNP/2007 11-01-2007 253477 25-07-2012 SUBSTITUTED IMIDAZOLE DERIVATIVES NOVARTIS VACCINES AND
DIAGNOSTICS, INC.
953/DELNP/2008 04-02-2008 253482 25-07-2012 BIS (THIO-HYDRAZIDE AMIDE) FORMULATION SYNTA PHARMACEUTICALS CORP.
3323/KOLNP/2006 13-11-2006 253493 25-07-2012 IMMEDIATE RELEASE PHARMACEUTICAL TABLETS WITH ACCU-BREAK TECHNOLOGIES INC.
HEIGHT GREATER THAN WIDTH
931/DELNP/2007 05-02-2007 253503 26-07-2012 "A 6-CYCLOPENTYL 4-HYDROXY-5,6-DIHYDRO-2-ONE PFIZER INC.
COMPOUND AND A PHARMACEUTICAL COMPOSITION
THEREOF"
444/KOLNP/2007 07-02-2007 253517 26-07-2012 BIVALENT LINKERS AND CONJUGATES THEREOF ENDOCYTE, INC.
388/KOLNP/2007 05-02-2007 253519 26-07-2012 HISTAMINE H3 RECEPTOR AGENTS, PREPARATION AND ELI LILLY AND COMPANY
THERAPEUTIC USES
1476/CHENP/2008 26-03-2008 253552 31-07-2012 OXADIAZOLYL PYRAZOLO-PYRIMIDINES AS MGLUR2 F. HOFFMANN-LA ROCHE AG
ANTAGONISTS
2692/DELNP/2006 12-05-2006 253571 01-08-2012 INJECTABLE SUSTAINED RELEASE IMPLANT HAVING A PSIVIDA INC.
BIOERODIBLE MATRIX CORE AND A BIOERODIBLE SKIN

3768/CHENP/2006 11-10-2006 253575 01-08-2012 TETRAHYDROPYRIDOINDOLE DERIVATIVES ACTELION PHARMACEUTICALS LTD


4136/DELNP/2007 31-05-2007 253581 02-08-2012 "A PIPERIDINYL CYANOIMINO-BENZIMIDAZOLE EURO-CELTIQUE, S.A.
COMPOUND OF FORMULA (IV)"
5205/DELNP/2006 11-09-2006 253587 03-08-2012 "COMPOSITION FOR ORAL ADMINISTRATION OF HANMI PHARM. CO., LTD.
TAMSULOSIN HYDROCHLORIDE"
2931/DELNP/2006 22-05-2006 253605 06-08-2012 2-PHENOXY PROPIONIC ACID COMPOUNDS AS PPAR F. HOFFMANN-LA ROCHE AG
AGONISTS
4625/KOLNP/2007 29-11-2007 253606 06-08-2012 HETEROAROYL-SUBSTITUTED SERINE AMIDES BASF AKTIENGESELLSCHAFT
3287/KOLNP/2006 09-11-2006 253619 07-08-2012 "TETRAHYDROISOQUINOLINE SULFONAMIDE SANOFI-AVENTIS
DERIVATIVES, THE PREPARATION THEREOF, AND THE
USE OF THE SAME IN THERAPEUTICS"
3518/CHENP/2006 25-09-2006 253630 08-08-2012 NOVEL ADENINE COMPOUND AND A PROCESS FOR DAINIPPON SUMITOMO PHARMA CO
PREPARING THE SAME LTD
9790/DELNP/2007 18-12-2007 253642 08-08-2012 "PHARMACEUTICAL COMPOSITION COMPRISING 2,3- OTSUKA PHARMACEUTICAL CO.,LTD.
DIHYDRO-6-NITROIMIDAZO[2,1-B]OXAZOLE
DERIVATIVES"
6872/DELNP/2006 17-11-2006 253644 08-08-2012 4-AMINO-5-CYANOPYRIMIDINE DERIVATIVES OTSUKA PHARMACEUTICAL CO., LTD
1223/KOLNP/2007 09-04-2007 253645 08-08-2012 A SUBSTITUTED CHROMAN DERIVATIVE MARSHALL EDWARDS, INC
690/MUMNP/2009 09-04-2009 253661 09-08-2012 A PHARMACEUTICAL FORMULATION BEN-GURION UNIVERSITY OF THE
NEGEV RESEACH AND DEVELOPMENT
AUTHORITY
3430/CHENP/2006 19-09-2006 253671 10-08-2012 PHARMACEUTICAL COMPOSITION COMPRISING A ARROW THERAPEUTICS LIMITED
BENZODIAZEPINE DERIVATIVE AND AN INHIBITOR OF
THE RSV FUSION PROTEIN
1046/MUMNP/2007 12-07-2007 253681 13-08-2012 TETRAHYDROQUINOLINE ANALOGUES ACADIA PHARMACEUTICALS INC
1522/MUMNP/2007 24-09-2007 253716 16-08-2012 SUBSTITUTED PYRIDINES AND PYRIDAZINES WITH BAYER CORPORATION
ANGIOGENESIS INHIBITING ACTIVITY
538/MUM/2006 05-04-2006 253721 17-08-2012 LIQUID ORAL FORMULATION CONTAINING STRIDES ARCOLAB LIMITED
FEXOFINADINE
952/KOLNP/2007 19-03-2007 253742 22-08-2012 MODULATORS OF MUSCARINIC RECEPTORS VERTEX PHARMACEUTICALS
INCORPORATED
7514/DELNP/2006 12-12-2006 253747 22-08-2012 "SUBSTITUTED HYDANTION COMPOUNDS FOR THE ASTRAZENECA AB
TREATMENT OF OBSTRUCTIVE AIRWAY DISEASE"
751/KOLNP/2007 01-03-2007 253750 22-08-2012 4-((PHENOXYALKYL) THIO)-PHENOXYACETIC ACIDS AND JANSSEN PHARMACEUTICA N.V.
ANALOGS
2579/KOLNP/2007 10-07-2007 253754 22-08-2012 N-(HETEROARYL)-1H-INDOLE-2-CARBOXAMIDE SANOFI AVENTIS
DERIVATIVES AND THEIR USE AS VANILLOID TRPV 1
RECEPTOR LIGANDS.
1443/KOLNP/2006 29-05-2006 253756 22-08-2012 QUINOLINES USEFUL IN TREATING CARDIOVASCULAR WYETH
DISEASE
637/KOLNP/2007 21-02-2007 253761 22-08-2012 "5-[3-(4-BENZYLOXYPHENYLTHIO)-FUR-2-YL]- QUEST PHARMACEUTICAL SERVICES
IMIDAZOLIDIN-2,4-DIONES (QPS)
2287/KOLNP/2006 10-08-2006 253771 23-08-2012 5,6-DIALKYL-7- AMINOTRIAZOLOPYRIMIDINES, THEIR BASF AKTIENGESELSCHAFT
PREPARATION AND COMPOSITIONS COMPRISING
THESE COMPOUNDS
461/MUMNP/2009 04-03-2009 253776 23-08-2012 KINASE INHIBITIRS USEFUL FOR THE TREATMENT OF DECIPHERA PHARMACEUTICALS LLC
PROLIFERATIVE DISEASES
2775/DELNP/2004 20-09-2004 253805 27-08-2012 "ORALLY ADMINISTRABLE COMPOSITION FOR THE SOCIETE DES PRODUITS NESTLE S.A
PHOTOPROTECTION OF THE SKIN"
2552/KOLNP/2007 09-07-2007 253821 28-08-2012 3, 5-DISUBSTITUTED AND 3,5,7-TRISUBSTITUTED-3H- ANADYS PHARMACEUTICALS, INC.
OXAZOLO AND 3H-THIAZOLO [4,5-D] PYRIMIDIN-2-ONE
COMPOUNDS AND PRODRUGS THEREOF

2595/DELNP/2006 09-05-2006 253825 28-08-2012 "N,2-DIMETHYL-{[7-(2-MORPHOLIN-4- PFIZER INC.


YLETHOXY)QUINOLIN-4-YL]OXY}-1-BENZOFURAN-3-
CARBOXAMIDE"
4841/DELNP/2007 22-06-2007 253890 30-08-2012 "TRANSDERMAL THERAPEUTIC SYSTEM (TTS), LTS LOHMANN THERAPIE-SYSTEME AG
COMPRISING A FIRST COMPARTMENT AND A SECOND
COMPARTMENT"
3059/CHENP/2006 22-08-2006 253897 31-08-2012 IMMUNOSUPPRESSANT COMPOUNDS IRM LLC
7158/DELNP/2007 17-09-2007 253900 31-08-2012 "BISHETEROCYCLE TANDEM COMPOUNDS USEFUL AS SHANGHAI INSTITUTE OF MATERIA
ANTIVIRAL AGENTS" MEDICA, CHINESE ACADEMY OF
SCIENCES
1892/DEL/2006 22-08-2006 253901 31-08-2012 "A NOVEL CYCLIC DONOR-ACCEPTOR COUNCIL OF SCIENTIFIC & INDUSTRIAL
CONJUGATE,PROCESS AND A SUPRAMOLECULAR RESEARCH
FLUORESCENT MARKER THEREOF"
3450/DEL/1997 01-12-1997 253903 31-08-2012 "1-ARYL-4-CYCLOPROPYLPYRAZOLE COMPOUNDS" PFIZER INC.,
1151/MUMNP/2009 16-06-2009 253922 03-09-2012 IMIDAZOLIDINONYL AMINOPYRIMIDINE COMPOUNDS ELI LILLY AND COMPANY
FOR THE TREATMENT OF CANCER
2485/KOLNP/2008 19-06-2008 253930 04-09-2012 3-(4-{[4-(4-{[3-(3,3-DIMETHYL-1-PIPERIDINYL) GLAXO GROUP LIMITED
PROPYL]0XY} PHENYL)-1-PIPERIDINYL] CARBONYL}-1-
NAPTHALENYL) PROPANOIC OR PROPENOIC ACID AS H1
AND H3 RECEPTOR ANTAGONISTS FOR THE TREATMENT
OF INFLAMMATORY AND/OR ALLERGIC DISORDERS

198/DEL/2008 24-01-2008 253942 05-09-2012 "A COMPOSITION COMPRISING METHYL N-(2,6- SYNGENTA PARTICIPATIONS AG
DIMETHYLPHENYL)-N-(METHOXYACETYL)-DL-
ALANINATE AND 3-ANILINO-5-METHYL-5-(4-
PHENOXYPHENYL)-1,3-OXAZOLIDINE-2,4-DIONE"
880/MUM/2004 13-08-2004 253950 06-09-2012 DISPERSIBLE SUSTAINED RELEASE PHARMACEUTICAL SINGH, KAMALINDER KAUR
COMPOSITIONS
4742/DELNP/2005 18-10-2005 253962 06-09-2012 "DELAYED RELEASE TABLET WITH DEFINED CORE JAGOTEC AG
GEOMETRY"
704/DEL/2005 30-03-2005 253965 07-09-2012 " ANTIFUNGAL STEROIDAL DIMERS, N1, N3- COUNCIL OF SCIENTIFIC & INDUSTRIAL
DIETHYLENETRIAMINE BIS [ CHOLIC ACID AMIDE] " RESEARCH
1020/CHENP/2008 29-02-2008 253968 07-09-2012 DIAMINOPYRIMIDINES AS P2X3 AND P3X2/3 F. HOFFMANN-LA ROCHE AG
MODULATORS
1195/DEL/2001 29-11-2001 253983 11-09-2012 AN ANTI BACTERIAL COMPOSITION COUNCIL OF SCIENTIFIC AND
INDUSTRIAL RESEARCH
2733/DELNP/2007 12-04-2007 253993 12-09-2012 "PYROZOLO (1,5-ALPHA), PYRIMIDINYL COMPOUND" SMITHKLINE BEECHAM (CORK) LIMITED

2115/DELNP/2006 19-04-2006 253996 12-09-2012 "NOVEL 17B HYDROSYSTEROID DEHYDROGENASE TYPE SOLVAY PHARMACEUTICALS GMBH
1 INHIBITORS"
3157/CHENP/2006 31-08-2006 254003 12-09-2012 IMIDAZO[1,2-C]PYRIMIDINYLACETIC ACID DERIVATIVES ACTIMIS PHARMACEUTICALS, INC.

674/KOLNP/2007 23-02-2007 254012 12-09-2012 NOVEL BENZO-FUSED HETEROARYL SULFAMIDE JANSSEN PHARMACEUTICA N.V.
DERIVATIVES USEFUL AS ANTICONVULSANT AGENTS
3767/DEL/1998 16-12-1998 254063 18-09-2012 "2,4-DUSULFONYL PHENYL BUTYL NITRONE" OKLAHOMA MEDICAL RESEARCH
FOUNDATION
2981/KOLNP/2006 16-10-2006 254073 18-09-2012 NOVEL COMPOUNDS AS OPIOID RECEPTOR JANSSEN PHARMACEUTICA N.V
MODULATORS
3074/KOLNP/2006 24-10-2006 254078 18-09-2012 TETRAHYDRO-INDAZOLE CANNABINO ID MODULATORS JANSSEN PHARMACEUTICA N.V.

2719/KOLNP/2007 23-07-2007 254080 18-09-2012 PEPTIDIC COMPOUNDS UNIVERSITY OF WOLLONGONG


1838/DELNP/2007 08-03-2007 254115 20-09-2012 "A COMPOUND 1-(4-BENZOYLPIPERAZIN-1-YL)-2-(4- BRISTOL-MYERS SQUIBB COMPANY
METHOXY-7-(3-METHYL-1H-1,2,4-TRIAZOL-1-YL)-1H-
PYRROLO[2,32-C]PYRIDIN-3-YL)ETHANE-1,2-DIONE"

3013/DEL/2005 10-11-2005 254119 21-09-2012 A NOVEL PYRROLO[2,1-C) [1,4]BENZODIAZEPINE COUNCIL OF SCIENTIFIC AND
HYBRIDS AND A PROCESS FOR PREPARATION THEREOF INDUSTRIAL RESEARCH

1162/DEL/1999 30-08-1999 254130 21-09-2012 "A PIPERAZINE OF THE FORMULA I" ASTRAZENECA UK LTD.,
42/MUMNP/2009 05-01-2009 254149 24-09-2012 IMPROVEMENTS RELATING TO PHARMACEUTICAL UNILEVER PLC
COMPOSITIONS
1568/MUM/2008 23-07-2008 254150 24-09-2012 NOVEL ANTICANCER HYDRAZINO DERIVATIVE OF INDIAN INSTITUTE OF TECHNOLOGY,
CURCUMIN AND PROCESS FOR PREPARATION THEREOF BOMBAY

5560/DELNP/2006 25-09-2006 254165 25-09-2012 "A PHARMACEUTICAL COMPOSITION FOR TREATING BRISTOL-MYERS SQUIBB COMPANY
HIV INFACTION"
2157/CHENP/2004 28-09-2004 254167 25-09-2012 5-SUBSTITUTED 1, 1-DIOXO-1,2,5-THIAZOLIDINE-3-ONE NOVARTIS AG
DERIVATIVES AS PTPASE IB INHIBITORS
4597/CHENP/2007 16-10-2007 254174 26-09-2012 SPIRO-OXINDOLE COMPOUNDS XENON PHARMACEUTICALS INC.
95/CHENP/2008 07-01-2008 254184 28-09-2012 A COMPOSITION FOR TOPICAL USE FIDIA FARMACEUTICI S.P.A
2225/CHENP/2006 21-06-2006 254201 01-10-2012 NOVEL THIAZOLIDIN-4-ONE DERIVATIVES ACTELION PHARMACEUTICALS LTD
706/MUM/2006 05-05-2006 254202 01-10-2012 NOVEL INTERMEDIATES, PROCESS FOR THEIR PIRAMAL HEALTHCARE LIMITED
PREPARATION AND PROCESS FOR THE PREPARATION
OF CoQ10 EMPLOYING THE SAID NOVEL
INTERMEDIATES
2788/DELNP/2008 03-04-2008 254214 03-10-2012 "5-(4-{[(2-FLUOROPHENYL)METHYL} PHENYL)- GLAXO GROUP LIMITED
PROLINAMIDE OF FORMULA (I) AND PROCESS OF
PREPARING THE SAME"
2892/KOLNP/2007 08-08-2007 254225 04-10-2012 HETEROCYCLYLAMIDE-SUBSTITUTED IMIDAZOLE AICURIS GMBH & CO. KG.
COMPOUNDS AND METHOD OF PREPARATION
THEREOF
757/DELNP/2006 15-02-2006 254229 04-10-2012 "LIQUID, AQUEOUS, PHARMACEUTICAL COMPOSITIONS NOVO NORDISK HEALTH CARE AG
OF FACTOR VII POLYPEPTIDES."
383/DEL/2006 13-02-2006 254250 09-10-2012 NOVEL BIS-PYRROLO[2,1-C][1,4] BENZODIAZEPINE- COUNCIL OF SCIENTIFIC AND
ANTHRAQUINONE CONJUGATES AND A PROCESS FOR INDUSTRIAL RESEARCH
THE PREPARATION THEREOF
3061/KOLNP/2006 23-10-2006 254255 10-10-2012 PROCESS AND INTERMEDIATE COMPOUNDS USEFUL IN REDX PHARMA LIMITED
THE PREPARATION OF STATINS, PARTICULARLY
ROSUVASTATIN
1725/CHENP/2006 17-05-2006 254261 10-10-2012 A PHARMACEUTICAL COMPOSITION COMPRISING A SANOFI PASTEUR
VACCINE ANTIGEN AND A PHOSPHORIC ESTER
DERIVATIVE OF PHOSPHATIDYLCHOLINE
6256/DELNP/2006 25-10-2006 254265 11-10-2012 "AN ADHESIVE PATCH FOR TREATMENT AND HUNTER-FLEMING LIMITED
COMPOSITION THEREOF"
1525/MUMNP/2007 24-09-2007 254285 17-10-2012 AN AQUEOUS DISINFECTANTS OR STERILANT SOLUTIONS BIOMED LLC
COMPOSITION
1030/KOLNP/2007 23-03-2007 254307 18-10-2012 BUTYLPHTHALIDE SELF-EMULSIFYING DRUG DELIVERY SHIJIAZHUANG PHARMA GROUP
SYSTEM, ITS PREPARATION METHOD AND APPLICATION ZHONGQI PHARMACEUTICAL
TECHNOLOGY (SHIJIAZHUANG) CO.,
LTD.
259/DELNP/2005 24-01-2005 254316 18-10-2012 BROADSPECTRUM 2-AMINO-BENZOTHIAZOLE TIBOTEC PHARMACEUTICALS LTD.
SULFONAMIDE HIV PROTEASE INHIBITORS"
6180/DELNP/2007 08-08-2007 254349 27-10-2012 "A SUBSTITUTED ECTEINASCIDIN COMPOUND" PHARMA MAR, S.A.
481/DELNP/2008 17-01-2008 254354 29-10-2012 "A COMPOUND, WHICH IS N-(3-FLUOROPHENYL)-1-[(4- GLAXO GROUP LIMITED
{[(-3S)-3-METHYL-1-
PIPERAZINYL]METHYL}PHENYL)ACETYL]-4-
PIPERIDINAMINE ANA PHARMACEUTICALLY
ACCEPTABLE SALT THEREOF"
5546/CHENP/2007 03-12-2007 254362 29-10-2012 A PHARMACEUTICAL FORMULATION FOR TREATING SCHERING CORPORATION
HCV INFECTION
2824/DELNP/2006 18-05-2006 254363 29-10-2012 "A TRIAZOLE COMPOUND OF FORMULA (I) AND PFIZER INC
COMPOSITION COMPRISING THE SAME"
529/DEL/2006 28-02-2006 254367 29-10-2012 "5-[2-(2,6,6,-TRIMENTHYL-CYCLOHEX-2-ENYL)- COUNCIL OF SCIENTIFIC & INDUSTRIAL
ENTHENYL]-ISOXAAZOLES" RESEARCH
977/CHE/2007 08-05-2007 254378 30-10-2012 A STABLE CONTROLLED RELEASE ORAL SOLID DOSAGE MEDREICH LIMITED
FORM COMPOSITION AND A PROCESS THEREOF

3715/DELNP/2007 18-05-2007 254427 02-11-2012 "A PHARMACEUTICAL COMPOSITION" ENDORECHERCHE, INC


7676/DELNP/2006 18-12-2006 254439 05-11-2012 HETEROCYCLE-SUBSTITUTED PYRROLIDINE AND GENENTECH, INC.
PIPERIDINE
2041/DELNP/2006 13-04-2006 254443 05-11-2012 "PELLETS CONTAINING VENLAFAXINE HYDROCHLORIDE" EGIS GYOGYSZERGYAR RT

3155/CHENP/2006 31-08-2006 254449 05-11-2012 HETEROARYL PIPERIDINE GLYCINE TRANSPORTER MERCK SHARP & DOHME CORP.
INHIBITORS
1565/MUM/2008 23-07-2008 254454 06-11-2012 STABLE INJECTABLE OIL-IN-WATER NANOEMULSION BHARAT SERUMS AND VACCINES LTD
3513/CHENP/2006 25-09-2006 254466 06-11-2012 PROGESTERONE RECEPTOR MODULATORS MSD Oss B.V.
2926/CHENP/2006 09-08-2006 254469 06-11-2012 COMPOUNDS AND COMPOSITIONS AS LXR IRM LLC
MODULATORS
2755/DEL/2005 13-10-2005 254474 07-11-2012 "A SUSTAINED RELEASE MONOTHILIC FORMULATION NATIONAL INSTITUTE OF
OF ROPINIROLE" PHARMACEUTICAL EDUCATION AND
RESEARCH
433/DELNP/2007 17-01-2007 254484 07-11-2012 "PYRIMIDINE DERIVATIVES" F. HOFFMANN-LA ROCHE AG
4535/DELNP/2006 04-08-2006 254505 09-11-2012 "A MICROEMULSION PREPARATION OF HIGH BIOAVAILABILITY INC
CONCENTRATION PROPOFOL FOR ANESTHETIC USES"

520/CHENP/2008 31-01-2008 254533 12-11-2012 ANTITUMORAL BIOCONJUGATES OF HYALURONIC ACID FIDIA FARMACEUTICI S.P.A
OR ITS DERIVATIVES
1623/DELNP/2006 24-03-2006 254541 15-11-2012 ISOTHIOCYANATE PRESERVATIVES AND METHODS OF THE PROCTER & GAMBLE COMPANY
THEIR USE
3149/DELNP/2007 26-04-2007 254551 17-11-2012 "ß-L-2'-DEOXY-NUCLEOSIDES FOR THE TREATMENT OF IDENIX (CAYMAN) LIMITED
HEPATITIS B"
3094/KOLNP/2006 25-10-2006 254567 20-11-2012 IMIDAZOLE COMPOUNDS. JANSSEN PHARMACEUTICA N.V.
1253/CHE/2006 19-07-2006 254572 20-11-2012 OXAZOLIDINONE DERIVATIVES ORCHID RESEARCH LABORATORIES LTD

1855/DELNP/2006 04-04-2006 254576 21-11-2012 "MORPHOLINE DERIVATIVES AS NOREPINEPHRINE ELI LILLY AND COMPANY LIMITED
REUPTAKE INHIBITORS"
5080/DELNP/2006 04-09-2006 254601 23-11-2012 NITROGENOUS FUSED-RING COMPOUND" KISSEI PHARMACEUTICAL CO., LTD.
2910/DELNP/2005 29-06-2005 254616 26-11-2012 "COMPOSITION HAVING ACTION PREVENTING OR SUNTORY HOLDINGS LIMITED.,
ALLEVIATING SYMPTOMS OR DISEASES DUE TO AGING
OF BLOOD VESSELS"
520/CHE/2005 02-05-2005 254638 29-11-2012 A PEPTIDE AND A METHOD THEREOF INDIAN INSTITUTE OF SCIENCE
4024/CHENP/2006 01-11-2006 254662 03-12-2012 A COMPOSITION FOR TREATING HYPERLIPAEMIA LUNAN PHARMACEUTICAL GROUP
CORPORATION
2300/CHENP/2006 23-06-2006 254675 05-12-2012 CONTROLLED-RELEASE PHARMACEUTICAL LEK PHARMACEUTICALS D.D.
FORMULATION
3843/DELNP/2004 03-12-2004 254678 05-12-2012 "A STABLE FENOFIBRATE COMPOSITION FOR ORAL ELAN PHARMA INTERNATIONAL, LTD
ADMINISTRATION"
2763/MAS/1998 09-12-1998 254706 07-12-2012 EPLERENONE COMPOSITIONS GD SEARLE & CO
5/CHE/2004 02-01-2004 254714 10-12-2012 "NOVEL INDENO [2,1A] INDENE AND ISOINDOLO [2,1-A] SUVEN LIFE SCIENCES LIMITED
INDOLES AS 5-HT 6 RECEPTORS
3601/KOLNP/2006 01-12-2006 254726 11-12-2012 AMIDO COMPOUNDS AND THEIR USE AS INCYTE CORPORATION
PHARMACEUTICALS
1424/CHENP/2008 24-03-2008 254730 12-12-2012 NOVEL PYRIDINE AND PYRIMIDINE COMPOUNDS EISAI R&D MANAGEMENT CO, LTD
372/MUMNP/2008 27-02-2008 254746 14-12-2012 NOVEL TRIAZOLE DERIVATIVES RECEPTORS AETERNA ZENTARIS GMBH
5303/DELNP/2006 13-09-2006 254758 14-12-2012 COMPOSITION COMPRISING AN HDAC INHIBITOR IN DSM IP ASSET B.V.
COMBINATION WITH A RETINOID
1350/KOLNP/2007 17-04-2007 254759 14-12-2012 HYDROXYBENZOATE SALT OF A METANICOTINE TARGACEPT, INC.
COMPOUND,PROCESS FOR ITS PREPARATION AND
COMPOSITION COMPRISING IT
1255/KOLNP/2006 12-05-2006 254788 18-12-2012 A TOCOPHEROL MODIFIED COMPOUND SONUS PHARMACEUTICALS, INC.
00558/DELNP/2003 16-04-2003 254813 21-12-2012 "CRYSTALLINE TIOTROPIUM BROMIDE MONOHYDRATE BOEHRINGER INGELHEIM PHARMA
AND PROCESS THEREOF " GMBH & CO. KG
3841/DELNP/2008 06-05-2008 254830 24-12-2012 "COMPOUNDS AS GLUCAGON RECEPTOR ELI LILLY AND COMPANY
ANTAGONISTS"
106/DELNP/2008 03-01-2008 254839 26-12-2012 "POLYMORPHIC FORMS OF RIFAXIMIN, PROCESSES FOR ALFA WASSERMANN S. P. A.
THEIR PRODUCTION AND USE THEREOF IN MEDICINAL
PREPARATIONS"
439/MUMNP/2007 26-03-2007 254845 26-12-2012 PRODRUGS CONTAINING NOVEL BIO-CLEAVABLE PIRAMAL ENTERPRISES LIMITED
LINKERS
4346/CHENP/2006 27-11-2006 254919 04-01-2013 BINDING MOLECULES CAPABLE OF NEUTRALIZING CRUCELL HOLLAND B.V
RABIES VIRUS
4727/CHENP/2006 22-12-2006 254921 04-01-2013 HETEROCYCLIC CARBOXAMIDES WITH MICROBIOCIDAL SYNGENTA PARTICIPATIONS AG
ACTIVITY
5185/CHENP/2007 16-11-2007 254930 07-01-2013 STREPTOGRAMINDERIVATIVES, THEIR PREPARATION AVENTIS PHARMA S.A
AND COMPOSITIONS WHICH CONTAIN THEM

5355/DELNP/2006 15-09-2006 254948 07-01-2013 A COMPOUND OF FORMULA I BRISTOL-MYERS SQUIBB COMPANY.


1046/CHENP/2006 27-03-2006 254955 08-01-2013 SUBSTITUTED THIENO [2,3-D] PYRIMIDINES AS HSP 90 M/S. VERNALIS (CAMBRIDGE) Ltd
INHIBITORS
1582/MUMNP/2008 25-07-2008 254957 09-01-2013 ACYLOXYALKYL CARBAMATE PRODUCTS, XENOPORT, INC.
1550/CHE/2006 29-08-2006 254994 11-01-2013 NOVEL DIPEPTIDYL PEPTIDASE IV INHIBITOR ORCHID CHEMICALS &amp;
PHARMACEUTICALS LTD
2064/DELNP/2004 19-07-2004 255028 16-01-2013 A CONTROLLED RELEASE PHARMACEUTICAL GLAXO GROUP LIMITED
FORMULATION
438/MUM/2008 03-03-2008 255029 16-01-2013 THIENO[2,3-D]-PYRIMIDINE-4(3H)-ONE COMPOUNDS NATIONAL CHEMICAL LABORATORY
AND PROCESS THEREOF
2163/MUMNP/2008 10-10-2008 255039 16-01-2013 COSMETIC COMPOSITION WITH SOFT FOCUS HINDUSTAN UNILEVER LIMITED
PROPERTIES
1589/KOLNP/2006 08-06-2006 255081 21-01-2013 AN ANTIBODY GLAXO GROUP LIMITED
5707/DELNP/2006 29-09-2006 255083 21-01-2013 COMPRESSED PHARMACEUTICAL COMPOSITIONS NORGINE B.V
COMPRISING PEG AND ELECTROLYTES
2046/DELNP/2003 12-02-2003 255111 23-01-2013 A PHARMACEUTICAL COMPOSITION FOR HF ARZNEIMITTELFORSCHUNG GMBH
PHARMACOLOGICAL ADDICTIVE SUBSTANCE OR
INTOXICANT THERAPY
1747/MUM/2006 20-10-2006 255115 23-01-2013 STABLE AEROSOL FORMULATION CIPLA LIMITED
4322/CHENP/2006 24-11-2006 255153 30-01-2013 THERAPEUTIC ENZYME FORMULATIONS AND USES THE BOARD OF TRUSTEES OF THE
THEREOF LELAND STANFORD JUNIOR UNIVERSITY

1276/CHENP/2008 14-03-2008 255154 30-01-2013 4-AMINO-THIENO[3,2-c]PYRIDINE-7-CARBOXYLIC ACID F. HOFFMANN-LA ROCHE AG


COMPOUNDS
1217/CHE/2006 12-07-2006 255172 31-01-2013 2-SUBSTITUTED METHYL PENAM DERIVATIVES ORCHID CHEMICALS &
PHARMACEUTICALS LTD
1904/DELNP/2005 05-05-2005 255194 01-02-2013 NOVEL BENZOXAZOCINES COMPOUNDS ARAKIS LTD
1607/DEL/1996 19-07-1996 255196 01-02-2013 A CONTROLLED RELEASE AND DELAYED RELEASE SMITHKLINE BEECHAM P.L.C.
FORMULATION
1514/DEL/1999 30-11-1999 255203 02-02-2013 FAST DISSOLVING PHARMACEUTICAL COMPOSITIONS IN PANACEA BIOTEC LIMITED
SOLID FORM WITH PROLONGED SWEET TASTE AND A
PROCESS FOR THE MANUFACTURE THEREOF

169/DELNP/2007 05-01-2007 255207 04-02-2013 SALTS OF BENZIMIDAZOLE DERIVATIVE EISAI R & D MANAGEMENT CO., LTD.
1726/KOLNP/2007 15-05-2007 255232 05-02-2013 PROCESS FOR PREPARING 4-(N-ALKYLAMINO)-5, 6- RAGACTIVES, S.L.
DIHYDRO-4H-THEINO-[2,3-B]-THIOPYRANS
3577/DELNP/2006 21-06-2006 255243 06-02-2013 A COMPOUND DENOTED 4-(((6-(3-((1S,1AR,7BR)-4,7- MEDIVIR AB.
DIFLUORO-1,1A,2,7B-
TETRAHYDROCYCLOPROPA[C]CHROMEN-1-
YL)UREIDO)PYRIDIN-3-YL)OXY)BENZENESULFONAMIDE

40/DEL/2006 04-01-2006 255262 07-02-2013 ORAL FORMULATIONS FOR ENAHANCING GASTRIC DIRECTOR GENERAL , DEFENCE
EMPTYING AND SPHINCTER RELAXATION INSTANTLY RESEARCH & DEVELOPMENT
AND A PROCESS OF PREPARTATION THEREOF ORGANISATION

2792/MUMNP/2008 30-12-2008 255273 08-02-2013 FLUOROALKYLOXYCOMBRETASTATIN DERIVATIVES, ZHEJIANG DADE PHARMACEUTICAL


METHODS FOR PRODUCING SAME GROUP CO. LTD.
1636/CHENP/2007 20-04-2007 255279 08-02-2013 (BIPHENYL)CARBOXYLIC ACIDS AND DERIVATIVES CELLZOME LIMITED
THEREOF
2725/DELNP/2006 16-05-2006 255287 09-02-2013 3- AMINOPYRROLIDONE DERIVATIVES NEWRON PHARMACEUTICALS S.p.A
6210/DELNP/2007 09-08-2007 255288 09-02-2013 A CYCLOHEPTA[B] PYRIDINE-3-CARBONYLGUANIDINE TOA EIYO LTD.
COMPOUND
7764/DELNP/2006 20-12-2006 255289 09-02-2013 PHARMACEUTICAL COMPOSITION COMPRISING A PFIZER PRODUCTS, INC
TABLET CORE OR CAPSULE FILL AND OPACIFYING COAT
AND POLISH COAT
3810/DELNP/2004 01-12-2004 255299 11-02-2013 COMPOSITION BASED ON SUBSTITUTED 1,3- GENFIT
DIPHENYLPROP-2-EN-1-ONE DERIVATIVES
3458/CHENP/2006 21-09-2006 255301 11-02-2013 INHIBITORS OF DIPEPTIDYLPEPTIDASE IV FOR TRUSTEES OF TUFTS COLLEGE
REGULATING GLUCOSE METABOLISM
592/KOLNP/2007 16-02-2007 255313 12-02-2013 A STAIN REMOVING ORAL COMPOSITION KRAFT FOODS GLOBAL BRANDS, LLC
1724/KOLNP/2007 15-05-2007 255543 01-03-2013 PYRAZOLO[1,5-A]PYRIMIDINES USEFUL AS INHIBITORS VERTEX PHARMACEUTICALS
OF PROTEIN KINASES INCORPORATED
17/MUM/2006 04-01-2006 255544 01-03-2013 PROCESS AND INTERMEDIATES FOR PREPARATION OF CIPLA LIMITED
DONEPEZIL HYDROCHLORIDE
4408/CHENP/2006 30-11-2006 255582 06-03-2013 3-AMINO-1-ARYLPROPYL INDOLES AS MONOAMINE F.HOFFMANN-LA ROCHE AG
REUPTAKE INHIBITOR
1733/CHE/2005 25-11-2005 255642 12-03-2013 SYNERGISTIC ANTIBACTERIAL COMPOSITION OF SRINIVAS JEGANNATHAN
CEFIXIME AND CLOXACILLIN / DICLOXACILLIN SODIUM
OR ANY OTHER OXACILLIN WITH CLAVULANIC ACID

533/DELNP/2007 19-01-2007 255673 14-03-2013 COMPOSITION COMPRISING ASPARTATE AND VITAMIN N.V. NUTRICIA
B12 OR BIOTIN FOR REGULATING KETONE BODIES

3141/DEL/2005 23-11-2005 255703 15-03-2013 A COMPOUND OF PROTECTED 4-AMINOMETHYLENE- LG LIFE SCIENCES LTD.
PYRROLIDIN-3-ONE
5661/DELNP/2007 23-07-2007 255745 20-03-2013 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY
750/KOLNP/2007 01-03-2007 255776 21-03-2013 4-(( PHENOXYALKYL)THIO) -PHENOXYACETIC ACIDS AND JANSSEN PHARMACEUTICA N.V.
ANALOGS
353/CHENP/2008 22-01-2008 255868 26-03-2013 AMPHOLYTIC COPOLYMER AND PRODUCTION THEREOF BASF AKTIENGESELLSCHAFT

119/KOLNP/2008 08-01-2008 255840 26-03-2013 SUBSTITUTED IMIDAZOLE COMPOUNDS AS KSP NOVARTIS AG


INHIBITORS
2353/CHENP/2008 12-05-2008 255979 12-04-2013 SUSTAINED RELEASE FILM FORMULATION FOR HEALING DAEWOONG CO., LTD
WOUND COMPRISING EPIDERMAL GROWTH FACTOR

4551/CHENP/2006 12-12-2006 255986 15-04-2013 SUBSTITUTED N-PHENYL BENZAMIDES PROTEOTECH INC.


7341/DELNP/2006 05-12-2006 255984 15-04-2013 "3-(HETEROARYL-OXY)-2-ALKYL-1-AZA-BICYCLOALKYL NOVARTIS AG,
DERIVATIVES AS ALPHA, 7-NACHR LIGANDS FOR THE
TREATMENT OF CNS DISEASES"
3035/DELNP/2007 23-04-2007 255996 17-04-2013 A COMPOUND 3'-{N'-[1-3,5-DIMETHYL-PHENYL)-6- LIGAND PHARMACEUTICALS,INC
TRIFLUOROMETHYL-2-OXO-1,2-DIHYDRO-INDOL-3-
YLIDENE]-HYDRAZINO}-2'-HYDROXY-BIPHENYL-3-
CARBOXYLIC ACID AND PHARMACEUTICALLY
ACCEPTABLE SALTS THEREOF, FOR MODULATING
THROMBOPOIETIN ACTIVITY
2461/DEL/2004 10-12-2004 256010 18-04-2013 "PHARMACEUTICAL COMPOSITION FOR IMPROVING COUNCIL OF SCIENTIFIC & INDUSTRIAL
PALATABILITY OF DRUGS AND PROCESS FOR RESEARCH
PREPARATION THEREOF"
1302/CHE/2005 15-09-2005 256019 19-04-2013 PYRIMIDINE CARBOXIMIDES ORCHID RESEARCH LABORATORIES LTD

26/DELNP/2008 01-01-2008 256021 19-04-2013 "HELIX 12 DIRECTED NON-STEROIDAL ENDORECHERCHE, INC.


ANTIANDROGENS"
1665/MUMNP/2008 04-08-2008 256023 22-04-2013 DEUTERATED CATECHOLAMINE DERIVATIVES AND BIRDS PHARMA GMBH BEROLINA
MEDICAMENTS COMPRISING SAID COMPOUNDS INNOVATIVE RESEARCH &
DEVELOPMENT SERVICES
5815/DELNP/2005 13-12-2005 256025 22-04-2013 "THIENOPYRIMIDINE DERIVATIVES AS POTASSIUM XENTION DISCOVERY LIMITED
CHANNEL INHIBITORS"
6550/DELNP/2007 23-08-2007 256032 22-04-2013 "OPTHALMOLOGIC COMPOSITIONS" LABORATOIRES THEA
4284/KOLNP/2007 07-11-2007 256041 23-04-2013 GLP-1 PEGYLATED COMPOUNDS ELI LILLY AND COMPANY
5224/DELNP/2006 11-09-2006 256046 24-04-2013 "COMPOUNDS USEFUL FOR INHIBITING MACROPHAGE CYTOKINE PHARMASCIENCES, INC.
MIGRATION INHIBITORY FACTOR"
1339/DEL/2005 25-05-2005 256052 26-04-2013 "A LIPOSOMAL FORMULATION AND USE THEREOF" COUNCIL OF SCIENTIFIC & INDUSTRIAL
RESEARCH
7052/DELNP/2006 23-11-2006 256066 29-04-2013 ANTIBODY DRUG CONJUGATES AND METHODS. GENENTECH, INC.
3073/DELNP/2004 07-10-2004 256069 29-04-2013 "NOVEL PYRAZOLO [4,3-D]PYRIMIDINES, PROCESSES USTAV EXPERIMENTALNI BOTANIKY AV
FOR THEIR PREPARATION AND METHODS FOR CR (INSTITUTE OF EXPERIMENTAL
THERAPY" BOTANY ACADEMY OF SCIENCES OF
THE CZECH REPUBLIC)
2449/DEL/2005 12-09-2005 256107 02-05-2013 "SUSTAINED RELEASE COMPOSITION" DELHI INSTITUTE OF PHARMACEUTICAL
SCIENCES & RESEARCH

32/KOLNP/2008 02-01-2008 256108 02-05-2013 N-(ARYLALKYL)-1H-PYRROLOPYRIDINE-2-CARBOXAMIDE SANOFI-AVENTIS


DERIVATIVES, PREPARATION AND THERAPEUTIC
COMPOSITION THEREOF
2192/DEL/2006 05-10-2006 256122 05-05-2013 A FORMULATION FOR THE STABILIZATION OF COUNCIL OF SCIENTIFIC & INDUSTRIAL
ALLERGENIC EXTRACTS USED IN DIAGNOSIS AND RESEARCH
THERAPY OF ALLERGY.
2335/DELNP/2007 26-03-2007 256125 06-05-2013 "NOVEL PYRAZOLE DERIVATIVE" KISSEI PHARMACEUTICAL CO.LTD.
2726/KOLNP/2007 24-07-2007 256132 07-05-2013 PROTEASOME INHIBITORS AND METHODS OF USING CEPHALON, INC
THE SAME
4247/CHENP/2006 17-11-2006 256182 13-05-2013 A MEDICAMENT COMPRISING GLYCOPYRROLATE AND NOVARTIS AG
(R)- 5-[2-(5,6-DIETHYL-INDAN-2-YLAMINO)-1-HYDROXY-
ETHYL]-8-HYDROXY-1H-QUINOLIN-2-ONE MALEATE

969/DELNP/2007 05-02-2007 256194 15-05-2013 "ORAL CARE COMPOSITION WITH CROSS-LINKED COLGATE-PAMOLIVE COMPANY
POLYMER PEROXIDE."
3232/DELNP/2006 05-06-2006 256230 20-05-2013 "A LIQUED PHARMACEUTICAL FORMULATION FOR THE FLAMEL TECHNOLOGIES
PROLONGED RELASE OF INTERLEUKIN(S)"
2324/DELNP/2004 10-08-2004 256262 24-05-2013 "INDOLAMID DERIVATIVES WHICH POSSESS ASTRAZENECA AB
GLYCOGENPHOSPHORYLASE INHIBITORY ACTIVITY"
1912/KOLNP/2007 28-05-2007 256282 29-05-2013 3-[2-(3-ACYLAMINO-2-OXO-2H-PYRIDIN-1-YL)- VERTEX PHARMACEUTICALS
ACETYLAMINO]-4-OXO-PENTANOIC ACID DERIVATIVES INCORPORATED
AS CASPASE INHIBITORS
1510/DELNP/2006 21-03-2006 256322 31-05-2013 "A CRTH2 ANTAGONIST OR PRODRUG THEREOF" OXAGEN LIMITED
1840/MUM/2007 20-09-2007 256350 05-06-2013 A NOVEL PHARMACEUTICAL COMPOSITION OF STATIN IPCA LABORATORIES LIMITED
WITH DMARDS
2813/DELNP/2008 04-04-2008 256396 11-06-2013 NOVEL HETEROBICYCLIC DERIVATIVES USEFUL AS F.HOFFMANN-LA ROCHE AG
INHIBITORS OF LIVER CARNITINE PALMITOYL
TRANSFERASE
4777/DELNP/2006 21-08-2006 256402 12-06-2013 "A PHARMACEUTICAL COMPOSITION AN INJECTION SMITHKLINE BEECHAM PLC
MOLDED CAPSULE SHELL, LINKER OR SPACER HAVING
SAID COMPOSITION"
577/MUM/2008 24-03-2008 256416 13-06-2013 MELT GRANULATED PHARMACEUTICAL COMPOSITIONS WOCKHARDT LTD
OF RHEIN OR DIACEREIN
9249/DELNP/2007 30-11-2007 256436 15-06-2013 "FK 228 DERIVATES AS HDAC INHIBITORS" UNIVERSITY OF SOUTHAMPTON
398/MUMNP/2009 20-02-2009 256458 19-06-2013 2-METHYLMORPHOLINE PYRIDO-, PYRAZO-AND KUDOS PHARMACEUTICALS LIMITED
PYRIMIDO-PYRIMIDINE DERIVATIVES AS MTOR
INHIBITORS
1718/KOLNP/2004 11-11-2004 256469 20-06-2013 NOVEL SUBSTITUTED SULFAMATE ANTICONVULSANT JANSSEN PHARMACEUTICAL N.V.
DERIVATIVES
1379/KOLNP/2006 23-05-2006 256470 20-06-2013 ALPHA-KETOAMIDE DERIVATIVE, AND PRODUCTION SENJU PHARMACEUTICAL CO., LTD.
METHOD AND USE THEREOF
1210/MUMNP/2010 07-06-2010 256475 21-06-2013 TRICYCLIC TRIAZOLIC COMPOUNDS LABORATORIOS DEL DR. ESTEVE S.A.
1200/CHENP/2007 22-03-2007 256485 24-06-2013 A FLUID COMPOSITION DOW GLOBAL TECHNOLOGIES , LLC
5460/DELNP/2007 16-07-2007 256481 24-06-2013 "ANTIBIOTIC 107891 AND PROCESS FOR PRODUCING Sentinella Pharmaceuticals, Inc.
THE SAME" ("Sentinella")
3973/KOLNP/2007 16-10-2007 256483 24-06-2013 ANTI-INFLAMMATORY AND/OR ANALGESIC ROQUETTE FRERES
COMPOSITION FOR THE INTESTINE COMPRISING
BRANCHED MALTODEXTRINS
2096/MUMNP/2009 10-11-2009 256516 27-06-2013 MONO-HYDROCHLORIC SALTS OF AN INHIBITOR OF JANSSEN PHARMACEUTICA NV
HISTONE DEACETYLASE.
668/DEL/2005 29-03-2005 256523 27-06-2013 "NOVEL POLYSACCHARIDES WITH ANTIOXIDANT NATIONAL INSTITUTE OF
PROPERTY" PHARMACEUTICAL EDUCATION AND
RESEARCH
7045/DELNP/2006 23-11-2006 256539 28-06-2013 "PHARMACEUTICAL COMPOSITIONS COMPRISING NOVARTIS AG.
POLYETHYLENE GLYCOL HAVING A MOLECULAR
WEIGHT OF LESS THAN 600 DALTONS"
158/DELNP/2007 05-01-2007 256614 08-07-2013 A PHARMACEUTICAL COMPOSITION COMPRISING MOKWALO SPF S.A.
STRONTIUM SALTS
1056/MUM/2009 22-04-2009 256607 08-07-2013 SOLUBILIZED BENZOYL PEROXIDE TOPICAL DRUG MODI PANKAJ
FORMULATION
3088/KOLNP/2007 22-08-2007 256627 09-07-2013 4-DEMETHYLPENCLOMEDINE COMPOUND, PROCESS SOUTHERN RESEARCH INSTITUTE
FOR ITS PREPARATION AND COMPOSITION
COMPRISING IT
3860/DELNP/2006 05-07-2006 256631 10-07-2013 "CYCLOPENTANYL CONTAINING MACROCYCLIC HCV NS- MEDIVIR AB.
3 PROTEASE INHIBITORS"
4401/CHENP/2006 30-11-2006 256658 12-07-2013 PYRIDIN-4-YL-ETHYNYL-IMIDAZOLES AND PYRAZOLES F. HOFFMANN-LA,ROCHE AG
AS MGLUR5 RECEPTOR ANTAGONISTS
7108/DELNP/2006 27-11-2006 256664 12-07-2013 ALKYL SUBSTITUTED INDOLOQUINOXALINES OXYPHARMA AB
452/MUMNP/2009 04-03-2009 256685 16-07-2013 AQUEOUS DISINFECTANTCOMPOSITION SOLUTIONS BIOMED LLC
2087/DELNP/2008 11-03-2008 256758 25-07-2013 CARBOXAMIDE DERIVATIVES AS MUSCARINIC PFIZER INC.
RECEPTOR ANTAGONISTS
3234/DELNP/2007 30-04-2007 256774 27-07-2013 "STABILISED OXYGEN RELEASING COMPOSITION" NGEN PHARMACEUTICALS N.V

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