120 Prototype Drugs Study Guide For Exam 3

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120 Study Guide for Exam 3 → Prototype Drugs

Chapter #14 Drugs For Seizures Anticonvulsants, Antiepileptics, Antiseizure meds, Hydantoins (sodium channel blockers), Succinimides
(calcium channel blockers)
T/Pg # Brand Generic Therapeutic Class Pharmacologic Class Sch
Barbiturate,
212 Luminal® phenobarbital Antiseizure, Sedative-Hypnotic C-IV
GABAA Receptor
Antiseizure,
Sedative-Hypnotic,
Benzodiazepine,
212 Valium® diazepam Anxiolytic, C-IV
GABA Receptor
Anesthetic Adjunct,
Skeletal Muscle Relaxant (Centrally Acting)
Hydantoin,
214 Dilantin® phenytoin Antiseizure, Antidysrhythmic
Sodium Influx Suppressing
Valproate,
Antiseizure,
Sodium Influx Suppressing,
215 Depakene® valproic acid Bipolar Disorder,
Calcium Influx Suppressing,
Migraine Prophylaxis
GABA Potentiating
Succinimide,
216 Zarontin® ethosuximide Antiseizure
Low-Threshold Calcium Channel Blocker
Per Elmore Vimpat® lacosamide Anticonvulsant C-V

Chapters 11 & 12(ADHD) CNS Stimulants & Drugs for Emotional, Mood & Behavioral Disorders
Antidepressants - SNRIs, SSRIs TCAs, MAOIs
Antipsychotics - Conventional/Traditional/Typical, Atypical/2 Gen, & - Dopamine-Serotonin System Stabilizers (DSSs) 3rd Gen
T/Pg # Brand Generic Therapeutic Class Pharmacologic Class Sch
146 Zoloft® sertraline Antidepressant SSRI
Tricyclic Antidepressant,
147 Tofranil® imipramine Antidepressant
5-HT & NE Reuptake Inhibitor
149 Nardil® phenelzine Antidepressant MAOI
CNS Stimulant, C-II
156 Ritalin® methylphenidate ADHD, Narcolepsy
NE & DA Releasing Agent
Pg. 153 Lithobid® Mania/Depressive Symptoms
lithium Monotherapy
ch12 ppt sl 39 Eskalith® Epilepsy/Psychosis
Conventional Antipsychotic, Phenothiazine
166 ® chlorpromazine
Schizophrenia Agent D2 Receptor Blocker
Conventional Antipsychotic, Nonphenothiazine,
168 Haldol® Haloperidol
Schizophrenia Agent D2 Receptor Blocker
Atypical Antipsychotic/2nd Gen
5-HT Receptor Antagonist,
171 Risperdal® risperidone Schizophrenia Agent,
DA Receptor Antagonist (weaker affinity)
Psychotic Depression Agent

Chapter #13 – Neurodegenerative Diseases -Drugs For Parkinson’s Disease, Alzheimer’s Disease, & Multiple Sclerosis
Dopaminergics, Anticholinergic , Antispasmodic, Centrally Acting Muscle Relaxants, Direct Acting (Peripheral) Skeletal Muscle Relaxants
T/Pg # Brand Generic Therapeutic Class Pharmacologic Class Sch.
Sinemet® carbidopa-levodopa Dopaminergic
184 Antiparkinson
Stalevo® carbidopa-levodopa-entacapone DA precursor
Antiparkinson
185 Cogentin® benztropine Used to relieve EPS Centrally Acting Cholinergic Receptor Blocker
-except Tardive Dyskinesia
186 Aricept® donepezil AD Acetylcholinerase Inhibitor
T 13.4 pg 187 Namenda® memantine AD NMDA Receptor Blocker
193 Flexeril® cyclobenzaprine Skeletal Muscle Relaxant (Centrally Acting) Catecholamine Reuptake Inhibitor
196 Dantrium® Dantrolene Skeletal Muscle Relaxant (Peripheral Acting) Skeletal Muscle Calcium Release Blocker

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