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Drugs Classification Pharmacology
Drugs Classification Pharmacology
Drugs Classification Pharmacology
1. Cholinergic drugs:
Direct acting Indirect acting agents
agents (Anticholinesterases:
Reversible Irreversible
Acetylcholine, Physostigmine, Parathion,
Arecholine, Neostigmine, Malathion,
Bethanechol. Pyridostigmine, Ecothiophate,
Carbachol, Edrophonium Tabun,
Muscarine, Sarin,
Pilocarpine Soman
2. Anticholinergic drugs:
a. Antimuscarinic drugs:
Atropine, Dicyclomine, Nortriptyline,
Biperiden. Diphenhydramine, Olanzapine,
Clomipramine, Doxepin, Scopolamine,
Clozapine, Imipramine, Trimipramine,
Desipramine, Meclizine
b. Antinicotinic agents:
Bupropion, Hexamethonium,
Dextromethorphan, Mecamylamine,
Doxacurium, Tubocurarine
4. Anti-Adrenergic drugs:
Alpha blockers Beta blockers
Nonequilibrium type: Nonselective (beta 1 and
Phenoxybenzamine. beta 2): Propranolol,
Equilibrium type Sotalol, Timolol, Pindolol,
(competitive): Labetalol, Carvedilol
A. Nonselective: Cardioselective (β1):
Ergotamine, Ergotoxine, Metoprolol, Atenolol,
Dihydroergotamine (DHE), Acebutolol, Bisoprolol,
Dihydroergotoxine,
6. Anticoagulants
Parenteral Anticoagulants: Heparin
Low Mol Wt Heparins: Enoxaparin, Dalteparin,
Tinzaparin, Nadoparin, Raviparin
Synthetic Heparin: Fondaparinux
Oral Anticoagulants
Dicumarol, Warfarin, Acenocumarol, Phenindione,
Anisindione
8. Antianginal drugs
2. Antidepressants
10. Opioids
Natural opium alkaloids: Morphine, Codeine
Semisynthetic: Diacetylmorphine (Heroin),
Pholcodeine, Ethylmorphine.
Synthetic: Pethidine, Fentanyl, Methadone,
Dextropropoxyphene, Tramadol.
11. NSAIDS
Nonselective Cox inhibitors: Aspirin, Indomethacin,
Sulindac, Ibuprofen, Naproxen, Ketoprofen, Mephenamic
acid, Diclofenac sodium, Piroxicam, Tenoxicam, Ketorolac
Preferential cox-2 inhibitor: Nimesulide, Meloxicam.
Selective cox- 2 inhibitors: Celecoxib,
Rofecoxib,Valdecoxib
Analgesics- Antipyretics: Paracetamol, Metamizol,
Nefopam (non opiod analgesic which donot inhibit PG
synthesis)
3. Classification of sulphonamides
4. Classification of Penicillins
5. Classification of Cephalosporins
First generation cephalosporins: Cefadroxil,
Cephalexin, Cefazolin, Cephradine.
Second generation cephalosporins: Cefaclor,
Cefuroxime, Cefotetan, Cefoxitin
Third generation cephalosporins: Cefixime,
Cefpodoxime, Ceftriaxone, Cefotaxime.
Fourth generation cephalosporins: Cefepime,
Cefluprenam, Cefozopran, Cefpirome.
Fifth generation cephalosporins: Ceftaroline,
Ceftobiprole
6. List of aminoglycosides
Streptomycin, Gentamicin, Sisomicin, Kanamycin ,
Tobramycin,
Amikacin, Neomycin, Soframycin
8. List of tetracyclines
Tetracycline, Oxytetracycline, Doxycycline, Minocycline
15. Antimalarials
4 aminoquinolines: – Chloroquine, Hydroxychloroquine,
Amodiaquine
8 aminoquinolines: – Primaquine, Tafenoquine, Bulaquine
Cinchona alkaloids: – Quinine, Quinidine
Quinoline methanol: Mefloquine
Biguanides – Proguanil, Chlorproguanil
Diaminopyrimidines Pyrimethamine
Sulfonamides – Sulfadoxine, dapsone
Tetracyclines: – tetracycline, doxycycline
1. Classify Autacoids
Amine autacoids: Histamine, 5-Hydroxytryptamine
(Serotonin)
Lipid derived autacoids: Prostaglandins, Leukotrienes,
Platelet activating factor
Peptide autacoids: Plasma kinins (Bradykinin, Kallidin),
Angiotensin
In addition, cytokines (interleukins, TNFα, GM-CSF,
etc.) and several peptides like gastrin, somatostatin,
vasoactive intestinal peptide and many others may be
considered as autacoids.
5. Antiemetics
Anticholinergic drug: Hyoscine, Dicyclomine
H1 Antihistaminics: Promethadine, Cinnarizine
Neuroleptics: Haloperidol,Chlorpromazine
Prokinetic drug: Domperidone,Cisapride, Mosapride,
Metochlopramide
5-HT3 Antagonist: Granisteron, Ondansteron
Adjuvant Antiemetics: Dexamethasone, Benzodiazepine,
Cannabinoids.
7. Nasal decongestants
Short-acting nasal decongestants
ephedrine
levmetamfetamine or L-desoxyephedrine
Naphazoline
Phenylephrine
Propylhexedrine
Long-acting decongestants (8 to 12 hours)
Xylometazoline, oxymetazoline
9. Progestins
1st generation: Norethindrone, Norethinodrel,
Lynestrenol
2nd generation: Norgestrel, Levonorgestrel
3rd generation: Desogestrel, Norgestimate, Gestodene
4th generation: Nomegestrol, Drospirenone
10. Bronchial asthma
A. BRONCHODILATORS
1. Selective β2- Agonists: Salbutamol, Terbutaline,
Remiterol, Fenoterol, Salmeterol, Formoterol, Bambuterol
2. Non-selective sympathomimetics: Epinephrine,
Ephedrine, Isoprenaline, Orciprenaline (Metaproterenol),
Isoetharine
3. Anticholinergics: Ipatropium, Tiotropium, Oxitropium
4. Methyl Xanthines: Theophylline, Aminophylline,
diprophylline.
1. Corticosteroids
A. Glucocorticoids:
a) Short acting (8-12 hours): Hydrocortisone, Cortisone
b) Intermediate acting (12-36 hours): Prednisolone,
Prednisone, Methyl Prednisolone, Triamcinolone
c) Long acting (36-72 hours): Betamethasone,
Dexamethasone
d) Local acting: Beclomethasone, Fluticasone, Budesonide
B. Mineralcorticoids: Aldosterone, Fludrocortisone,
Desoxycorticosterone acetate
3. Insulin types
A.Ultra-short acting insulins: Insulin lispro, Insulin
aspart & Insulin glulisine. Their action starts within 10- 20
min & lasts for 3-4 hrs.
B.Short acting insulins: These are Regular insulin,
Prompt Insulin-Zn Suspension or Semilente. Their effect
starts within 30 min & lasts for 5 – 8 hrs. These are soluble
crystalline Zn-Insulins made by recombinant DNA
techniques which are identical to human insulin.
C.Intermediate acting Insulins: These are NPH or
Isophane insulin & Lente Insulin. These have slower onset
(1-3 hrs) but longer duration of action (16-20 hrs).
D.Longer acting insulins: These are Ultralente & Insulin
Glargine. Ultralente is a cloudy Zn-suspension at neutral
pH in acetate buffer. It is usually combined with semilente
preparation & given s.c.
5. Anti-androgens
Steroid synthesis inhibitors: Ketoconazole
5-α reductase inhibitors: Finasteride and dutasteride
Androgen receptor inhibitors: Cyproterone and
cyproterone acetate, Flutamide, bicalutamide, enzalutamide
and nilutamide
Aldosterone Antagonist: Spironolactone
7. Diuretics
• Osmotic diuretics: mannitol (urea, glycerin, isosorbide)
• Carbonic anhydrase inhibitors: acetazolamide
(dichlorphenamide, metazolamide)
• Loop diuretics: furosemide, bumetanide, ethacrynic acid
• Thiazides, thiazide-like diuretics: (chlorothiazide),
hydrochlorothiazide, clopamide, indapamide, chlorthalidone
• Na+ channel antagonists: amiloride, triamterene
• Aldosterone antagonists: spironolactone, (canrenoate),
eplerenone
9. Antiinfluenza drugs
Amantadine, Rimantadine, Oseltamivir, Zanamivir
10. Cathartics/drastics/laxatives/purgatives
A According to b Osmotic
mechanism of action • Glycerin
(MOA) • Lactose
1 Stimulant/irritant • Mannitol
purgatives • Sorbitol
a Small gut: Castor oil, • Saline purgatives
Resins 3 Fecal softeners:
b Large gut: Bisacodyl, Docusate Na+,
Anthracene Lubricants (arachis oil,
2 Bulk-forming liquid paraffin)
purgatives 4 Miscellaneous
a Colloidal • Calomel
• Agar-agar • Colocynth
• Bran • Croton oil
• Calcium polycarbophil • Opioid receptor
• Frangula antagonist
• Isphagol husk • Parasympathomimetics
• Methyl-cellulose • Sulphur
• Malt soup extract • 5-HT4 receptor agonist
• Psyllium husk B According to site of
• Sterculia action