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Agonist Antagonist

α1 oxymetazoline, phenylephrine doxazosin, prazosin, tamsulosin,


terazosin
α2 brimonidine, clonidine, Idazoxan, mirtazapine, esmirtazapine,
dexmedetomidine lurasidone
β1 dobutamine, norepinephrine esmolol, metoprolol, atenolol,
dopamine (in high doses) carvedilol, nebivolol, bisoprolol,
β2 salbutamol/albuterol, terbutaline propranolol, nadolol, timolol, carvedilol
salmeterol, formoterol, indacaterol
β3 mirabegron

M1 bethanechol, pilocarpine atropine, scopolamine, ipratropium,


tiotropium, glycopyrrolate
M2
M3 solifenacin, trospium, darifenacin
M4
M5

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